-
1
-
-
0027241691
-
The synthesis of novel GABA uptake inhibitors. 1. Elucidation of the structure-activity studies leading to the choice of (R)-1-[4,4-Bis(3-methyl-2-thienyl)-3-butenyl]-3-piperidinecarboxylic acid (Tiagabine) as an anticonvulsant drug candidate
-
(1993)
J Med Chem
, vol.36
, pp. 1716-1725
-
-
Andersen, K.E.1
Braestrup, C.2
Gronwald, F.C.3
Jorgensen, A.S.4
Nielsen, E.B.5
Sonnewald, U.6
Sorensen, P.O.7
Suzdak, P.D.8
Knutsen, L.J.S.9
-
3
-
-
0001055353
-
Midbrain periaqueductal gray control of defensive behavior in the cat and the rat
-
Depaulis A, Bandler R, editors. The midbrain periaqueductal gray matter. Functional, anatomical and neurochemical organization. New York: Plenum Press
-
(1991)
, pp. 175-198
-
-
Bandler, R.1
Depaulis, A.2
-
5
-
-
0002007829
-
Emerging principles of organization of the midbrain periaqueductal gray matter
-
Depaulis A, Bandler R, editors. The midbrain periaqueductal gray matter. Functional, anatomical and neurochemical organization. New York: Plenum Press
-
(1991)
, pp. 1-8
-
-
Bandler, R.1
Carrive, P.2
Depaulis, A.3
-
10
-
-
0002119177
-
Localization of putative amino acid transmitters in the PAG and their relationship to the PAG-raphe magnus pathway
-
Depaulis A, Bandler R, editors. The midbrain periaqueductal gray matter. Functional, anatomical, and neurochemical organization. New York: Plenum Press
-
(1991)
, pp. 305-327
-
-
Beitz, A.J.1
Williams, F.G.2
-
15
-
-
0030272426
-
GABA transporter heterogeneity: Pharmacology and cellular localization
-
(1996)
Neurochem Int
, vol.29
, pp. 335-356
-
-
Borden, L.A.1
-
17
-
-
0028149954
-
Tiagabine, SK and F 89976-A, CI-966, and NCC-711 are selective for the cloned GABA transporter GAT-1
-
(1994)
Eur J Pharmacol
, vol.269
, pp. 219-224
-
-
Borden, L.A.1
Murali Dhar, T.G.2
Smith, K.E.3
Weinshank, R.L.4
Branchek, T.A.5
Gluchowski, C.6
-
19
-
-
0025068791
-
(R)-N-[4,4-bis(3-methyl-2-thienyl)but-3-en-1-yl]nipecotic acid binds with high affinity to the brain γ-aminobutyric acid uptake carrier
-
(1990)
J Neurochem
, vol.54
, pp. 639-647
-
-
Braestrup, C.1
Nielsen, E.B.2
Sonnewald, U.3
Knutsen, L.J.S.4
Andersen, K.E.5
Jansen, J.A.6
Frederiksen, K.7
Andersen, P.H.8
Mortensen, A.9
Suzdak, P.D.10
-
23
-
-
0030271375
-
Increased responsiveness and failure of habituation in neurons of the external nucleus of inferior colliculus associated with audiogenic seizures of the genetically epilepsy-prone rat
-
(1996)
Exp Neurol
, vol.141
, pp. 280-286
-
-
Chakravarty, D.N.1
Faingold, C.L.2
-
24
-
-
0030787936
-
Aberrant neuronal responsiveness in the genetically epilepsy-prone rat: Acoustic responses and influences of the central nucleus upon the external nucleus of the inferior colliculus
-
(1997)
Brain Res
, vol.761
, pp. 263-270
-
-
Chakravarty, D.N.1
Faingold, C.L.2
-
25
-
-
0027993991
-
Stable expression of a neuronal γ-aminobutyric acid transporter, GAT-3 in mammalian cells demonstrates unique pharmacological properties and ion dependence
-
(1994)
Mol Pharmacol
, vol.46
, pp. 550-557
-
-
Clark, J.A.1
Amara, S.G.2
-
27
-
-
0032557811
-
Neuronal and glial localization of GAT-1, a high-affinity γ-aminobutyric acid plasma membrane transporter, in human cerebral cortex: With a note on its distribution in monkey cortex
-
(1998)
J Comp Neurol
, vol.396
, pp. 51-63
-
-
Conti, F.1
Melone, M.2
De Biasi, S.3
Minelli, A.4
Brecha, N.C.5
Ducati, A.6
-
28
-
-
0033526902
-
Neuronal, glial, and epithelial localization of γ-aminobutyric acid transporter 2, a high-affinity γ-aminobutyric acid plasma membrane transporter, in the cerebral cortex and neighboring structures
-
(1999)
J Comp Neurol
, vol.409
, pp. 482-494
-
-
Conti, F.1
Vitellaro-Zuccarello, L.2
Barbaresi, P.3
Minelli, A.4
Brecha, N.C.5
Melone, M.6
-
32
-
-
0029294529
-
The ependyma: A protective barrier between brain and cerebrospinal fluid
-
(1995)
Glia
, vol.14
, pp. 1-13
-
-
Del Bigio, M.R.1
-
34
-
-
0022270903
-
γ-Aminobutyric acid uptake and termination of inhibitory synaptic potentials in the rat hippocampal slice
-
(1985)
J Physiol
, vol.366
, pp. 387-409
-
-
Dingledine, R.1
Korn, S.J.2
-
39
-
-
0026709603
-
The γ-aminobutyric acid (GABA) uptake inhibitor, tiagabine, increases extracellular brain levels of GABA in awake rats
-
(1992)
Eur J Pharmacol
, vol.220
, pp. 197-201
-
-
Fink-Jensen, A.1
Suzdak, P.D.2
Swedberg, M.D.B.3
Judge, M.E.4
Hansen, L.5
Nielsen, P.G.6
-
40
-
-
0025048435
-
Cloning and expression of a rat brain GABA transporter
-
(1990)
Science
, vol.249
, pp. 1303-1306
-
-
Guastella, J.1
Nelson, N.2
Nelson, H.3
Czyzyk, L.4
Keynan, S.5
Miedel, M.C.6
Davidson, N.7
Lester, H.A.8
Kanner, B.I.9
-
43
-
-
0019440458
-
Behavioural effects of GABA-agonists and antagonists infused in the mesencephalic reticular formation-deep layers of superior colliculus
-
(1981)
Brain Res
, vol.224
, pp. 185-194
-
-
Imperato, A.1
DiChiara, G.2
-
48
-
-
0002857597
-
Neurochemical study of PAG control of vocal behavior
-
Depaulis A, Bandler R, editors. The midbrain periaqueductal gray matter. Functional, anatomical, and neurochemical organization. New York: Plenum Press
-
(1991)
, pp. 11-21
-
-
Jurgens, U.1
-
53
-
-
0029789256
-
GAT-3, a high-affinity GABA plasma membrane transporter, is localized to astrocytic processes, and it is not confined to the vicinity of GABAergic synapses in the cerebral cortex
-
(1996)
J Neurosci
, vol.16
, pp. 6255-6264
-
-
Minelli, A.1
De Biasi, S.2
Brecha, N.C.3
Vitellaro-Zuccarello, L.4
Conti, F.5
-
54
-
-
0023035577
-
Evidence for GABA involvement in midbrain control of medullary neurons that modulate nociceptive transmission
-
(1986)
Brain Res
, vol.397
, pp. 37-46
-
-
Moreau, J.-L.1
Fields, H.L.2
-
55
-
-
0029164759
-
Pharmacological characterization of presynaptic and postsynaptic GABA(B) receptors in the deep nuclei of rat cerebellar slices
-
(1995)
Neuroscience
, vol.68
, pp. 1127-1137
-
-
Morishita, W.1
Sastry, B.R.2
-
57
-
-
0031889360
-
Periaqueductal gray neurons exhibit increased responsiveness associated with audiogenic seizures in the genetically epilepsy-prone rat
-
(1998)
Neuroscience
, vol.84
, pp. 619-625
-
-
N'Gouemo, P.1
Faingold, C.L.2
-
58
-
-
0032955375
-
The periaqueductal grey is a critical site in the neuronal network for audiogenic seizures: Modulation by GABA(A), NMDA and opioid receptors
-
(1999)
Epilepsy Res
, vol.35
, pp. 39-46
-
-
N'Gouemo, P.1
Faingold, C.L.2
-
60
-
-
0002939696
-
The neuroglial cells of the central nervous system
-
Pannese E, editor. Neurocytology. Fine structure of neurons, nerve processes, and neuroglial cells. New York: Thieme
-
(1994)
, pp. 156-189
-
-
Pannese, E.1
-
61
-
-
0002955958
-
The neuroglial cells
-
Peters A, Palay SL, Webster HDF, editors. The fine structure of the nervous system. Neurons and their supporting cells, 3rd ed. New York: Oxford University Press
-
(1991)
, pp. 273-311
-
-
Peters, A.1
Palay, S.L.2
Webster, H.D.F.3
-
63
-
-
0024565066
-
Two distinct mechanisms, differentially affected by excitatory amino acids, trigger GABA release from fetal mouse striatal neurons in primary culture
-
(1989)
J Neurosci
, vol.9
, pp. 648-656
-
-
Pin, J.-P.1
Bockaert, J.2
-
66
-
-
0000028220
-
GABAergic neuronal circuitry in the periaqueductal gray matter
-
Depaulis A, Bandler R, editors. The midbrain periaqueductal gray matter. Functional, anatomical, and neurochemical organization. New York: Plenum Press
-
(1991)
, pp. 329-344
-
-
Reichling, D.B.1
-
71
-
-
0020005029
-
Calcium-independent release of GABA from isolated horizontal cells of the toad retina
-
(1982)
J Physiol
, vol.323
, pp. 211-227
-
-
Schwartz, E.A.1
-
74
-
-
0020002312
-
A note on the use of picric acid-paraformaldehyde-glutaraldehyde fixative for correlated light and electron microscopic immunocytochemistry
-
(1982)
Neuroscience
, vol.7
, pp. 1779-1783
-
-
Somogyi, P.1
Takagi, H.2
-
78
-
-
0025049807
-
Ultrastructural morphometric analysis of GABA-immunoreactive terminals in the ventrocaudal periaqueductal grey: Analysis of the relationship of GABA terminals and the GABA(A) receptor to periaqueductal grey-raphe magnus projection neurons
-
(1990)
J Neurocytol
, vol.19
, pp. 686-696
-
-
Williams, F.G.1
Beitz, A.J.2
-
80
-
-
0032511829
-
Sodium and chloride-dependent high and low-affinity uptakes of GABA by brain capillary endothelial cells
-
(1998)
Brain Res
, vol.808
, pp. 1-7
-
-
Zhang, Y.1
Liu, G.-Q.2
-
81
-
-
0022346679
-
GABA uptake inhibitors produce a greater antinociceptive response in the mouse tail-immersion assay than other types of GABAergic drugs
-
(1985)
Life Sci
, vol.37
, pp. 1901-1912
-
-
Zorn, S.H.1
Enna, S.J.2
|