SCOPUS 정보 검색 플랫폼

Biochemistry

Volumn 40, Issue 45, 2001, Pages 13538-13547

Unexpected formation of an epoxide-derived multisubstrate adduct inhibitor on the active site of GAR transformylase

(7) Greasley, S E a Marsilje, T H a Cai, H a,b Baker, S c Benkovic, S J c Boger, D L a Wilson, I A a

a SCRIPPS RESEARCH INSTITUTE (United States)

b JOHNSON AND JOHNSON PHARMACEUTICAL RESEARCH AND DEVELOPMENT (United States)

c PENNSYLVANIA STATE UNIVERSITY (United States)

Author keywords

[No Author keywords available]

Indexed keywords

CELLULAR FOLATE TRANSPORT SYSTEMS;

BROMINE COMPOUNDS; CELLS; CRYSTAL STRUCTURE; ENZYME INHIBITION; ESCHERICHIA COLI; PHOSPHATES;

ENZYMES;

10 BROMO 10 BROMOMETHYL 5,8,10 TRIDEAZAFOLIC ACID; AZIRIDINE; BROMINE DERIVATIVE; ENZYME INHIBITOR; EPOXIDE; FOLIC ACID DERIVATIVE; MULTISUBSTRATE ADDUCT INHIBITOR; PHOSPHORIBOSYLGLYCINAMIDE FORMYLTRANSFERASE; PHOSPHORIBOSYLGLYCINAMIDE FORMYLTRANSFERASE INHIBITOR; UNCLASSIFIED DRUG;

ARTICLE; BIOAVAILABILITY; CELL TRANSPORT; CRYSTAL STRUCTURE; DENSITY; DRUG DESIGN; DRUG SYNTHESIS; ELECTRON; ENZYME ACTIVE SITE; ENZYME INHIBITION; ENZYME SUBSTRATE; ESCHERICHIA COLI; NONHUMAN; OPTICAL RESOLUTION; PRIORITY JOURNAL; REACTION ANALYSIS; TIME;

BINDING SITES; CRYSTALLIZATION; CRYSTALLOGRAPHY, X-RAY; ENZYME INHIBITORS; EPOXY COMPOUNDS; ESCHERICHIA COLI; HYDROXYMETHYL AND FORMYL TRANSFERASES; LIGANDS; MODELS, MOLECULAR; MOLECULAR CONFORMATION; PHOSPHORIBOSYLGLYCINAMIDE FORMYLTRANSFERASE; PROTEIN CONFORMATION;

ESCHERICHIA COLI; NEGIBACTERIA;

EID: 0035856543 PISSN: 00062960 EISSN: None Source Type: Journal
DOI: 10.1021/bi011482+ Document Type: Article

Times cited : (44)

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* 이 정보는 Elsevier사의 SCOPUS DB에서 KISTI가 분석하여 추출한 것입니다.