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Volumn 9, Issue 10, 2001, Pages 2709-2726
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2-Alkynyl-8-aryladenines possessing an amide moiety: Their synthesis and structure-activity relationships of effects on hepatic glucose production induced via agonism of the A2B adenosine receptor
a
a
EISAI CO LTD
(Japan)
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Author keywords
[No Author keywords available]
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Indexed keywords
2 (2 HYDROXYETHYL) 1 [3 (2 PHENYLPYRAZOLO[1,5 A]PYRIDIN 3 YL)ACRYLOYL]PIPERIDINE;
3 [(2 AMINO 6 CHLORO 5 NITRO 4 PYRIMIDINYL)AMINO]BENZOIC ACID;
3 [6 AMINO 8 (3 FLUOROPHENYL) 2 [2 (1 HYDROXYCYCLOHEXYL) 1 ETHYNYL] 9H 9 PURINYL]BENZAMIDE;
8 (3,4 DIMETHOXYSTYRYL) 7 METHYL 1,3 DIPROPYLXANTHINE;
9 (N ETHYL)BENZAMIDOADENINE DERIVATIVE;
ADENINE DERIVATIVE;
ADENOSINE 5' (N ETHYLCARBOXAMIDE);
ADENOSINE A1 RECEPTOR;
ADENOSINE A2A RECEPTOR;
ADENOSINE A2B RECEPTOR;
ADENOSINE A2B RECEPTOR ANTAGONIST;
ADENOSINE RECEPTOR BLOCKING AGENT;
ADENOSINE RECEPTOR STIMULATING AGENT;
AMIDE;
BENZAMIDE DERIVATIVE;
BENZENE DERIVATIVE;
CARBON;
CYCLIC AMP;
GLUCOSE;
N1 ETHYL 4 [6 AMINO 8 (3 FLUOROPHENYL) 2 [2 (1 HYDROXYCYCLOHEXYL) 1 ETHYNYL] 9H 9 PURINYL]BUTANAMIDE;
UNCLASSIFIED DRUG;
ANIMAL CELL;
BINDING AFFINITY;
BIOASSAY;
CELL CULTURE;
CHEMICAL REACTION;
CHO CELL;
CONFERENCE PAPER;
CONTROLLED STUDY;
CORRELATION FUNCTION;
DIAGNOSTIC VALUE;
DRUG ACTIVITY;
DRUG EFFECT;
DRUG POTENCY;
DRUG STRUCTURE;
DRUG SYNTHESIS;
GLUCONEOGENESIS;
HUMAN;
IC 50;
LIVER CELL;
MALE;
NONHUMAN;
RAT;
REACTION ANALYSIS;
STRUCTURE ACTIVITY RELATION;
ADENINE;
ALKYNES;
ANIMALS;
BENZAMIDES;
CELLS, CULTURED;
CHO CELLS;
CRICETINAE;
EMBRYO;
FEMALE;
GLUCOSE;
HEPATOCYTES;
HUMANS;
HYPOGLYCEMIC AGENTS;
INHIBITORY CONCENTRATION 50;
KIDNEY;
LIVER;
MAGNETIC RESONANCE SPECTROSCOPY;
MALE;
MASS SPECTROMETRY;
OVARY;
PURINES;
RADIOLIGAND ASSAY;
RATS;
RATS, WISTAR;
RECEPTORS, PURINERGIC P1;
STRUCTURE-ACTIVITY RELATIONSHIP;
TRANSFECTION;
CRICETINAE;
CRICETULUS GRISEUS;
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EID: 0034842262
PISSN: 09680896
EISSN: None
Source Type: Journal
DOI: 10.1016/S0968-0896(01)00201-2 Document Type: Conference Paper |
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Times cited : (40)
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References (28)
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