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Volumn 16, Issue 1, 2001, Pages 15-34

Potential of pyrazolooxadiazinone derivatives as serine protease inhibitors

(11) Vicentini, C B a Guarneri, M a Andrisano, V a Guccione, S a Langer, T a Marschhofer, R a Chabin, R a Edison, A M a Huang, X a Knight, W B a Giori, P a

a UNIVERSITY OF CATANIA (Italy)

Author keywords

FlexX docking; Mechanism based inhibitors; Pyrazolo 4,3 c 1,2,5 oxadiazin 3(5H) ones; Serine Proteases

Indexed keywords

ALIPHATIC COMPOUND; AROMATIC COMPOUND; LEUKOCYTE ELASTASE; OXYGEN; PYRAZOLE; PYRAZOLOOXADIAZINONE DERIVATIVE; SERINE PROTEINASE INHIBITOR; SULFUR; UNCLASSIFIED DRUG;

ARTICLE; CHEMICAL INTERACTION; CHEMICAL MODIFICATION; CONTROLLED STUDY; DRUG STRUCTURE; ENZYME ACTIVE SITE; ENZYME INHIBITION; HUMAN; HYDROLYSIS; MOLECULAR MODEL; PRIORITY JOURNAL; STRUCTURE ACTIVITY RELATION; ULTRAVIOLET SPECTROPHOTOMETRY;

STAPHYLOCOCCUS PHAGE 3A;

EID: 0035057967 PISSN: 87555093 EISSN: None Source Type: Journal
DOI: 10.1080/14756360109162352 Document Type: Article

Times cited : (6)

References (50)

1
- 0017880439
- (1978) Agents and Action , vol.8 , pp. 3
- Baggiolini, M.¹ Bretz, U.² Dewald, B.³ Feigenson, M.E.⁴

2
- 0028240276
- (1994) Am. Respir. Crit. Care Med. , vol.150 , pp. 207-213
- Birrer, P.¹ McElvaney, N.G.² Rudeburg, A.³ Wirz-Sommer, C.⁴ Liecht-Gallati, S.⁵ Kraemer, R.⁶ Hubbard, R.⁷ Crystal, R.G.⁸

3
- 0004303261
- Boca Raton, Florida: CRC Press
- (1990) Focus on Pulmonary Pharmacology and Toxicology
- Weinbaum, G.¹ Groutas, W.C.²

4
- 77956791952
- Human leukocyte elastase inhibitors
- (Bristol, J.A., Editor) San Diego: Academic Press, Inc.
- (1994) Annu. Rep. Med. Chem. , pp. 195
- Hlasta, D.J.¹ Pagani, E.D.²

5
- 0004006847
- (Coxon, J.M. Editor). Boca Raton, Florida: CRC Press Inc.
- (1988) Mechanism-Based Enzyme Inactivation: Chemistry and Enzymology
- Silverman, R.B.¹

6
- 0005284631
- Greenwich, Connecticut: JAI PRESS INC.
- (1992) Advances in Detailed Reaction Mechanisms , vol.2 , pp. 243
- Abell, A.D.¹

7
- 0028925509
- (1995) Eur. J. Med. Chem. , vol.30 , pp. 199
- Vergely, I.¹ Boggetto, N.² Okochi, V.³ Golpayegani, S.⁴ Reboud-Ravaux, M.⁵ Kobaiter, R.⁶ Joyeau, R.⁷ Wakselman, M.⁸

8
- 0029034742
- (1995) J. Med. Chem. , vol.38 , pp. 2449
- Finke, P.A.¹ Shrenik, K.S.² Fletcher, D.S.³ Ashe, B.M.⁴ Brause, K.A.⁵ Chandler, G.O.⁶ Dellea, P.S.⁷ Hand, K.M.⁸ Maycock, A.L.⁹ Osinga, D.G.¹⁰ Underwood, D.J.¹¹ Weston, H.¹² Davies, P.¹³ Doherty, J.B.¹⁴

9
- 0022447698
- (1986) J. Heterocylic Chem. , vol.23 , pp. 585
- Giori, P.¹ Veronese, A.C.² Poli, T.³ Vicentini, C.B.⁴ Manfrini, M.⁵ Guarneri, M.⁶

10
- 85037407836
- Tesi di Dottorato di Ricerca (Italian PhD)
- (1992)
- Guccione, S.¹

11
- 0015937153
- (1973) Biochemistry , vol.12 , pp. 828
- Brown, W.E.¹ Wold, F.²

12
- 0000540529
- (1982) J. Am. Chem. Soc. , vol.104 , pp. 6785
- Moorman, A.R.¹ Abeles, R.H.²

13
- 0026725323
- (1992) Biochemistry , vol.31 , pp. 4980
- Knight, W.B.¹ Maycock, A.L.² Green, B.G.³ Ashe, B.M.⁴ Gale, P.⁵ Weston, H.⁶ Finke, P.E.⁷ Hagmann, W.K.⁸ Shah, S.K.⁹ Doherty, J.B.¹⁰

14
- 0025098316
- and references therein
- (1990) J. Med. Chem. , vol.33 , pp. 464
- Krantz, A.¹ Spencer, R.W.² Fat Tam, T.³ Liak, T.J.⁴ Copp, L.J.⁵ Thomas, E.M.⁶ Rafferty, S.P.⁷

15
- 0005237831
- The Chemistry of Functional Groups, Supplement S: The Chemistry of Sulphur-containing Functional Groups Chichester: John Wiley and Sons Ltd, Baffins Lane
- (1993)
- Patai, S.¹ Rappopart, Z.²

16
- 0005238547
- 1
- (1909) J. Pr. Chem. , vol.2 , pp. 79
- Mohr, E.¹

17
- 0005320194
- (1959) J. Am. Chem. Soc. , vol.81 , pp. 2456
- Taylor, E.C.¹ Hartke, K.S.²

18
- 0019799625
- (1981) II Farmaco Ed. Sc. , vol.36 , pp. 1019
- Giori, P.¹ Mazzotta, D.² Vertuani, G.³ Guarneri, M.⁴ Pancaldi, D.⁵ Brunelli, A.⁶

19
- 0024245377
- (1988) II Farmaco Ed. Sc. , vol.43 , pp. 891
- Ferroni, R.¹ Milani, L.² Simoni, D.³ Orlandini, P.⁴ Poli, T.⁵ Guarneri, M.⁶ Taddeo, U.⁷

20
- 0005310970
- and references therein
- (1996) Heterocyclic Chem. , vol.33 , pp. 459
- Guccione, S.¹ Monsù-Scolaro, L.² Russo, F.J.³

21
- 84980900145
- (1956) Helv. Chim. Acta. , vol.39 , pp. 986
- Schmidt, P.¹ Druey, J.²

22
- 0000818685
- (1969) Bull. Chem. Soc. Jpn. , vol.42 , pp. 1653
- Baba, H.¹ Hori, I.² Hayashi, T.³ Midorikawa, K.⁴

23
- 0002700305
- (H.R. Snyder, Ed.). New York: John Wiley and Sons, Inc.
- (1948) Org. Syntheses , vol.28 , pp. 89
- Frank, R.L.¹ Smith, P.V.²

24
- 0005324868
- (1934) J. Am. Chem. Soc. , vol.56 , pp. 1408
- Douglass, I.B.¹ Dains, F.B.²

25
- 85037420376
- The program SYBYL 6.5 is available from Tripos Associates, 1699 South Hanley Road, St Louis, MO 63144, USA.
- (1999)

26
- 85037417462
- Gaussian Inc, Pittsburgh, Pasadena, USA.

27
- 4243263213
- Chem. Rev. , vol.86 , pp. 681
- Feller, D.¹ Davidson, E.R.²

28
- 0005237832
- (1987) Proc. Natl. Acad. Sci. USA , vol.84 , pp. 2228
- Sinha, S.¹ Watorek, W.² Karr, S.³ Giles, J.⁴ Bode, W.⁵ Travis, J.⁶

29
- 0022701771
- (1986) EMBO J. , vol.5 , pp. 813
- Bode, W.¹ Papmokos, E.² Musil, D.³ Seem, U.⁴ Iler⁵

30
- 0013956919
- and references therein
- (1966) Biochem. J. , vol.101 , pp. 229
- Hartley, B.S.¹ Kauffman, D.L.²

31
- 0022801412
- (1986) EMBO J. , vol.5 , pp. 2453
- Bode, W.¹ Wei, A.² Huber, R.³ Meyer, E.⁴ Travis, J.⁵ Neumann, S.⁶

32
- 85037419057
- Internet Address: Gopher://pdbpdbbnlgov

33
- 0023721908
- (1988) FEBS Lett. , vol.234 , pp. 367
- Wei, A.¹ Mayr, I.² Bode, W.³

34
- 0030076041
- (1996) J. Comput-Aided Mol. Des. , vol.10 , pp. 41
- Rarey, M.¹ Wefing, S.² Lengauer, T.³

35
- 84988115618
- (1989) J. Comput. Chem. , vol.10 , pp. 982
- Clark, M.¹ Cramer III, R.² Van Opdenbosh, N.³

36
- 0026662213
- (1992) Biochemistry , vol.31 , pp. 8160
- Knight, W.B.¹ Green, B.G.² Chabin, R.³ Gale, P.⁴ Maycock, A.L.⁵ Weston, H.⁶ Kuo, D.⁷ Westler, W.M.⁸ Dorn, C.P.⁹ Finke, P.E.¹⁰ Hagmann, W.K.¹¹ Hale, J.J.¹² Liesch, J.¹³ MacCoss, M.¹⁴ Navia, M.¹⁵ Shah, S.K.¹⁶ Underwood, D.¹⁷ Doherty, J.B.¹⁸

37
- 0025914721
- (1991) Arch. Biochem. Biophys. , vol.286 , pp. 284
- Green, B.G.¹ Weston, H.² Ashe, B.M.³ Doherty, J.B.⁴ Finke, P.⁵ Hagmann, W.⁶ Lark, M.⁷ Mao, J.⁸ Maycock, A.⁹ Mumford, R.¹⁰ Walakovits, L.¹¹ Knight, W.B.¹²

38
- 0000325609
- (1983) Adv. Enzymol. , vol.61 , pp. 201
- Morrison, J.F.¹ Walsh, C.T.²

39
- 0019817468
- (1981) Biochim. Biophys. Acta , vol.661 , pp. 342
- Fujii, S.¹ Hitomi, Y.²

40
- 0014211618
- (1967) Biochem. Biophys. Res. Commun. , vol.27 , pp. 157
- Schechter, I.¹ Berger, A.²

41
- 0026589236
- (1992) J. Med. Chem. , vol.35 , pp. 1121
- Hernandez, M.A.¹ Powers, J.C.² Glinski, J.³ Oleksyszyn, J.⁴ Vijayalakshmi, J.⁵ Meyer E.F., Jr.⁶

42
- 0005358577
- (C. Nagata Ed.). Amsterdam: Elsevier
- (1985) Biomolecules , vol.21
- Umeyama, H.¹ Nakagawa, S.²

43
- 0026027796
- (1991) Tetrahedron , vol.47 , pp. 2649
- Zimmerman, S.C.¹ Korthals, J.S.² Cramer, K.D.³

44
- 0029025244
- (1995) J. Med. Chem. , vol.38 , pp. 76
- Edwards, P.D.¹ Wolanin, D.J.² Andisik, D.W.³ Davis, M.W.⁴

45
- 0001477758
- (1993) J. Org. Chem. , vol.58 , pp. 6155
- Ganesan, A.¹ Heathcock, C.H.²

46
- 85037420892
- 3D QSAR in Drug Design: Theory, Methods and Applications Leiden: ESCOM
- (1993)
- Kubinyi, H.¹

47
- 0005285693
- QSAR; Hansch Analysis and Related Approaches, Methods and Principles in Medicinal Chemistry Weinheim: VCH.
- (1993)
- Kubinyi, H.¹

48
- 0027772480
- (1993) Drug Design and Discovery , vol.10 , pp. 297
- Barth, A.¹ Wahab, M.² Brandt, W.³ Frost, K.⁴

49
- 0001706111
- (1993) Heterocycles , vol.36 , pp. 2291
- Vicentini, C.B.¹ Veronese, A.C.² Manfrini, M.³ Guccione, S.⁴ Guarneri, M.⁵ Giori, P.⁶

50
- 77953081439
- (2000) Synthesis , vol.1 , pp. 72
- Baraldi, P.G.¹ Pineda de las Infantas, M.J.² Manfredini, S.³ Romagnoli, R.⁴

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