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Volumn 9, Issue 10, 2001, Pages 2609-2624
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Parallel synthesis and biological activity of a new class of high affinity and selective δ-opioid ligand
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Author keywords
[No Author keywords available]
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Indexed keywords
1 [2 (1,3 DIHYDRO 1,3 DIOXO 2H ISOINDOL 2 YL)ETHYL] 1,2,3,4 TETRAHYDRO 2 [(4 METHYLPHENYL)SULFONYL]ISOQUINOLINE;
1 [2 [[(6 METHYL 3 PYRIDINYL)CARBONYL]AMINO]ETHYL] 1,2,3,4 TETRAHYDRO 2 [(4 METHYLPHENYL)SULFONYL]ISOQUINOLINE;
1,2,3,4,4A,5,12,12AALPHA OCTAHYDRO 4AALPHA (3 HYDROXYPHENYL) 2 METHYLQUINOLINO[2,3 G]ISOQUINOLINE;
4 [ALPHA (4 ALLYL 2,5 DIMETHYL 1 PIPERAZINYL) 3 METHOXYBENZYL] N,N DIETHYLBENZAMIDE;
ACETAMIDE DERIVATIVE;
ANALGESIC AGENT;
DELTA OPIATE RECEPTOR;
FENTANYL;
FORMALDEHYDE;
ISOQUINOLINE DERIVATIVE;
KAPPA OPIATE RECEPTOR;
LIGAND;
MORPHINE;
MU OPIATE RECEPTOR;
MU OPIATE RECEPTOR AGONIST;
N [[[2 [1,2,3,4 TETRAHYDRO 2 [(4 BUTYLPHENYL)SULFONYL] 1 ISOQUINOLINYL]ETHYL]AMINO]CARBONYL] 1H IMIDAZOL 1 ACETAMIDE;
N METHYL N [7 (1 PYRROLIDINYL) 1 OXASPIRO[4.5]DEC 8 YL]BENZENEACETAMIDE;
NALTRINDOLE;
PHTHALIMIDE DERIVATIVE;
TETRAHYDROISOQUINOLINE DERIVATIVE;
TETRAHYDROISOQUINOLINE SULFONAMIDE;
UNCLASSIFIED DRUG;
ANALGESIC ACTIVITY;
ANIMAL CELL;
ANIMAL EXPERIMENT;
ANIMAL MODEL;
ANIMAL TISSUE;
ANTINOCICEPTION;
BINDING AFFINITY;
CHO CELL;
COMPARATIVE STUDY;
CONFERENCE PAPER;
CONTROLLED STUDY;
DOSE RESPONSE;
DRUG ACTIVITY;
DRUG POTENCY;
DRUG RECEPTOR BINDING;
DRUG SELECTIVITY;
DRUG SOLUBILITY;
DRUG STRUCTURE;
DRUG SYNTHESIS;
HUMAN;
IN VIVO STUDY;
LIGAND BINDING;
MALE;
MOLECULAR CLONING;
MOUSE;
NONHUMAN;
PAIN;
RAT;
STRUCTURE ACTIVITY RELATION;
AMIDES;
ANALGESICS, OPIOID;
ANIMALS;
BENZAMIDES;
BRAIN;
CATALYSIS;
COMBINATORIAL CHEMISTRY TECHNIQUES;
GUINEA PIGS;
HUMANS;
INHIBITORY CONCENTRATION 50;
ISOQUINOLINES;
LIGANDS;
MALE;
MALEIMIDES;
MEMBRANE PROTEINS;
MICE;
MICE, INBRED ICR;
MOLECULAR STRUCTURE;
MORPHINE;
NALTREXONE;
NERVE TISSUE PROTEINS;
PAIN MEASUREMENT;
PHTHALIMIDES;
PIPERAZINES;
QUINOLINES;
RATS;
RATS, WISTAR;
RECEPTORS, OPIOID, DELTA;
STRUCTURE-ACTIVITY RELATIONSHIP;
SUCCINIMIDES;
SULFONAMIDES;
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EID: 0034857529
PISSN: 09680896
EISSN: None
Source Type: Journal
DOI: 10.1016/S0968-0896(01)00017-7 Document Type: Article |
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Times cited : (17)
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References (16)
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