Design, synthesis, and evaluation of novel A2A adenosine receptor agonists

Journal of Medicinal Chemistry

Volumn 44, Issue 4, 2001, Pages 531-539

  Rieger, J M ^a   Brown, M L ^a   Sullivan, G W ^b   Linden, J ^b   Macdonald, T L ^a  

^a UNIVERSITY OF VIRGINIA   (United States)

^b UNIVERSITY OF VIRGINIA   (United States)

Author keywords

[No Author keywords available]

Indexed keywords

2 [4 (2 CARBOXYETHYL)PHENETHYLAMINO]ADENOSINE 5' (N ETHYLCARBOXAMIDE); ADENOSINE RECEPTOR STIMULATING AGENT; ADENOSINE TRIPHOSPHATE; BRAIN RECEPTOR; GUANINE NUCLEOTIDE BINDING PROTEIN; LIGAND; PURINE RECEPTOR; RNA;

ANIMAL TISSUE; ARTICLE; BINDING AFFINITY; LIGAND BINDING; NONHUMAN; PHARMACOPHORE; PHYSICAL CHEMISTRY; RAT; RECEPTOR BINDING; STRUCTURE ACTIVITY RELATION; SYNTHESIS;

ALKYNES; ANIMALS; CEREBRAL CORTEX; COMBINATORIAL CHEMISTRY TECHNIQUES; CORPUS STRIATUM; CRYSTALLOGRAPHY, X-RAY; DRUG DESIGN; FURANS; LIGANDS; MODELS, MOLECULAR; PURINES; RADIOLIGAND ASSAY; RATS; RECEPTOR, ADENOSINE A2A; RECEPTORS, PURINERGIC P1; REGRESSION ANALYSIS; STRUCTURE-ACTIVITY RELATIONSHIP;

EID: 0035865778     PISSN: 00222623     EISSN: None     Source Type: Journal    
DOI: 10.1021/jm0003642     Document Type: Article

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