Low-affinity M2 receptor binding state mediates mouse atrial bradycardia: Comparative effects of carbamylcholine and the M1 receptor agonists sabcomeline and xanomeline

Journal of Pharmacology and Experimental Therapeutics

Volumn 296, Issue 3, 2001, Pages 818-824

  Stengel, Peter W ^a   Cohen, Marlene L ^a  

^a ELI LILLY AND COMPANY   (United States)

Author keywords

[No Author keywords available]

Indexed keywords

ATROPINE; CARBACHOL; MUSCARINIC M1 RECEPTOR AGONIST; MUSCARINIC M2 RECEPTOR; MUSCARINIC M2 RECEPTOR AGONIST; SABCOMELINE; XANOMELINE;

ALZHEIMER DISEASE; ANIMAL EXPERIMENT; ANIMAL MODEL; ANIMAL TISSUE; ARTICLE; BRADYCARDIA; CONTROLLED STUDY; DISSOCIATION CONSTANT; DRUG ANTAGONISM; DRUG RECEPTOR BINDING; HEART ATRIUM; MOUSE; NONHUMAN; PKA; PRIORITY JOURNAL; RECEPTOR AFFINITY; RECEPTOR OCCUPANCY;

ANIMALS; ATROPINE; BRADYCARDIA; CARBACHOL; DRUG INTERACTIONS; HEART; HEART RATE; IMINES; MICE; MUSCARINIC AGONISTS; PYRIDINES; QUINUCLIDINES; RECEPTOR, MUSCARINIC M1; RECEPTOR, MUSCARINIC M2; RECEPTORS, MUSCARINIC; THIADIAZOLES;

EID: 0035123318     PISSN: 00223565     EISSN: None     Source Type: Journal    
DOI: None     Document Type: Article

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