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Volumn 16, Issue 1, 2001, Pages 1-13

Protease inhibitors, part 13: Specific, weakly basic thrombin inhibitors incorporating sulfonyl dicyandiamide moieties in their structure

(3) Clare, B W a Scozzafava, A a Supuran, C T a

a UNIVERSITY OF FLORENCE (Italy)

Author keywords

Dicyandiamide; Inhibitor; Reduced basicity; Sulfonyl; Tautomerism; Thrombin; Trypsin

Indexed keywords

ASPARTIC ACID; DIAMIDE; GUANIDINE; PROTEINASE INHIBITOR; SERINE PROTEINASE; SULFONE DERIVATIVE; THROMBIN; THROMBIN INHIBITOR; TRYPSIN;

ALKALINITY; ARTICLE; BINDING AFFINITY; CHEMICAL INTERACTION; CONTROLLED STUDY; DERIVATIZATION; DRUG STRUCTURE; ENZYME ACTIVE SITE; ENZYME INHIBITION; ENZYME SUBSTRATE; PRIORITY JOURNAL; STRUCTURE ANALYSIS;

EID: 0035054632 PISSN: 87555093 EISSN: None Source Type: Journal
DOI: 10.1080/14756360109162351 Document Type: Article

Times cited : (6)

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