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Volumn 40, Issue 40, 2001, Pages 12039-12050
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Constitutive activation of the μ opioid receptor by mutation of d3.49(164), but not d3.32(147): D3.49(164) Is critical for stabilization of the inactive form of the receptor and for its expression
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Author keywords
[No Author keywords available]
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Indexed keywords
TRANSMEMBRANE DOMAIN;
AFLATOXINS;
AMINO ACIDS;
BINDING ENERGY;
COMPUTER SIMULATION;
MEMBRANES;
MUTAGENESIS;
17 METHYLNALOXONE;
DIPRENORPHINE;
ENKEPHALIN[2 DEXTRO ALANINE 4 METHYLPHENYLALANINE 5 GLYCINE];
G PROTEIN COUPLED RECEPTOR;
GUANINE NUCLEOTIDE BINDING PROTEIN;
GUANOSINE 5' O (3 THIOTRIPHOSPHATE);
GUANOSINE DIPHOSPHATE;
MONOCLONAL ANTIBODY;
MU OPIATE RECEPTOR;
MU OPIATE RECEPTOR AGONIST;
NALOXONE;
NALTREXONE;
PERTUSSIS TOXIN;
TRITIUM;
ANALGESIA;
ARTICLE;
BINDING AFFINITY;
CHO CELL;
DRUG RECEPTOR BINDING;
EMBRYO;
GENE EXPRESSION;
GENE MUTATION;
HUMAN;
HUMAN CELL;
KIDNEY CELL;
MOLECULAR MODEL;
NEUROPHARMACOLOGY;
PRIORITY JOURNAL;
AMINO ACID SEQUENCE;
ANIMALS;
CELL LINE;
CRICETINAE;
DIPRENORPHINE;
GUANOSINE 5'-O-(3-THIOTRIPHOSPHATE);
HUMANS;
HYDROGEN BONDING;
MOLECULAR SEQUENCE DATA;
MUTAGENESIS, SITE-DIRECTED;
PERTUSSIS TOXIN;
PROTEIN BINDING;
RATS;
RECEPTORS, OPIOID, MU;
SEQUENCE HOMOLOGY, AMINO ACID;
VIRULENCE FACTORS, BORDETELLA;
TRITIUM;
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EID: 0035834092
PISSN: 00062960
EISSN: None
Source Type: Journal
DOI: 10.1021/bi0100945 Document Type: Article |
Times cited : (66)
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References (61)
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