Structure-activity relationships in a series of 8-substituted xanthines as A1-adenosine receptor antagonists

Bioorganic and Medicinal Chemistry

Volumn 9, Issue 3, 2001, Pages 575-583

  Strappaghetti, Giovannella ^a   Corsano, Stefano ^a   Barbaro, Roberta ^a   Giannaccini, Gino ^b   Betti, Laura ^b  

^a UNIVERSITY OF PERUGIA   (Italy)

^b UNIVERSITY OF PISA   (Italy)

Author keywords

DCC; Dicyclohexylcarbodiimide

Indexed keywords

2 [4 (2 CARBOXYETHYL)PHENETHYLAMINO]ADENOSINE 5' (N ETHYLCARBOXAMIDE); ADENOSINE A1 RECEPTOR; ADENOSINE A2A RECEPTOR; CAFFEINE; THEOPHYLLINE; XANTHINE DERIVATIVE;

ANIMAL TISSUE; ARTICLE; BRAIN CORTEX; CATTLE; CORPUS STRIATUM; DRUG RECEPTOR BINDING; DRUG SYNTHESIS; NONHUMAN; NUCLEAR MAGNETIC RESONANCE SPECTROSCOPY; RECEPTOR AFFINITY; STRUCTURE ACTIVITY RELATION;

ANIMALS; BINDING, COMPETITIVE; CATTLE; CELL MEMBRANE; CEREBRAL CORTEX; CORPUS STRIATUM; RADIOLIGAND ASSAY; RECEPTORS, PURINERGIC P1; STRUCTURE-ACTIVITY RELATIONSHIP; THEOPHYLLINE; XANTHINES;

EID: 0035105396     PISSN: 09680896     EISSN: None     Source Type: Journal    
DOI: 10.1016/S0968-0896(00)00271-6     Document Type: Article

References (18)