Major Photoaffinity Drug Binding Sites in Multidrug Resistance Protein 1 (MRP1) Are within Transmembrane Domains 10-11 and 16-17

Journal of Biological Chemistry

Volumn 276, Issue 15, 2001, Pages 12324-12330

  Daoud, Roni ^a   Julien, Michel ^a   Gros, Philippe ^a   Georges, Elias ^a  

^a MCGILL UNIVERSITY   (Canada)

Author keywords

[No Author keywords available]

Indexed keywords

AMINO ACIDS; CELL MEMBRANES; DRUG PRODUCTS; HYDROPHOBICITY; PROTEINS;

DRUG BINDING;

BIOCHEMISTRY;

ABC TRANSPORTER; EPITOPE; HEMAGGLUTININ; IODOAZIDORHODAMINE 123; MONOCLONAL ANTIBODY; MULTIDRUG RESISTANCE PROTEIN 1; N 2 HYDROXY 4 AZIDO 5 IODOPHENYLACETYLDIHYDRO 7 CHLORO 8 AMINOCINCHONAN 9 OL; NATURAL PRODUCT; RHODAMINE 123; UNCLASSIFIED DRUG; DRUG; MULTIDRUG RESISTANCE PROTEIN;

AMINO ACID SEQUENCE; ARTICLE; BINDING SITE; CONCENTRATION RESPONSE; CONTROLLED STUDY; DRUG BINDING; DRUG PROTEIN BINDING; DRUG TRANSPORT; HUMAN; HUMAN CELL; IMMUNOPRECIPITATION; MOLECULAR WEIGHT; MULTIDRUG RESISTANCE; PHOTOAFFINITY LABELING; PRIORITY JOURNAL; PROTEIN BINDING; PROTEIN DOMAIN; PROTEIN LOCALIZATION; PROTEIN MODIFICATION; PROTEIN STRUCTURE; STAPHYLOCOCCUS AUREUS; WILD TYPE; CHEMISTRY; HELA CELL; METABOLISM; MOLECULAR GENETICS; POLYACRYLAMIDE GEL ELECTROPHORESIS; WESTERN BLOTTING;

SIGANUS; STAPHYLOCOCCUS; STAPHYLOCOCCUS AUREUS;

AMINO ACID SEQUENCE; ATP-BINDING CASSETTE TRANSPORTERS; BINDING SITES; BLOTTING, WESTERN; ELECTROPHORESIS, POLYACRYLAMIDE GEL; HELA CELLS; HUMANS; MOLECULAR SEQUENCE DATA; MULTIDRUG RESISTANCE-ASSOCIATED PROTEINS; PHARMACEUTICAL PREPARATIONS; PHOTOAFFINITY LABELS;

EID: 0035853848     PISSN: 00219258     EISSN: None     Source Type: Journal    
DOI: 10.1074/jbc.M009782200     Document Type: Article

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