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Volumn 36, Issue 2, 2001, Pages 185-193

Synthesis and inhibitory activity towards human leukocyte elastase of new 7α-methoxy and 7α-chloro (2-acyloxymethyl) cephem derivatives

(8) Balsamo, Aldo a Cercignani, Giovanni a Gentili, Daniela a Lapucci, Annalina a Macchia, Marco a Orlandini, Elisabetta a Rapposelli, Simona a Rossello, Armando a

a UNIVERSITY OF PISA (Italy)

Author keywords

C 2 hydroxymethyl cephem derivative; Cephalosporin derivative; Elastase inhibitor; HLE inhibitor

Indexed keywords

3 ACETOXYMETHYL 2 [(4 FLUOROBENZOYL)OXYMETHYL] 8 OXO (6H) 5 THIA 1 AZABICYCLO[4.2.0]OCT 2 EN 7C CHLORO 5,5 DIOXIDE; 3 ACETOXYMETHYL 2 [(4 FLUOROBENZOYL)OXYMETHYL] 8 OXO (6H) 5 THIA 1 AZABICYCLO[4.2.0]OCT 2 EN 7C METHYLOXY 5,5 DIOXIDE; 3 ACETOXYMETHYL 2 BENZOYLOXYMETHYL 8 OXO (6H) 5 THIA 1 AZABICYCLO[4.2.0]OCT 2 EN 7C CHLORO 5,5 DIOXIDE; 3 ACETOXYMETHYL 2 BENZOYLOXYMETHYL 8 OXO (6H) 5 THIA 1 AZABICYCLO[4.2.0]OCT 2 EN 7C METHYLOXY 5,5 DIOXIDE; 3 ACETOXYMETHYL 2 PIVALOYLOXYMETHYL 8 OXO (6H) 5 THIA 1 AZABICYCLO[4.2.0]OCT 2 EN 7C METHYLOXY 5,5 DIOXIDE; CEPHEM DERIVATIVE; LEUKOCYTE ELASTASE; PANCREATIC ELASTASE; UNCLASSIFIED DRUG;

ARTICLE; DRUG STRUCTURE; DRUG SYNTHESIS; ENZYME ACTIVITY; ENZYME INHIBITION; STRUCTURE ACTIVITY RELATION;

ANIMALS; CEPHALOSPORINS; ENZYME INHIBITORS; HUMANS; KINETICS; LACTAMS; LEUKOCYTES; PANCREAS; PANCREATIC ELASTASE; STRUCTURE-ACTIVITY RELATIONSHIP; SWINE;

EID: 0035246590 PISSN: 02235234 EISSN: None Source Type: Journal
DOI: 10.1016/S0223-5234(01)01211-9 Document Type: Article

Times cited : (8)

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* 이 정보는 Elsevier사의 SCOPUS DB에서 KISTI가 분석하여 추출한 것입니다.