Terfenadine-β-cyclodextrin inclusion complex with antihistaminic activity enhancement

Drug Development and Industrial Pharmacy

Volumn 27, Issue 8, 2001, Pages 857-862

  Choi, Han Gon ^a   Lee, Beom Jin ^b   Han, Jeong Hee ^a   Lee, Mi Kyung ^a   Park, Kyung Mi ^a   Yong, Chul Soon ^c   Rhee, Jong Dal ^c   Kim, Yang Bae ^a   Kim, Chong Kook ^a  

^a Seoul National University   (South Korea)

^b Kangwon National University   (South Korea)

^c Yeungnam University   (South Korea)

Author keywords

Antihistaminic activity; Inclusion; Solubility; Terfenadine

Indexed keywords

ANTIHISTAMINIC AGENT; BETA CYCLODEXTRIN; TERFENADINE;

ANIMAL EXPERIMENT; ANIMAL MODEL; ARTICLE; CONTROLLED STUDY; DRUG ABSORPTION; DRUG ACTIVITY; DRUG BIOAVAILABILITY; DRUG FORMULATION; DRUG POTENCY; DRUG SOLUBILITY; HISTAMINE BLOOD LEVEL; HISTAMINE RELEASE; MALE; MATHEMATICAL COMPUTING; NONHUMAN; PH; POWDER; RAT;

ALGORITHMS; ANIMALS; BETA-CYCLODEXTRINS; CALORIMETRY, DIFFERENTIAL SCANNING; CHEMISTRY, PHYSICAL; CYCLODEXTRINS; EXCIPIENTS; HISTAMINE H1 ANTAGONISTS; HISTAMINE RELEASE; HYDROGEN-ION CONCENTRATION; KINETICS; MALE; PASSIVE CUTANEOUS ANAPHYLAXIS; POWDERS; RATS; RATS, SPRAGUE-DAWLEY; SOLUBILITY; SPECTROPHOTOMETRY, ULTRAVIOLET; TERFENADINE;

EID: 0034752911     PISSN: 03639045     EISSN: None     Source Type: Journal    
DOI: 10.1081/DDC-100107250     Document Type: Article

References (15)

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