Dynamics of p2x7 receptor pore dilation: Pharmacological and functional consequences

Drug Development Research

Volumn 53, Issue 2-3, 2001, Pages 60-65

  Chessell, I P ^a   Grahames, C B A ^b   Michel, A D ^a   Humphrey, P P A ^a  

^a GLAXOSMITHKLINE   (United Kingdom)

^b PFIZER GLOBAL RESEARCH AND DEVELOPMENT   (United Kingdom)

Author keywords

Interleukin; P2X7; Pore dilation; Purinoceptor

Indexed keywords

2' O (4 BENZOYLBENZOYL) ADENOSINE TRIPHOSPHATE; 3' O (4 BENZOYLBENZOYL) ADENOSINE TRIPHOSPHATE; INTERLEUKIN 1BETA; MONOCLONAL ANTIBODY; PURINE P2X RECEPTOR; UNCLASSIFIED DRUG;

CELL TRANSPORT; CHANNEL GATING; CONCENTRATION RESPONSE; CONFERENCE PAPER; CONTROLLED STUDY; CYTOKINE RELEASE; CYTOLYSIS; DRUG CONFORMATION; DRUG DEGRADATION; DRUG MECHANISM; DRUG POTENCY; EMBRYO; HUMAN; HUMAN CELL; PHARMACODYNAMICS; POROSITY; PROTEIN EXPRESSION; RECEPTOR DENSITY;

EID: 0034841875     PISSN: 02724391     EISSN: None     Source Type: Journal    
DOI: 10.1002/ddr.1171     Document Type: Conference Paper

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