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Bioorganic and Medicinal Chemistry Letters

Volumn 11, Issue 20, 2001, Pages 2759-2762

Potent second generation vinyl sulfonamide inhibitors of the trypanosomal cysteine protease cruzain

(7) Roush, William R a Cheng, Jianming a Knapp Reed, Beth a Alvarez Hernandez, Alejandro a McKerrow, James H b Hansell, Elizabeth b Engel, Juan C b

a UNIVERSITY OF MICHIGAN (United States)

b UNIVERSITY OF CALIFORNIA (United States)

Author keywords

[No Author keywords available]

Indexed keywords

CRUZIPAIN; CYSTEINE PROTEINASE; ENZYME INHIBITOR; N ALKOXYVINYLSULFONAMIDE INHIBITOR; N SULFONYL HYDROXYLAMINE DERIVATIVE; UNCLASSIFIED DRUG;

ANIMAL CELL; ARTICLE; CONTROLLED STUDY; DRUG ACTIVITY; DRUG EFFICACY; DRUG POTENCY; DRUG STRUCTURE; DRUG SYNTHESIS; ENZYME INHIBITION; MOUSE; NONHUMAN; TISSUE CULTURE; TRYPANOSOMA CRUZI; TRYPOMASTIGOTE;

ANIMALS; CYSTEINE ENDOPEPTIDASES; CYSTEINE PROTEINASE INHIBITORS; PARASITIC SENSITIVITY TESTS; PROTOZOAN PROTEINS; SULFONAMIDES; TRYPANOCIDAL AGENTS; TRYPANOSOMA CRUZI;

EID: 0035935182 PISSN: 0960894X EISSN: None Source Type: Journal
DOI: 10.1016/S0960-894X(01)00566-2 Document Type: Article

Times cited : (91)

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