Further characterization of β3-adrenoceptors in the guinea pig gastric fundus: Stereoselectivity, β-adrenoceptor alkylation, and structure-activity relationship

Canadian Journal of Physiology and Pharmacology

Volumn 79, Issue 12, 2001, Pages 985-995

  Horinouchi, Takahiro ^a   Koike, Katsuo ^a  

^a TOHO UNIVERSITY   (Japan)

Author keywords

3 adrenoceptor, stereoselectivity, adrenoceptor alkylating, structure activity relationship, guinea pig gastric fundus

Indexed keywords

4 (3 TERT BUTYLAMINO 2 HYDROXYPROPOXY) 2 BENZIMIDAZOLONE; 4 [2 [[2 (3 CHLOROPHENYL) 2 HYDROXYETHYL]AMINO]PROPYL]PHENOXYACETIC ACID; ADRENALIN; ALKYLATING AGENT; BETA 1 ADRENERGIC RECEPTOR; BETA 2 ADRENERGIC RECEPTOR; BETA 3 ADRENERGIC RECEPTOR; BETA 3 ADRENERGIC RECEPTOR STIMULATING AGENT; CATECHOLAMINE; DOBUTAMINE; DOPAMINE; HYDROXYL GROUP; ISOPRENALINE; NADOLOL; NORADRENALIN; PHENYLEPHRINE; BETA ADRENERGIC RECEPTOR STIMULATING AGENT; DRUG DERIVATIVE; PINDOBIND; PINDOLOL; SEROTONIN ANTAGONIST;

ALKYLATION; ANIMAL EXPERIMENT; ANIMAL TISSUE; ARTICLE; CONCENTRATION RESPONSE; CONTROLLED STUDY; DRUG SELECTIVITY; GUINEA PIG; HEART ATRIUM; ISOMER; MALE; NONHUMAN; PRIORITY JOURNAL; PROTEIN ANALYSIS; RECEPTOR BLOCKING; STEREOCHEMISTRY; STOMACH FUNDUS; STRUCTURE ACTIVITY RELATION; TRACHEA; ANIMAL; IN VITRO STUDY; METABOLISM; STEREOISOMERISM; STOMACH;

ADRENERGIC BETA-AGONISTS; ALKYLATION; ANIMALS; GASTRIC FUNDUS; GUINEA PIGS; MALE; PINDOLOL; RECEPTORS, ADRENERGIC, BETA-3; SEROTONIN ANTAGONISTS; STEREOISOMERISM; STOMACH; STRUCTURE-ACTIVITY RELATIONSHIP;

EID: 0035544769     PISSN: 00084212     EISSN: None     Source Type: Journal    
DOI: 10.1139/cjpp-79-12-985     Document Type: Article

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