Conformation of the tripeptide Cbz-Pro-Leu-Trp-OBzl(CF3)2 deduced from two-dimensional 1H-NMR and conformational energy calculations is related to its affinity for NK1-receptor

Journal of Peptide Science

Volumn 7, Issue 6, 2001, Pages 323-330

  Millet, Régis ^a   Goossens, Laurence ^a   Goossens, Jean Franois ^a   Chavatte, Philippe ^a   Bertrand Caumont, Karine ^a   Houssin, Raymond ^a   Hénichart, Jean Pierre ^a  

^a Faculté des Sciences Pharmaceutiques et Biologiques Université de Lille   (France)

Author keywords

Conformational analysis; Neurokinin A; NMR; Substance P

Indexed keywords

HYDROGEN; LIGAND; TACHYKININ RECEPTOR; TRIPEPTIDE;

ARTICLE; CALCULATION; CHEMICAL MODIFICATION; CONTROLLED STUDY; ENERGY; HYDROGEN BOND; NUCLEAR MAGNETIC RESONANCE; PARAMETER; PEPTIDE ANALYSIS; PRIORITY JOURNAL; PROTEIN CONFORMATION; RECEPTOR AFFINITY; RIGIDITY;

EID: 0034931327     PISSN: 10752617     EISSN: None     Source Type: Journal    
DOI: 10.1002/psc.326     Document Type: Article

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