SCOPUS 정보 검색 플랫폼

Bioorganic and Medicinal Chemistry Letters

Volumn 11, Issue 18, 2001, Pages 2555-2559

New leads for selective inhibitors of α-L-fucosidases. Synthesis and glycosidase inhibitory activities of [(2R,3S,4R)-3,4-dihydroxypyrrolidin-2-yl]furan derivatives

(6) Robina, Inmaculada a Moreno Vargas, Antonio J a Fernández Bolaos, José G a Fuentes, José a Demange, Raynald b Vogel, Pierre b

a UNIVERSITY OF SEVILLE (Spain)

b UNIVERSITY OF LAUSANNE (Switzerland)

Author keywords

[No Author keywords available]

Indexed keywords

5 (3,4 DIHYDROXYPYRROLIDIN 2 YL)FURAN DERIVATIVE; ALPHA GALACTOSIDASE; ALPHA LEVO FUCOSIDASE; ALPHA MANNOSIDASE; ALPHA N ACETYLGALACTOSAMINIDASE; BETA GALACTOSIDASE; BETA MANNOSIDASE; ENZYME INHIBITOR; GLUCAN 1,4 ALPHA GLUCOSIDASE; GLUCOSE; N ACETYL BETA GLUCOSAMINIDASE; PYRROLIDINE DERIVATIVE; UNCLASSIFIED DRUG;

ANIMAL TISSUE; ARTICLE; CATTLE; CHEMICAL REACTION; DRUG ACTIVITY; DRUG STRUCTURE; DRUG SYNTHESIS; ENZYME INHIBITION; EPIDIDYMIS; HUMAN; HUMAN TISSUE; NONHUMAN; PLACENTA; REACTION ANALYSIS; STRUCTURE ACTIVITY RELATION;

ALPHA-L-FUCOSIDASE; ANIMALS; CATTLE; DRUG DESIGN; DRUG EVALUATION, PRECLINICAL; ENZYME INHIBITORS; EPIDIDYMIS; FEMALE; FURANS; INHIBITORY CONCENTRATION 50; MALE; PLACENTA; PREGNANCY;

BOVINAE;

EID: 0035903835 PISSN: 0960894X EISSN: None Source Type: Journal
DOI: 10.1016/S0960-894X(01)00497-8 Document Type: Article

Times cited : (44)

References (57)

1
- 0023159808
- (1987) Annu. Rev. Biochem. , vol.56 , pp. 497
- Albein, A.D.¹

2
- 0001094662
- (1996) Chem. Rev. , vol.96 , pp. 683
- Dwek, R.A.¹

3
- 0034513388
- (2000) Chem. Rev. , vol.100 , pp. 4697
- Branza-Nichita, N.¹ Petrescu, A.J.² Negroin, G.³ Dwek, R.A.⁴ Petrescu, S.M.⁵

4
- 0003447494
- (1994) Nat. Prod. Rep. , pp. 35
- Hughs, A.B.¹ Rudge, A.J.²

5
- 0028874529
- (1995) Curr. Opin. Struct. Biol. , vol.5 , pp. 605
- Jacobs, G.S.¹

6
- 0033135747
- (1999) Bioessays , vol.21 , pp. 412
- Dennis, J.W.¹ Granovsky, M.² Warren, C.E.³

7
- 0029819131
- (1996) J. Virol. , vol.70 , pp. 7143
- Fischer, P.B.¹ Karlsson, G.B.² Butters, T.D.³ Dwek, R.A.⁴ Platt, F.M.⁵

8
- 0031058830
- (1997) Proc. Natl. Acad. Sci. U.S.A. , vol.94 , pp. 1822
- Mehta, A.¹ Lu, X.Y.² Block, J.M.³ Blumberg, B.S.⁴ Dwek, R.A.⁵

9
- 0031809225
- (1998) Nature Med. , vol.4 , pp. 610
- Block, T.M.¹ Lu, X.Y.² Mehta, A.S.³ Blumberg, B.S.⁴ Tennant, B.⁵ Ebling, M.⁶ Korba, B.⁷ Lansky, D.M.⁸ Jacob, G.S.⁹ Dwek, R.A.¹⁰

10
- 0032694353
- (1999) Proc. Natl. Acad. Sci. U.S.A. , vol.96 , pp. 11878
- Zitzmann, N.¹ Mehta, A.S.² Carrouee, S.³ Butters, T.D.⁴ Platt, F.M.⁵ McCauly, J.⁶ Blumberg, B.S.⁷ Dwek, R.A.⁸ Block, T.M.⁹

11
- 0030878261
- (1997) Clin. Cancer Res. , vol.3 , pp. 1077
- Goss, P.E.¹ Reid, C.L.² Bailey, D.³ Dennis, J.W.⁴

12
- 0025018353
- (1990) Cell , vol.63 , pp. 475
- Lowe, J.B.¹ Stoolman, L.M.² Nair, R.P.³ Larsen, R.D.⁴ Berhend, T.L.⁵ Marks, R.M.⁶

13
- 0025917249
- (1991) J. Biol. Chem. , vol.266 , pp. 14869
- Berg, E.L.¹ Robinson, M.K.² Mansson, O.³ Butcher, E.C.⁴ Magnani, J.L.⁵

14
- 0025799998
- (1991) J. Natl. Cancer Inst. , vol.83 , pp. 1321
- Lauri, D.¹ Needham, L.² Martin-Padura, I.³ Dejana, E.⁴

15
- 0023268507
- (1987) J. Cancer Res. , vol.47 , pp. 4634
- Niedbala, M.J.¹ Madiyalakan, R.² Matta, K.³ Crickard, K.⁴ Sharma, M.⁵ Bernacki, R.⁶

16
- 0025063976
- (1990) Biochem. J. , vol.265 , pp. 277
- Winchester, B.¹ Barker, C.² Baines, S.³ Jacob, G.S.⁴ Namgoong, S.K.⁵ Fleet, G.W.J.⁶

17
- 0031660015
- (1998) J. Androl. , vol.19 , pp. 444
- Veeramachaneni, D.N.R.¹ Smith, M.O.² Ellinwood, N.M.³

18
- 37049097621
- (1985) J. Chem. Soc., Chem. Commun. , pp. 841
- Fleet, G.W.J.¹ Shaw, A.N.² Evans, S.V.³ Fellows, L.E.⁴

19
- 0004267587
- (1999) Modern Drug Discovery , pp. 55
- Lipper, R.A.¹

20
- 0031024171
- (1997) Adv. Drug Delivery Rev. , vol.23 , pp. 3
- Lipinsky, C.A.¹ Lombardo, F.² Dominy, B.W.³ Feeney, P.J.⁴

21
- 84986661786
- (1990) Liebigs Ann. Chem. , pp. 953
- Paulsen, H.¹ Matzke, M.² Orthen, B.³ Nuck, R.⁴ Reutter, W.⁵

22
- 0029155704
- (1995) Carbohydr. Res. , vol.272 , pp. 17
- Legler, G.¹ Stütz, A.E.² Immich, H.³

23
- 0000419306
- (1997) Topics Curr. Chem. , vol.187 , pp. 157
- De Raadt, A.¹ Ekhart, C.W.² Ebner, M.³ Stütz, A.E.⁴

24
- 0003532642
- Stütz, A. E., Ed.; Wiley-VCH: Weinheim
- (1999) Iminosugars as Glycosidases Inhibitors, Nojirimycin and Beyond , pp. 254
- Ekhart, C.W.¹ Fechter, M.H.² Hadwiger, P.³ Mlaker, E.⁴ Stütz, A.E.⁵ Tauss, A.⁶ Wrodnigg, T.M.⁷

25
- 0032814101
- (1999) Helv. Chim. Acta , vol.82 , pp. 1044
- Peer, A.¹ Vasella, A.²

26
- 0026498495
- (1992) Tetrahedron , vol.48 , pp. 10191
- Bruce, I.¹ Fleet, G.W.J.² Cenci di Bello, I.³ Winchester, B.⁴

27
- 0028364924
- (1994) Tetrahedron Lett. , vol.35 , pp. 3845
- Schedler, D.J.A.¹ Bowen, B.R.² Ganem, B.³

28
- 0030822159
- (1997) J. Am. Chem. Soc. , vol.119 , pp. 8146
- Takayama, S.¹ Martin, R.² Wu, J.³ Laszlo, K.⁴ Siuzdak, G.⁵ Wong, C.-H.⁶

29
- 0034007669
- (2000) Bioorg. Med. Chem. , vol.8 , pp. 135
- McCort, I.¹ Fort, S.² Duréault, A.³ Depezay, J.-C.⁴

30
- 0033582974
- (1999) Tetrahedron Lett. , vol.40 , pp. 2351
- Nishimura, Y.¹ Shitara, E.² Takeuchi, T.³

31
- 0033997821
- (2000) Bioorg. Med. Chem. , vol.8 , pp. 343
- Shitara, E.¹ Nishimura, Y.² Kojima, F.³ Takechi, T.⁴

32
- 0034083484
- (2000) Eur. J. Org. Chem , pp. 2089
- Ogawa, S.¹ Sekura, R.² Maruyama, A.³ Yuasa, H.⁴ Hashimoto, H.⁵

33
- 0033802030
- (2000) Carbohydr. Lett. , vol.4 , pp. 13
- Ogawa, S.¹ Sekura, R.² Maruyama, A.³ Odagir, T.⁴ Yuasa, H.⁵ Hashimoto, H.⁶

34
- 0344712476
- (1997) Bioorg. Med. Chem. , vol.5 , pp. 519
- Le Merrer, Y.¹ Poitout, L.² Depezay, J.-C.³ Dosbâo, I.⁴ Geoffroy, S.⁵ Foglietti, M.-J.⁶

35
- 0029840739
- (1996) J. Am. Chem. Soc. , vol.118 , pp. 7647
- Moris-Varas, F.¹ Quiam, X.-H.² Wong, C.-H.³

36
- 0033621928
- (2000) Bioorg. Med. Chem. , vol.8 , pp. 307
- Le Merrer, Y.¹ Gauzy, L.² Gravier-Pelletier, C.³ Depezay, J.-C.⁴

37
- 0025167326
- (1990) Carbohydr. Chem. , vol.9 , pp. 683
- Hashimoto, H.¹ Fujimori, T.² Yuasa, H.J.³

38
- 0002354831
- (1996) Carbohydr. Lett. , vol.2 , pp. 23
- Yuasa, H.¹ Nakano, Y.² Hashimoto, H.³

39
- 0030972056
- (1997) J. Org. Chem. , vol.62 , pp. 992
- Isumi, M.¹ Tsuruta, O.² Harayama, S.³ Hashimoto, H.⁴

40
- 0028020315
- (1994) Tetrahedron: Asymmetry , vol.5 , pp. 2351
- Hashimoto, H.¹ Shimada, K.² Horito, S.³

41
- 0032542079
- (1998) Bioorg. Med. Chem. Lett. , vol.8 , pp. 3265
- Witczak, Z.¹ Boryczewski, D.²

42
- 0000094845
- (1999) Org. Lett. , vol.1 , pp. 775
- Leroy, E.¹ Reymond, J.-L.²

43
- 0034719245
- (2000) Org. Lett. , vol.2 , pp. 151
- Boss, O.¹ Leroy, E.² Blaser, A.³ Reymond, J.-L.⁴

44
- 0032894786
- (1999) Helv. Chim. Acta , vol.82 , pp. 760
- Blaser, A.¹ Reymond, J.-L.²

45
- 0034658825
- (2000) Org. Lett. , vol.2 , pp. 1733
- Blaser, A.¹ Reymond, J.-L.²

46
- 0028905327
- (1995) J. Org. Chem. , vol.60 , pp. 1492
- Wong, C.-H.¹ Provencher, L.² Porco J.A., Jr.³ Jung, S.-H.⁴ Wang, Y.-F.⁵ Chen, L.⁶ Wang, R.⁷ Steerisma, D.M.⁸

47
- 0033549740
- (1999) Angew. Chem. Int. Ed. , vol.38 , pp. 2300
- Sears, P.¹ Wang, C.-H.²

48
- 0033800019
- (2000) Synlett , pp. 1366
- Joubert, M.¹ Defoin, A.² Tarmus, C.³ Streith, J.⁴

49
- 33847276476
- (1984) J. Chem. Soc., Chem. Commun. , pp. 1240
- Fleet, G.W.J.¹ Smith, P.W.² Evans, S.V.³ Fellows, L.E.⁴

50
- 0032491895
- (1998) J. Chem. Soc., Chem. Commun. , pp. 119
- Kiess, F.-M.¹ Poggendorf, P.² Picasso, S.³ Jäger, V.⁴

51
- 0003744599
- unpublished
- Robina, I.¹ Carmona-Asenjo, A.T.² Moreno-Vargas, A.J.³ Demange, R.⁴ Vogel, P.⁵

52
- 0034635386
- (2000) Tetrahedron , vol.56 , pp. 971
- Sifferlen, T.¹ Defoin, A.² Streith, J.³ Le Nouen, D.⁴ Tarnus, C.⁵ Dosbâo, I.⁶ Foglietti, M.-J.⁷

53
- 39149116144
- (1956) Adv. Carbohydr. Chem. , vol.11 , pp. 97
- García-González, F.¹

54
- 0001136978
- (1972) Tetrahedron Lett. , pp. 4339
- Corey, E.J.¹ Kim, C.U.² Takeda, M.³

55
- 0003816228
- unpublished
- Moreno-Vargas, A.J.¹ Robina, I.²

56
- 0002515981
- (1994) Carbohydr. Lett. , vol.1 , pp. 1
- Picasso, S.¹ Chen, Y.² Vogel, P.³

57
- 0028866076
- (1995) J. Org. Chem. , vol.60 , pp. 6806
- Brandi, A.¹ Cicchi, S.² Cordero, F.M.³ Fignoli, B.⁴ Goti, A.⁵ Picasso, S.⁶ Vogel, P.⁷

* 이 정보는 Elsevier사의 SCOPUS DB에서 KISTI가 분석하여 추출한 것입니다.