Molecular targets for cannabidiol and its synthetic analogues: Effect on vanilloid VR1 receptors and on the cellular uptake and enzymatic hydrolysis of anandamide

British Journal of Pharmacology

Volumn 134, Issue 4, 2001, Pages 845-852

  Bisogno, Tiziana ^a   Hanuš, Lumír ^b   De Petrocellis, Luciano ^c   Tchilibon, Susanna ^b   Ponde, Datta E ^b   Brandi, Ines ^a   Moriello, Aniello Schiano ^c   Davis, John B ^d   Mechoulam, Raphael ^b   Di Marzo, Vincenzo ^a  

^a CNR   (Italy)

^b HEBREW UNIVERSITY OF JERUSALEM   (Israel)

^c CNR   (Italy)

^d GLAXOSMITHKLINE   (United Kingdom)

Author keywords

Anandam ide transporter; Cannabinoid; Endocannabinoid; FAAH; Receptors; Vanilloid

Indexed keywords

5' DIMETHYLHEPTYLCANNABIDIOL; 7 HYDROXY 5' DIMETHYLHEPTYLCANNABIDIOL; 7 HYDROXYCANNABIDIOL; ANANDAMIDE; CANNABIDIOL; CANNABIDIOL DERIVATIVE; CANNABINOID 1 RECEPTOR; CANNABINOID 2 RECEPTOR; CAPSAICIN; IONOMYCIN; UNCLASSIFIED DRUG; VANILLOID RECEPTOR; VANILLOID RECEPTOR 1;

ARTICLE; CONCENTRATION RESPONSE; CONTROLLED STUDY; DRUG RECEPTOR BINDING; DRUG SELECTIVITY; DRUG UPTAKE; HUMAN; HUMAN CELL; MOLECULAR DYNAMICS; PRIORITY JOURNAL;

EID: 0034751335     PISSN: 00071188     EISSN: None     Source Type: Journal    
DOI: 10.1038/sj.bjp.0704327     Document Type: Article

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