New D-modified androstane derivatives as aromatase inhibitors

Steroids

Volumn 66, Issue 8, 2001, Pages 645-653

  Penov Gaši, Katarina M ^a   Stanković, Slobodanka M ^a   Csanádi, János J ^a   Djurendić, Evgenija A ^a   Sakač, Marija N ^a   Medić Mijačević, Ljubica ^a   Arcson, Otto N ^a   Stojanović, Srdjan Z ^a   Andrić, Silvana ^a   Molnar Gabor, Dora ^a   Kovačević, Radmila ^a  

^a UNIVERSITY OF NOVI SAD   (Serbia)

Author keywords

Androgens synthesis; D Secosteroids; Inhibition of aromatase activity

Indexed keywords

AMINOGLUTETHIMIDE; ANDROSTANE DERIVATIVE; AROMATASE; AROMATASE INHIBITOR; SECOSTEROID;

ANIMAL TISSUE; ARTICLE; CARBON NUCLEAR MAGNETIC RESONANCE; CONTROLLED STUDY; DRUG STRUCTURE; DRUG SYNTHESIS; ENZYME ACTIVITY; ENZYME KINETICS; FEMALE; HYDROLYSIS; NONHUMAN; OVARY; OXIDATION; PROTON NUCLEAR MAGNETIC RESONANCE; RAT; REACTION ANALYSIS; X RAY CRYSTALLOGRAPHY;

ANDROSTANES; ANIMALS; AROMATASE INHIBITORS; BENZOQUINONES; BINDING, COMPETITIVE; CRYSTALLOGRAPHY, X-RAY; FEMALE; HYDROLYSIS; INHIBITORY CONCENTRATION 50; KINETICS; MAGNETIC RESONANCE SPECTROSCOPY; MODELS, MOLECULAR; RATS; RATS, WISTAR;

EID: 0034950269     PISSN: 0039128X     EISSN: None     Source Type: Journal    
DOI: 10.1016/S0039-128X(01)00096-4     Document Type: Article

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