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Volumn 334, Issue 2, 2001, Pages 45-52

Benzophenone derivatives and related compounds as potent histamine H3-receptor antagonists and potential PET/SPECT ligands

(10) Sasse, Astrid a Ligneau, Xavier c Sadek, Bassem a Elz, Sigurd a Pertz, Heinz H a Ganellin, C Robin c Arrang, Jean Michel b Schwartz, Jean Charles b Schunack, Walter a Stark, Holger d

a FREIE UNIVERSITÄT BERLIN (Germany)

b CENTRE PAUL BROCA (France)

c Laboratoire Bioprojet (France)

d GOETHE UNIVERSITY (Germany)

Author keywords

Benzophenone; H3 receptor; Histamine; PET; SPECT

Indexed keywords

3 FLUOROPHENYL 4 [3 (1H IMIDAZOL 4 YL)PROPYLOXY]PHENYLMETHANONE; 4 [3 (1H IMIDAZOL 4 YL)PROPYLOXY]PHENYL 3 IODOPHENYL METHANONE; 4 [3 (1H IMIDAZOL 4 YL)PROPYLOXY]PHENYLPHENYLMETHANONE; BENZOPHENONE DERIVATIVE; FLUORINE; HALOGEN; HISTAMINE H3 RECEPTOR ANTAGONIST; IMIDAZOLE DERIVATIVE; IODINE; LIGAND; UNCLASSIFIED DRUG;

ANIMAL EXPERIMENT; ANIMAL TISSUE; CONFERENCE PAPER; DRUG POTENCY; DRUG SELECTIVITY; DRUG STRUCTURE; DRUG SYNTHESIS; GUINEA PIG; MALE; MOUSE; NONHUMAN; POSITRON EMISSION TOMOGRAPHY; PRIORITY JOURNAL; RAT; RECEPTOR BLOCKING; SINGLE PHOTON EMISSION COMPUTER TOMOGRAPHY; STRUCTURE ACTIVITY RELATION;

ANIMALS; BENZOPHENONES; CEREBRAL CORTEX; GUINEA PIGS; HISTAMINE ANTAGONISTS; LIGANDS; MALE; MICE; MUSCLE, SMOOTH; RATS; RECEPTORS, HISTAMINE H3; STRUCTURE-ACTIVITY RELATIONSHIP; TOMOGRAPHY, EMISSION-COMPUTED; TOMOGRAPHY, EMISSION-COMPUTED, SINGLE-PHOTON;

EID: 0035106626 PISSN: 03656233 EISSN: None Source Type: Journal
DOI: 10.1002/1521-4184(200102)334:2<45::AID-ARDP45>3.0.CO;2-2 Document Type: Conference Paper

Times cited : (21)

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