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Biochemistry

Volumn 40, Issue 32, 2001, Pages 9513-9521

Selection and characterization of a new class of peptide exosite inhibitors of coagulation factor VIIa

(4) Dennis, M S a Roberge, M a Quan, C a Lazarus, R A a

a GENENTECH INC (United States)

Author keywords

[No Author keywords available]

Indexed keywords

PEPTIDES;

BIOASSAY; CHEMICAL BONDS; COAGULATION; PROTEINS; TISSUE;

BIOCHEMISTRY;

A 100 Z; A 183; BLOOD CLOTTING FACTOR 10; BLOOD CLOTTING FACTOR 7A; BLOOD CLOTTING FACTOR 9; PEPTIDE A 100 Z; PEPTIDE A 183; PEPTIDE LIBRARY; PROTEIN INHIBITOR; SYNTHETIC PEPTIDE; UNCLASSIFIED DRUG;

ARTICLE; COMPETITIVE INHIBITION; ENZYME ACTIVE SITE; HUMAN; IC 50; INHIBITION KINETICS; PARTIAL THROMBOPLASTIN TIME; PEPTIDE ANALYSIS; PEPTIDE SYNTHESIS; PRIORITY JOURNAL; PROTEIN EXPRESSION; PROTEIN STRUCTURE; PROTHROMBIN TIME;

AMINO ACID SEQUENCE; BINDING SITES; BLOOD COAGULATION; DOSE-RESPONSE RELATIONSHIP, DRUG; FACTOR VIIA; HUMANS; KINETICS; MOLECULAR SEQUENCE DATA; PEPTIDE FRAGMENTS; PEPTIDE LIBRARY; PEPTIDES; PROTEASE INHIBITORS; PROTEIN BINDING; RECOMBINANT PROTEINS;

EID: 0035859911 PISSN: 00062960 EISSN: None Source Type: Journal
DOI: 10.1021/bi010591l Document Type: Article

Times cited : (41)

References (41)

1
- 0026337077
- (1991) Biochemistry , vol.30 , pp. 10363-10370
- Davie, E.W.¹ Fujikawa, K.² Kisiel, W.³

2
- 0032697618
- (1999) Thromb. Haemost. , vol.82 , pp. 165-174
- Mann, K.G.¹

3
- 0028932993
- (1995) Annu. Rev. Med. , vol.46 , pp. 103-112
- Broze G.J., Jr.¹

4
- 0029153045
- (1995) Thromb. Haemost. , vol.74 , pp. 7-17
- Rapaport, S.I.¹ Rao, L.V.M.²

5
- 0030666922
- (1997) Trends Cardiovasc. Med. , vol.7 , pp. 316-324
- Kirchhofer, D.¹ Banner, D.W.²

6
- 0032053072
- (1998) Int. J. Hematol. , vol.67 , pp. 229-241
- Higashi, S.¹ Iwanaga, S.²

7
- 0004257108
- (Uprichard, A. C. G., and Gallagher, K. P., Eds.), Springer-Verlag, Berlin
- (1999) Antithrombotics , pp. 1-39
- Leblond, L.¹ Winocour, P.D.²

8
- 0001612176
- (Uprichard, A. C. G., and Gallagher, K. P., Eds.), Springer-Verlag, Berlin
- (1999) Antithrombotics , pp. 421-445
- Gallagher, K.P.¹ Mertz, T.E.² Chi, L.³ Rubin, J.R.⁴ Uprichard, A.C.G.⁵

9
- 0026434005
- (1991) New Engl. J. Med. , vol.324 , pp. 1565-1574
- Hirsh, J.¹

10
- 0002776444
- (Colman, R. W., Hirsh, J., Marder, V. J., and Salzman, E. W., Eds.), J. B. Lippincott Company, Philadelphia
- (1994) Hemostasis and thrombosis: Basic principles and clinical practice , pp. 1567-1583
- Hirsh, J.¹ Ginsberg, J.S.² Marder, V.J.³

11
- 0030858230
- (1997) N. Engl. J. Med. , vol.337 , pp. 688-698
- Weitz, J.I.¹

12
- 24344446880
- (Uprichard, A. C. G., and Gallagher, K. P., Eds.), Springer-Verlag, Berlin
- (1999) Antithrombotics , pp. 447-476
- Esmon, C.T.¹

13
- 0031862826
- (1998) Coronary Artery Dis. , vol.9 , pp. 83-87
- Johnson, K.¹ Hung, D.²

14
- 0034628448
- (2000) J. Med. Chem. , vol.43 , pp. 305-341
- Leung, D.¹ Abbenante, G.² Fairlie, D.P.³

15
- 0021273620
- (1984) Science , vol.224 , pp. 350-357
- Neurath, H.¹

16
- 0030811924
- (1997) Thromb. Haemost. , vol.78 , pp. 501-511
- Bode, W.¹ Brandstetter, H.² Mather, T.³ Stubbs, M.T.⁴

17
- 0028914722
- (1995) Protein Sci. , vol.4 , pp. 337-360
- Perona, J.J.¹ Craik, C.S.²

18
- 0034665994
- (2000) Biochemistry , vol.275 , pp. 28826-28833
- Baugh, R.J.¹ Dickinson, C.D.² Ruf, W.³ Krishnaswamy, S.⁴

19
- 0034720739
- (2000) Biochemistry , vol.39 , pp. 7380-7387
- Kirchhofer, D.¹ Lipari, M.T.² Moran, P.³ Eigenbrot, C.⁴ Kelley, R.F.⁵

20
- 0034732235
- (2000) Nature , vol.404 , pp. 465-470
- Dennis, M.S.¹ Eigenbrot, C.² Skelton, N.J.³ Ultsch, M.H.⁴ Santell, L.⁵ Dwyer, M.A.⁶ O'Connell, M.P.⁷ Lazarus, R.A.⁸

21
- 0035859944
- (2001) Biochemistry , vol.40 , pp. 9522-9531
- Roberge, M.¹ Santell, L.² Dennis, M.S.³ Eigenbrot, C.⁴ Dwyer, M.A.⁵ Lazarus, R.A.⁶

22
- 0032560603
- (1998) Biochemistry , vol.37 , pp. 8870-8878
- Lowman, H.B.¹ Chen, Y.M.² Skelton, N.J.³ Mortensen, D.L.⁴ Tomlinson, E.E.⁵ Sadick, M.D.⁶ Robinson, I.C.A.F.⁷ Clark, R.G.⁸

23
- 0033731476
- (2000) Methods Enzymol. , vol.328 , pp. 333-363
- Sidhu, S.S.¹ Lowman, H.B.² Cunningham, B.C.³ Wells, J.A.⁴

24
- 0028243847
- (1994) J. Med. Chem. , vol.37 , pp. 1233-1251
- Gallop, M.A.¹ Barrett, R.W.² Dower, W.J.³ Fodor, S.P.A.⁴ Gordon, E.M.⁵

25
- 0023613953
- (1987) Methods Enzymol. , vol.154 , pp. 367-382
- Kunkel, T.A.¹ Roberts, J.D.² Zakour, R.A.³

26
- 0032806923
- (1999) Protein Sci. , vol.8 , pp. 1423-1431
- Starovasnik, M.A.¹ O'Connell, M.P.² Fairbrother, W.J.³ Kelley, R.F.⁴

27
- 0023270946
- (1987) Gene , vol.55 , pp. 189-196
- Chang, C.N.¹ Rey, M.² Bochner, B.³ Heyneker, H.⁴ Gray, G.⁵

28
- 0027465426
- (1993) Proteins: Struct., Funct., Genet. , vol.15 , pp. 312-321
- Dennis, M.S.¹ Carter, P.² Lazarus, R.A.³

29
- 0004249010
- Springer, Berlin
- (1984) Principles of Peptide Synthesis
- Bodansky, M.¹

30
- 0030917536
- (1997) Blood , vol.89 , pp. 3219-3227
- Kelley, R.F.¹ Refino, C.J.² O'Connell, M.P.³ Modi, N.⁴ Sehl, P.⁵ Lowe, D.⁶ Pater, C.⁷ Bunting, S.⁸

31
- 0032826356
- (1999) Thromb. Haemost. , vol.82 , pp. 1188-1195
- Refino, C.J.¹ Himber, J.² Burcklen, L.³ Moran, P.⁴ Peek, M.⁵ Suggett, S.⁶ Devaux, B.⁷ Kirchhofer, D.⁸

32
- 0033588095
- (1999) J. Biol. Chem. , vol.274 , pp. 24171-24175
- Shobe, J.¹ Dickinson, C.D.² Edgington, T.S.³ Ruf, W.⁴

33
- 0003518480
- John Wiley and Sons, Inc., New York
- (1975) Enzyme Kinetics
- Segel, I.H.¹

34
- 0031876832
- (1998) Drug Discovery Today , vol.3 , pp. 370-378
- Kay, B.K.¹ Kurakin, A.V.² Hyde-DeRuyscher, R.³

35
- 0034092470
- (2000) Chem. Biol. , vol.7 , pp. 17-25
- Hyde-DeRuyscher, R.¹ Paige, L.A.² Christensen, D.J.³ Hyde-DeRuyscher, N.⁴ Lim, N.⁵ Fredericks, Z.L.⁶ Kranz, J.⁷ Gallant, P.⁸ Zhang, J.⁹ Rocklage, S.M.¹⁰ Fowlkes, D.M.¹¹ Wendler, P.A.¹² Hamilton, P.T.¹³

36
- 0004342237
- US Patent No. 6090916
- (2000)
- Vlasuk, G.P.¹ Stanssens, P.E.H.² Messens, J.H.L.³ Lauwereys, M.J.⁴ LaRoche, Y.R.⁵ Jespers, L.S.⁶ Gansemans, Y.G.J.⁷ Moyle, M.⁸ Bergum, P.W.⁹

37
- 0000455702
- (1996) Proc. Natl. Acad. Sci. U.S.A. , vol.93 , pp. 2149-2154
- Stanssens, P.¹ Bergum, P.W.² Gansemans, Y.³ Jespers, L.⁴ Laroche, Y.⁵ Huang, S.⁶ Maki, S.⁷ Messens, J.⁸ Lauwereys, M.⁹ Cappello, M.¹⁰ Hotez, P.J.¹¹ Lasters, I.¹² Vlasuk, G.P.¹³

38
- 0033569932
- (1999) Eur. J. Biochem. , vol.265 , pp. 539-548
- Duggan, B.M.¹ Dyson, H.J.² Wright, P.E.³

39
- 0034941729
- (2001) Structure , vol.9 , pp. 627-636
- Eigenbrot, C.¹ Kirchhofer, D.² Dennis, M.S.³ Santell, L.⁴ Lazarus, R.A.⁵ Stamos, J.⁶ Ultsch, M.H.⁷

40
- 0032502818
- (1998) J. Mol. Biol. , vol.277 , pp. 959-971
- Dickinson, C.D.¹ Shobe, J.² Ruf, W.³

41
- 0027136111
- (1993) J. Mol. Biol. , vol.234 , pp. 564-578
- Lowman, H.B.¹ Wells, J.A.²

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