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Journal of Organic Chemistry

Volumn 66, Issue 11, 2001, Pages 3797-3805

Synthesis of oxa-bridged analogues of farnesyltransferase inhibitor RPR 115135

(3) Martin, C a Mailliet, P b Maddaluno, J a

a UNIVERSITÉ DE ROUEN (France)

b SANOFI (France)

Author keywords

[No Author keywords available]

Indexed keywords

STEREOSELECTIVITY;

CONDENSATION; OXIDATION; OXYGEN; SYNTHESIS (CHEMICAL);

REACTION KINETICS;

ACRYLIC ACID DERIVATIVE; ACRYLIC ACID METHYL ESTER; ALPHA PHENYLSELENOACRYLATE; BENZOFURAN DERIVATIVE; PHENYLISOBENZOFURAN; PROTEIN FARNESYLTRANSFERASE INHIBITOR; PYRROLIDINE DERIVATIVE; PYRROLINE DERIVATIVE; RPR 115135; RPR 222490; RPR 225370; UNCLASSIFIED DRUG;

ARTICLE; CHEMICAL MODIFICATION; CHEMICAL REACTION; DRUG ACTIVITY; DRUG MECHANISM; DRUG STRUCTURE; DRUG SYNTHESIS; ENZYME INHIBITION; OXIDATION; POLYMERIZATION; PROTON TRANSPORT; REACTION ANALYSIS; STEREOCHEMISTRY; STRUCTURE ACTIVITY RELATION;

ALKYL AND ARYL TRANSFERASES; BRIDGED COMPOUNDS; CYCLIZATION; ENZYME INHIBITORS; FARNESYLTRANSTRANSFERASE; INDICATORS AND REAGENTS; INDOLES; MAGNETIC RESONANCE SPECTROSCOPY; X-RAY DIFFRACTION;

EID: 0035356379 PISSN: 00223263 EISSN: None Source Type: Journal
DOI: 10.1021/jo0100188 Document Type: Article

Times cited : (32)

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