SCOPUS 정보 검색 플랫폼

Volumn 54, Issue 2, 2001, Pages 227-239

Synthesis and biological evaluation of two new radiolabelled estrogens: [125I](E)-3-methoxy-17α-iodovinylestra-1,3,5(10),6-tetraen-17β-ol and [125I](Z)-3-methoxy-17α-iodovinylestra-1,3,5(10),6-tetraen-17β-ol

(7) Melo e Silva, M Cristina a Patrício, Luciana a Gano, Lurdes a Sa e Melo M Luisa b Inohae, Eiko c Mataka, Shuntaro c Thiemann, Thies c

a INSTITUTO TECNOLÓGICO E NUCLEAR (Portugal)

b UNIVERSITY OF COIMBRA (Portugal)

c KYUSHU UNIVERSITY (Japan)

Author keywords

[No Author keywords available]

Indexed keywords

CHEMICAL BONDS; ISOMERS; SYNTHESIS (CHEMICAL); TISSUE;

RADIOLABELLED ESTROGEN;

HORMONES;

17ALPHA (2 IODOVINYL) 3 METHOXYESTRA 1,3,5(10),6 TETRAEN 17BETA OL; ESTROGEN; ESTROGEN RECEPTOR; IODINE 125; RADIOPHARMACEUTICAL AGENT; UNCLASSIFIED DRUG;

ANIMAL EXPERIMENT; ARTICLE; DRUG DISTRIBUTION; DRUG RECEPTOR BINDING; DRUG SYNTHESIS; ENANTIOMER; FEMALE; IN VITRO STUDY; INFRARED SPECTROPHOTOMETRY; ISOTOPE LABELING; MASS SPECTROMETRY; MOUSE; NONHUMAN; NUCLEAR MAGNETIC RESONANCE; PRIORITY JOURNAL;

ANIMALS; BREAST NEOPLASMS; ESTRADIOL; ESTRADIOL CONGENERS; FEMALE; HUMANS; IODINE RADIOISOTOPES; MICE; RECEPTORS, ESTROGEN; STEREOISOMERISM; TISSUE DISTRIBUTION; UTERUS;

EID: 0035255412 PISSN: 09698043 EISSN: None Source Type: Journal
DOI: 10.1016/S0969-8043(99)00258-4 Document Type: Article

Times cited : (44)

References (18)

1
- 0023740588
- 125I]iodo-19-norpregna-1,3,5(10),20-tetr aene-3,17-diol
- (1988) J. Med. Chem. , vol.31 , pp. 1946-1950
- Ali, H.¹ Rousseau, J.² Ghaffari, M.A.³ van Lier, J.E.⁴

2
- 0027443712
- 125I] iodovinylestradiols: effect on receptor binding and receptor-mediated target tissue uptake
- (1993) J. Med. Chem. , vol.36 , pp. 3061-3072
- Ali, H.¹ Rousseau, J.² van Lier, J.E.³

3
- 0025055583
- Synthesis and structure-affinity of a series of 7α-undecylestradiol derivatives: a potential vector for therapy and imaging of estrogen-receptor-positive cancers
- (1990) J. Med. Chem. , vol.33 , pp. 430-434
- Da Silva, J.N.¹ van Lier, J.E.²

4
- 50749132499
- 123I]Iodovinyl-11β-methoxyestradiol (MIVE2)- Part I. Radiotracer preparation and characterization
- (1992) Nucl. Med. Biol. , vol.19 , pp. 257-261
- Foulon, C.¹ Guilloteau, D.² Baulieu, J.L.³ Ribeiro-Barras, M.J.⁴ Desplanches, G.⁵ Frangis, Y.⁶ Besnard, J.⁷

5
- 0021148156
- Radioiodinated ligands for the estrogen receptor: effect of 3-O-methylation on tissue distribution
- (1984) J. Nucl. Med. , vol.25 , pp. 1116-1121
- Franke, L.¹ Hanson, R.²

6
- 0024487459
- 125I]Iodo-11-substituted-19-norpregna-1, 3,5(10),20-tetraene-3,17β-diols: the influence of 11-stereochemistry on tissue distribution of radioiodinated estrogens
- (1989) Nucl. Med. Biol. , vol.16 , pp. 3-9
- Hanson, R.¹ Frank, L.² Kaplan, M.³

7
- 0027409128
- 125I]iodovinyl 11β-ethyl-estradiol
- (1993) Nucl. Med. Biol. , vol.20 , pp. 351-358
- Hanson, R.¹ Ghoshal, M.² Murphy, F.³ Rosenthal, C.⁴ Gibson, R.⁵ Ferreira, N.⁶ Sood, V.⁷ Ruch, J.⁸

8
- 0022600603
- Synthesis of 17α-bromovinyl- and 17α-iodovinylnortestosterone derivatives
- (1986) Tetrahedron , vol.42 , pp. 3575-3578
- Hofmeister, H.¹ Laurent, H.² Schulze, P.E.³ Wiechert, R.⁴

9
- 0031081794
- Uptake and interconversion of the Z and E isomers of 17α-iodovinyl-11β-methoxyestradiol in the immature female rat
- (1997) Steroids , vol.62 , pp. 244-252
- Hughes, A.¹ Larson, S.M.² Hanson, R.N.³ DeSombre, E.R.⁴

10
- 0002228188
- Synthesis of 7-ω-amidoalkyl-substituted 6,7-dehydroestra-3,17β-diols
- (1999) Kyushu Daigaku Kino-bushitsu Kenkyusho Hokoku , vol.13 , Issue.1 , pp. 31-36
- Inohae, E.¹ Thiemann, T.² Mataka, S.³ Melo e Silva, M.C.⁴ Patricio, L.⁵

11
- 0025945627
- Structure-activity relationships of estrogenic ligands: synthesis and evaluation of (17α,20E)-and (17α,20Z)-21-halo-19-norpregna-1,3,5(10),20-tetraene-3,17β-diols
- (1991) J. Med. Chem. , vol.34 , pp. 2754-2759
- Napolitano, E.¹ Fiaschi, R.² Hanson, R.N.³

12
- 50749135432
- 123I]Iodovinyl-11β-methoxyestradiol (MIVE2)-Part II. Preliminary results in patients with breast carcinoma
- (1992) Nucl. Med. Biol. , vol.19 , pp. 263-267
- Ribeiro-Barras, M.J.¹ Foulon, C.² Baulieu, J.L.³ Guilloteau, D.⁴ Bougnous, P.⁵ Lansac, J.⁶ Besnard, J.C.⁷

13
- 0030790124
- Imaging of estrogen receptors in primary and metastatic breast cancer patients with iodine-123-labeled Z-MIVE
- (1997) J. Clin. Oncol. , vol.15 , pp. 2536-2545
- Rijks, L.J.¹ Bakker, P.J.² van Tienhoven, G.³ Noorduyn, L.A.⁴ Boer, G.J.⁵ Rietbroek, R.C.⁶ Taat, C.W.⁷ Janssen, A.G.⁸ Veenhof, C.H.⁹ van Royen, E.A.¹⁰

14
- 0030907782
- 123I]iodovinylestradiol is a promising radioligand for estrogen receptor imaging in human breast cancer
- (1997) Nucl. Med. Biol. , vol.24 , pp. 65-75
- Rijks, L.J.M.¹ Boer, G.J.² Endert, E.³ de Bruin, K.⁴ Janssen, A.G.⁵ van Royen, E.A.⁶

15
- 6844259881
- Biodistribution and dosimetry of iodine-123-labelled Z-MIVE: an oestrogen receptor ligand for breast cancer imaging
- (1998) Eur. J. Nucl. Med. , vol.25 , pp. 40-47
- Rijks, L.J.¹ Sokole, E.B.² Stabin, M.G.³ de Bruin, K.⁴ Janssen, A.G.⁵ van Royen, E.A.⁶

16
- 0006935996
- Takagishi, S., Schlosser, M., 1991 Fluorine- and trifluoromethyl-substituted toluenes: Site selective metalation of aromatic or benzylic positions, Synlett 119-121

17
- 0006936241
- Tedesco, R., Fiaschi, R., Napolitano, , E, , 1995 6-Oxoestradiols from estradiols: Exploiting site selective metalation of aralkyl systems with superbases, Synthesis 1493-1495

18
- 0030069547
- 123I]-labeled-Z-17α-iodovinyl-11β-chloromethyl-estradiol
- (1996) Nucl. Med. Biol. , vol.23 , pp. 69-73
- Zeicher, M.¹ Delcorde, A.² Quivy, J.³ Dupuis, Y.⁴ Vervist, A.⁵ Fruhling, J.⁶

* 이 정보는 Elsevier사의 SCOPUS DB에서 KISTI가 분석하여 추출한 것입니다.