Mild and regioselective oxidative bromination of anilines using potassium bromide and sodium perborate

Tetrahedron Letters

Volumn 41, Issue 13, 2000, Pages 2083-2085

  Roche, Didier ^a   Prasad, Kapa ^a   Repic, Oljan ^a   Blacklock, Thomas J ^a  

^a NOVARTIS INSTITUTES FOR BIOMEDICAL RESEARCH   (United States)

Author keywords

[No Author keywords available]

Indexed keywords

AMMONIUM DERIVATIVE; BORIC ACID; MOLYBDENUM; POTASSIUM BROMIDE; SODIUM DERIVATIVE;

ARTICLE; BROMINATION; CHEMICAL REACTION; OXIDATION; REACTION ANALYSIS;

EID: 0034719745     PISSN: 00404039     EISSN: None     Source Type: Journal    
DOI: 10.1016/S0040-4039(00)00119-2     Document Type: Article

References (12)

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7. (f) Hanson, J. R.; Harpel, S.; Rodriguez Medina, I. C.; Rose, D. J. Chem. Res. 1997, 432-433.
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12. 4-Bromo-2-iodoanilines are common intermediates in the synthesis of indoles: Ezquerra, J.; Pedregal, C.; Lamas, C. J. Org. Chem. 1996, 61, 5804-5812 and references cited therein.