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Canadian Journal of Chemistry

Volumn 79, Issue 4, 2001, Pages 377-387

Synthesis and evaluation of novel β-lactam inhibitors of human leukocyte elastase

(4) Koteva, K P a Cantin, A M a Neugebauer, W A a Escher, E a

a UNIVERSITY OF SHERBROOKE (Canada)

Author keywords

Neutrophil elastase; Peptides; Protease inhibitors; lactams

Indexed keywords

CELLULOSE DERIVATIVES; HYDROPHOBICITY; ORGANIC ACIDS; PULMONARY DISEASES;

STRUCTURE-ACTIVITY RELATIONSHIP;

ENZYME INHIBITION;

1 BENZHYDRYLPIPERAZINE; 7ALPHA METHOXY CEPHALOSPORANIC ACID; BETA LACTAM DERIVATIVE; CEPHALOSPORANIC ACID DERIVATIVE; LEUKOCYTE ELASTASE; PROTEINASE INHIBITOR; SERINE PROTEINASE; TRYPTOPHANYL 9 FLUORENYLMETHYL ESTER; UNCLASSIFIED DRUG;

ARTICLE; DRUG POTENCY; DRUG SYNTHESIS; IC 50; LUNG DISEASE; STRUCTURE ACTIVITY RELATION;

EID: 0034881139 PISSN: 00084042 EISSN: None Source Type: Journal
DOI: 10.1139/v01-062 Document Type: Article

Times cited : (10)

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