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Journal of Enzyme Inhibition

Volumn 16, Issue 5, 2001, Pages 401-416

Enantioselectivity of some 1-[(benzofuran-2-yl) phenylmethyl] imidazoles as aromatase (P450AROM) inhibitors

(4) Khodarahmi, G A a Laughton, C A a Smith, H J a Nicholls, P J a

a CARDIFF UNIVERSITY (United Kingdom)

Author keywords

Aromatase; Docking; Enantioselectivity; Inhibition; Modelling; P450AROM

Indexed keywords

1 [(BENZOFURAN 2 YL)(4' FLUOROPHENYL)METHYL] 1H IMIDAZOLE DIBENZOYL TARTRATE; 1 [(BENZOFURAN 2 YL)(4' METHYLPHENYL)METHYL] 1H IMIDAZOLE; 1 [(BENZOFURAN 2 YL)(4' METHYLPHENYL)METHYL] 1H IMIDAZOLE DIBENZOYL TARTRATE; 1 [(BENZOFURAN 2 YL)PHENYLMETHYL]IMIDAZOLE DERIVATIVE; AMINOGLUTETHIMIDE; AROMATASE INHIBITOR; FADRAZOLE; STEROID; UNCLASSIFIED DRUG;

ARTICLE; CHIRALITY; CONTROLLED STUDY; DRUG STRUCTURE; ENANTIOMER; ENZYME ACTIVE SITE; ENZYME ACTIVITY; ENZYME SUBSTRATE; HYDROPHOBICITY; IC 50; MOLECULAR MODEL; PRIORITY JOURNAL;

EID: 0035695774 PISSN: 87555093 EISSN: None Source Type: Journal
DOI: 10.1080/14756360109162389 Document Type: Article

Times cited : (8)

References (33)

1
- 0007883030
- "Design of Enzyme Inhibitors as Drugs"
- Sandler, M. and Smith, H.J., eds, (Oxford Science Publications, Oxford)
- (1994) , pp. 414-438
- Brodie, A.¹

2
- 0025778267
- (1991) Biochem. Soc. Trans. , vol.19 , pp. 456-459
- Kaye, B.¹

3
- 0028122470
- (1994) Chirality , vol.6 , pp. 400-404
- Pepper, C.J.¹ Smith, H.J.² Nicholls, P.J.³ Barrell, K.J.⁴ Hewlins, M.J.E.⁵

4
- 0018365924
- (1979) Endocrinology , vol.105 , pp. 52-57
- Graves, P.E.¹ Salhanick, H.A.²

5
- 0001934943
- "Design of Enzyme Inhibitors as Drugs"
- Sandler, M. and Smith, H.J., eds, (Oxford University Press, Oxford)
- (1994) , vol.2 , pp. 1-41
- Luscombe, D.K.¹ Tucker, M.² Pepper, C.J.³ Nicholls, P.J.⁴ Sandler, M.⁵ Smith, H.J.⁶

6
- 0031760523
- (1998) J. Pharm. Pharmacol. , vol.50 , pp. 1321-1330
- Khodarahmi, G.A.¹ Smith, H.J.² Nicholls, P.J.³ Ahmadi, M.⁴

7
- 0027255772
- (1993) J. Steroid Biochem. Mol. Biol. , vol.44 , pp. 675-676
- Whomsley, R.¹ Fernandez, E.² Nicholls, P.J.³ Smith, H.J.⁴ Lombardi, P.⁵ Pestillini, V.⁶

8
- 0027167698
- (1993) J. Med. Chem. , vol.36 , pp. 1393-1400
- Furet, P.¹ Batzl, C.² Bhatnager, A.S.³ Francotte, E.⁴ Rihs, G.⁵ Lang, M.⁶

9
- 0027175244
- (1993) J. Steroid Biochem. Mol. Biol. , vol.44 , pp. 399-407
- Laughton, C.A.¹ Zvelebil, M.J.J.M.² Neidel, S.³

10
- 0023905437
- (1988) Eur. J. Med. Chem. , vol.23 , pp. 203-206
- Pestillini, V.¹ Giolitti, A.² Pasqui, F.³ Abelli, L.⁴ Cutrufo, C.⁵

11
- 0023278237
- (1987) Chemioterapia , vol.6 , pp. 269-271
- Pestillini, V.¹ Gianotti, A.² Giolitti, A.³ Fanto, N.⁴ Riviera, L.⁵ Bellotti, M.G.⁶

12
- 0016272566
- (1974) J. Biol. Chem. , vol.249 , pp. 5373-5378
- Thompson, E.A.¹ Siiteri, P.K.²

13
- 85037294813
- AMBER 4.0 (University of California, San Francisco)
- (1991)
- Pearlman, A.D.¹ Case, D.A.² Caldwell, J.C.³ Seibel, G.L.⁴ Chandra Singh, U.⁵ Weiner, P.⁶ Kollman, P.A.⁷

14
- 0023977089
- (1988) J. Mol. Graphics , vol.6 , pp. 13-27
- Ferrin, T.E.¹ Haung, C.C.² Jarvis, L.E.³ Langridge, R.⁴

15
- 85037297958
- Mopac 6.0 (QCPE), available from the Quantum Chemistry Programme Exchange, Indiana University, Bloomington, IN
- Stewart, J.P.P.¹

16
- 0028100793
- (1994) J. Biol. Chem. , vol.269 , pp. 19501-19508
- Zhou, D.J.¹ Cam, L.L.² Laughton, C.A.³ Korzekwa, K.R.⁴ Chen, S.⁵

17
- 0030013560
- (1996) Cancer Res. , vol.56 , pp. 3451-3460
- Kao, Y.C.¹ Cam, L.L.² Laughton, C.A.³ Zhou, D.J.⁴ Chen, S.A.⁵

18
- 0033970047
- (2000) Mol. Cell. , vol.5 , pp. 121
- Williams, P.A.¹ Cosme, J.² Sridhar, V.³ Johnson, E.F.⁴ McRee, D.E.⁵

19
- 0022273620
- (1985) J. Biol. Chem. , vol.260 , pp. 16122-16130
- Poulos, T.L.¹ Finzel, B.C.² Gunsalus, I.C.³ Wagner, G.C.⁴ Kraut, J.⁵

20
- 0023583624
- (1987) Biochemistry , vol.26 , pp. 8165-8174
- Poulos, T.L.¹ Howard, A.J.²

21
- 0027326717
- (1993) Science , vol.261 , pp. 731-736
- Ravichandran, K.G.¹ Boddupalli, S.S.² Hasemann, C.A.³ Peterson, J.A.⁴ Deisenhofer, J.⁵

22
- 0028267490
- (1994) J. Mol. Biol. , vol.236 , pp. 1169-1185
- Hasemann, C.A.¹ Ravichandran, K.G.² Peterson, J.A.³ Deisenhofer, J.⁴

23
- 0029586252
- (1995) Struct. Biol. , vol.2 , pp. 144-153
- Cupp-Vickery, J.R.¹ Poulos, T.L.²

24
- 0023691843
- (1988) Biochem. Biophys. Res. Commun. , vol.156 , pp. 725-732
- Harada, N.¹

25
- 0006656956
- (1988) Natl. Acad. Sci. USA , vol.85 , pp. 8948-8952
- Corbin, C.J.¹ Graham-Lorence, S.² McPhaul, M.³ Mason, J.I.⁴ Mendelson, C.R.⁵ Simpson, E.R.⁶

26
- 0024506487
- (1989) FEBS Lett. , vol.247 , pp. 371-376
- Toda, K.¹ Teashima, M.² Mitsuuchi, Y.³ Yamasaki, Y.⁴ Yokoyama, Y.⁵ Najima, S.⁶

27
- 0024424777
- (1989) Mol. Endocrinol. , vol.3 , pp. 1477-1487
- Pompon, D.¹ Liu, R.Y.K.² Besman, M.J.³ Wang, P.L.⁴ Shively, J.E.⁵ Chen, S.⁶

28
- 0025965047
- (1991) Proc. Natl. Acad. Sci. USA , vol.88 , pp. 410-414
- Zhou, D.¹ Pompon, D.² Chen, S.³

29
- 0026558679
- (1992) J. Biol. Chem. , vol.267 , pp. 762-768
- Zhou, D.¹ Korzekw, K.R.² Bulos, T.³ Chen, S.⁴

30
- 0028100793
- (1994) J. Biol. Chem. , vol.269 , pp. 19501-19508
- Zhou, D.¹ Cam, L.² Laughton, C.A.³ Korzekw, K.R.⁴ Chen, S.⁵

31
- 0029056146
- (1995) J. Steroid Biochem. Mol. Biol. , vol.53 , pp. 191-197
- Koymans, L.M.H.¹ Moereels, H.² Vanden Bossche, H.³

32
- 85037303315
- unpublished work
- Kao, Y.C.¹ Cam, L.L.² Laughton, C.A.³ Zhou, D.⁴ Chen, S.⁵

33
- 85037295508
- private communication
- Whomsley, R.¹

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