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Volumn 415, Issue 1, 2001, Pages 39-44

Characterisation of the effects of a non-peptide CGRP receptor antagonist in SK-N-MC cells and isolated human cerebral arteries

(9) Edvinsson, Lars a Sams, Anette b Jansen Olesen, Inger b Tajti, Janos c Kane, Stefanie A d Rutledge, Ruth Z d Koblan, Kenneth S d Hill, Raymond G e Longmore, Jenny e

a LUND UNIVERSITY HOSPITAL (Sweden)

b UNIVERSITY OF COPENHAGEN (Denmark)

c Department of Neurology and Pathology ^* (Hungary)

d MERCK RESEARCH LABORATORIES (United States)

e NEUROSCIENCE RESEARCH CENTRE (United Kingdom)

Author keywords

cAMP production; Cerebral vessel; CGRP receptor; Dilatation; Human

Indexed keywords

4 (2 OXO 2,3 DIHYDRO BENZOIMIDAZOL 1 YL) PIPERIDINE 1 CARBOSYLIC ACID [1 (3,5 DIBROMO 4 HYDROXY BENZYL)2 OXO 2 (4 PHENYL PIPERAZIN 1 YL)ETHYL AMIDE; AMIDE; CALCITONIN GENE RELATED PEPTIDE RECEPTOR; CYCLIC AMP; UNCLASSIFIED DRUG;

ANIMAL TISSUE; ARTICLE; BASILAR ARTERY; BRAIN ARTERY; BRAIN BLOOD VESSEL; CELL MEMBRANE; DRUG EFFECT; DRUG MECHANISM; DRUG STRUCTURE; GUINEA PIG; HUMAN; HUMAN TISSUE; MYOGRAPHY; NEUROBLASTOMA CELL; NONHUMAN; PRIORITY JOURNAL; RECEPTOR BINDING; VASODILATATION;

ANIMALS; BINDING, COMPETITIVE; CALCITONIN GENE-RELATED PEPTIDE; CELL MEMBRANE; CEREBRAL ARTERIES; CYCLIC AMP; DOSE-RESPONSE RELATIONSHIP, DRUG; GUINEA PIGS; HUMANS; PEPTIDE FRAGMENTS; PIPERAZINES; PIPERIDINES; RECEPTORS, CALCITONIN GENE-RELATED PEPTIDE; TUMOR CELLS, CULTURED; VASODILATION;

EID: 0035831167 PISSN: 00142999 EISSN: None Source Type: Journal
DOI: 10.1016/S0014-2999(00)00934-1 Document Type: Article

Times cited : (59)

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