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Volumn 753, Issue 2, 2001, Pages 321-326
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High-throughput cytochrome P450 (CYP) inhibition screening via cassette probe-dosing strategy: II. Validation of a direct injection/on-line guard cartridge extraction-tandem mass spectrometry method for CYP2D6 inhibition assessment
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Author keywords
Cassette probe dosing; Cytochrome P450
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Indexed keywords
CARBON;
CYTOCHROME P450;
DEXTROMETHORPHAN;
DEXTRORPHAN;
DRUG METABOLITE;
FORMIC ACID;
PHENACETIN;
QUINIDINE;
ACCURACY;
ANALYTIC METHOD;
ARTICLE;
CENTRIFUGATION;
CONTROLLED STUDY;
ENZYME INHIBITION;
HUMAN;
IC 50;
LIVER MICROSOME;
PRIORITY JOURNAL;
SUPERNATANT;
TANDEM MASS SPECTROMETRY;
VALIDATION PROCESS;
CALIBRATION;
CYTOCHROME P-450 CYP2D6;
ENZYME INHIBITORS;
HUMANS;
MASS SPECTROMETRY;
MICROSOMES, LIVER;
MOLECULAR PROBES;
REPRODUCIBILITY OF RESULTS;
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EID: 0035810338
PISSN: 13872273
EISSN: None
Source Type: Journal
DOI: 10.1016/S0378-4347(00)00570-3 Document Type: Article |
Times cited : (16)
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References (11)
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