Microscopic kinetics and energetics distinguish GABAA receptor agonists from antagonists

Biophysical Journal

Volumn 81, Issue 5, 2001, Pages 2660-2670

  Jones, Mathew V ^a   Jonas, Peter ^b   Sahara, Yoshinori ^c   Westbrook, Gary L ^d  

^a UNIVERSITY OF WISCONSIN MADISON   (United States)

^b UNIVERSITY OF FREIBURG   (Germany)

^c TOKYO MEDICAL AND DENTAL UNIVERSITY   (Japan)

^d OREGON HEALTH AND SCIENCE UNIVERSITY   (United States)

Author keywords

[No Author keywords available]

Indexed keywords

3 AMINO 2 (3 CARBOXYPROPYL) 6 (4 METHOXYPHENYL)PYRIDAZINIUM BROMIDE; 3 PIPERIDEINE DERIVATIVE; 4 AMINOBUTYRIC ACID A RECEPTOR; 4 AMINOBUTYRIC ACID A RECEPTOR BLOCKING AGENT; 4 AMINOBUTYRIC ACID A RECEPTOR STIMULATING AGENT; BICUCULLINE METHIODIDE; FAMIRAPRINE; METHYLPHOSPHONIC ACID; NICOTINIC RECEPTOR;

ANIMAL TISSUE; ARTICLE; CHANNEL GATING; COMPETITIVE INHIBITION; CONFORMATIONAL TRANSITION; CONTROLLED STUDY; DIFFUSION; DRUG BINDING SITE; DRUG RECEPTOR BINDING; DRUG STRUCTURE; ENERGY TRANSFER; HIPPOCAMPUS; NONHUMAN; RAT;

ANIMALIA;

EID: 0034753212     PISSN: 00063495     EISSN: None     Source Type: Journal    
DOI: 10.1016/S0006-3495(01)75909-7     Document Type: Article

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