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Volumn 43, Issue 2, 2000, Pages 190-198

A potential melanoma tracer: Synthesis, radiolabeling, and biodistribution in mice of a new nitridotechnetium bis(aminothiol) derivative pharmacomodulated by a N-(diethylaminoethyl)benzamide

Author keywords

[No Author keywords available]

Indexed keywords

BENZAMIDE DERIVATIVE; NITRIDOTECHNETIUM BIS(AMINOTHIOL); RADIOPHARMACEUTICAL AGENT; TRACER; UNCLASSIFIED DRUG;

EID: 0034719436     PISSN: 00222623     EISSN: None     Source Type: Journal    
DOI: 10.1021/jm981089a     Document Type: Article
Times cited : (21)

References (43)
  • 1
    • 0000757256 scopus 로고
    • Epidemiology on malignant melanoma in Europe
    • Osterlind, A. Epidemiology on malignant melanoma in Europe. Rev. Oncol. 1992, 5, 903.
    • (1992) Rev. Oncol. , vol.5 , pp. 903
    • Osterlind, A.1
  • 6
    • 0343172534 scopus 로고    scopus 로고
    • La mortalité par cancer en France
    • Hill, C.; Doyon, F. La mortalité par cancer en France. Med. Sci. 1997, 13, 172-175.
    • (1997) Med. Sci. , vol.13 , pp. 172-175
    • Hill, C.1    Doyon, F.2
  • 14
    • 0032474746 scopus 로고    scopus 로고
    • Substitued halogenated arylsulfonamides: A new class of σ receptor binding tumor imaging agents
    • John, C. S.; Lim, B. B.; Vilner, B. J.; Geyer, B. C.; Bowen, W. D. Substitued halogenated arylsulfonamides: a new class of σ receptor binding tumor imaging agents. J. Med. Chem. 1998, 41, 2445-2450.
    • (1998) J. Med. Chem. , vol.41 , pp. 2445-2450
    • John, C.S.1    Lim, B.B.2    Vilner, B.J.3    Geyer, B.C.4    Bowen, W.D.5
  • 15
    • 0027141936 scopus 로고
    • A malignant melanoma imaging agent: Synthesis, characterization, in vitro binding and biodistribution of iodine-125-(2-piperidinylaminoethyl)4-iodobenzamide
    • John, C. S.; Bowen, W. D.; Saga, T.; Kinuya, S.; Vilner, B. J.; Baumgold, J.; Paik, C. H.; Reba, R. C.; Neuman, R. D.; Varma, V. M.; McAfee, J. G. A malignant melanoma imaging agent: synthesis, characterization, in vitro binding and biodistribution of iodine-125-(2-piperidinylaminoethyl)4-iodobenzamide. J. Nucl. Med. 1993, 34, 2169-2175.
    • (1993) J. Nucl. Med. , vol.34 , pp. 2169-2175
    • John, C.S.1    Bowen, W.D.2    Saga, T.3    Kinuya, S.4    Vilner, B.J.5    Baumgold, J.6    Paik, C.H.7    Reba, R.C.8    Neuman, R.D.9    Varma, V.M.10    McAfee, J.G.11
  • 17
    • 0028795145 scopus 로고
    • Sigma-1 and sigma-2 receptors are expressed in a wide variety of human and rodent tumor cell lines
    • Vilner, B. J.; John, C. S.; Bowen, W. D. Sigma-1 and sigma-2 receptors are expressed in a wide variety of human and rodent tumor cell lines. Cancer Res. 1995, 55, 408-413.
    • (1995) Cancer Res. , vol.55 , pp. 408-413
    • Vilner, B.J.1    John, C.S.2    Bowen, W.D.3
  • 20
    • 0032919295 scopus 로고    scopus 로고
    • In vitro studies on the cellular uptake of melanoma imaging aminoalkyl-iodobenzamide derivatives (ABA)
    • Dittman, H.; Coenen, H. H.; Zölzer, P.; Dutschka, K.; Brandau, W.; Streffer, C. In vitro studies on the cellular uptake of melanoma imaging aminoalkyl-iodobenzamide derivatives (ABA). Nucl. Med. Biol. 1999, 26, 51-56.
    • (1999) Nucl. Med. Biol. , vol.26 , pp. 51-56
    • Dittman, H.1    Coenen, H.H.2    Zölzer, P.3    Dutschka, K.4    Brandau, W.5    Streffer, C.6
  • 21
    • 0001594875 scopus 로고
    • Dialkylaminoalkyl-4-iodobenzamides: Influence of specific activity and substituents on melanoma uptake and biodistribution
    • Nicholl, C.; Mohammed, A.; Eisenhut, M. Dialkylaminoalkyl-4-iodobenzamides: Influence of specific activity and substituents on melanoma uptake and biodistribution. J. Labelled Compd. Radiopharm. 1995, 37, 277-279.
    • (1995) J. Labelled Compd. Radiopharm. , vol.37 , pp. 277-279
    • Nicholl, C.1    Mohammed, A.2    Eisenhut, M.3
  • 22
    • 0001294083 scopus 로고    scopus 로고
    • Potential technetium small molecule radiopharmaceuticals
    • Jurisson, S. S.; Lydon, J. D. Potential technetium small molecule radiopharmaceuticals. Chem. Rev. 1999, 99, 2205-2218.
    • (1999) Chem. Rev. , vol.99 , pp. 2205-2218
    • Jurisson, S.S.1    Lydon, J.D.2
  • 23
    • 0008883289 scopus 로고    scopus 로고
    • 99mTc-labeled small peptides as diagnostic radiopharmaceuticals
    • 99mTc-labeled small peptides as diagnostic radiopharmaceuticals. Chem. Rev. 1999, 99, 2235-2268.
    • (1999) Chem. Rev. , vol.99 , pp. 2235-2268
    • Liu, S.1    Edwards, D.S.2
  • 24
    • 0030808619 scopus 로고    scopus 로고
    • Technetium-99m-labeled receptor-specific small-molecule radiopharmaceuticals: Recent developments and encouraging results
    • Hom, R. K.; Katzenellengogen, J. A. Technetium-99m-labeled receptor-specific small-molecule radiopharmaceuticals: recent developments and encouraging results. Nucl. Med. Biol. 1997, 24, 485-498.
    • (1997) Nucl. Med. Biol. , vol.24 , pp. 485-498
    • Hom, R.K.1    Katzenellengogen, J.A.2
  • 28
    • 0000939490 scopus 로고
    • Conversion of esters to amides with dimethylaluminium amides: N,N-dimethylcyclohexanecarboxamide
    • John Wiley & Sons: New York
    • Lipton, M. F.; Basha, A.; Weinreb, M. Conversion of esters to amides with dimethylaluminium amides: N,N-dimethylcyclohexanecarboxamide. Organic syntheses; John Wiley & Sons: New York, 1988; Vol. 6, pp 492-495.
    • (1988) Organic Syntheses , vol.6 , pp. 492-495
    • Lipton, M.F.1    Basha, A.2    Weinreb, M.3
  • 29
    • 0001528499 scopus 로고
    • Transannular cyclisation of 1,2-dithia-5,8-diazacyclodeca-4,8-dienes during borohydride reduction
    • Joshua, A. V.; Scott, J. R.; Sondhi, S. M.; Ball, R. G.; Lown, J. W. Transannular cyclisation of 1,2-dithia-5,8-diazacyclodeca-4,8-dienes during borohydride reduction. J. Org. Chem. 1987, 52, 2447-2451.
    • (1987) J. Org. Chem. , vol.52 , pp. 2447-2451
    • Joshua, A.V.1    Scott, J.R.2    Sondhi, S.M.3    Ball, R.G.4    Lown, J.W.5
  • 31
    • 0026014547 scopus 로고
    • Synthesis of technetium-99m labeled diaminodithiol for bifunctional chelating agent
    • Shiba, K.; Mori, H.; Matsuda, H.; Tsuji, S.; Kinuya, K.; Hisada, K.; Synthesis of technetium-99m labeled diaminodithiol for bifunctional chelating agent. Appl. Radiat. Isot. 1991, 42, 1159-1164.
    • (1991) Appl. Radiat. Isot. , vol.42 , pp. 1159-1164
    • Shiba, K.1    Mori, H.2    Matsuda, H.3    Tsuji, S.4    Kinuya, K.5    Hisada, K.6
  • 32
    • 0024332355 scopus 로고
    • 99mTc-glucoheptonate and N-benzyl-N-methylpiperazinyl-bis-(aminoethanethiol) (BPA-BAT)
    • 99mTc-glucoheptonate and N-benzyl-N-methylpiperazinyl-bis-(aminoethanethiol) (BPA-BAT). Appl. Radiat. Isot. 1989, 40, 677-681.
    • (1989) Appl. Radiat. Isot. , vol.40 , pp. 677-681
    • Kung, H.F.1    Liu, B.L.2    Pan, S.3
  • 35
    • 0026016432 scopus 로고
    • A new method for the preparation of Tc-99m radiopharmaceuticals containing the Tc≡ N multiple bond. Eighth international symposium on radiopharmaceutical chemistry abstracts
    • Duatti, A.; Marchi, A.; Pasqualini, R. A new method for the preparation of Tc-99m radiopharmaceuticals containing the Tc≡ N multiple bond. Eighth international symposium on radiopharmaceutical chemistry abstracts. J. Labelled Compds. Radiopharm. 1991, 30, 13.
    • (1991) J. Labelled Compds. Radiopharm. , vol.30 , pp. 13
    • Duatti, A.1    Marchi, A.2    Pasqualini, R.3
  • 38
    • 37049107411 scopus 로고
    • Studies of technetium complexes. Part 6. The preparation, characterisation, and electron spin resonance spectra of salts of tetrachloroand tetrabromo-nitridotechnetate(vi): Crystal structure of tetraphenyl-arsonium tetrachloro-nitridotechnetate(vi)
    • Baldas, J.; Boas, J. F.; Bonnyman, J.; Williams, G. A. Studies of technetium complexes. Part 6. The preparation, characterisation, and electron spin resonance spectra of salts of tetrachloroand tetrabromo-nitridotechnetate(vi): crystal structure of tetraphenyl-arsonium tetrachloro-nitridotechnetate(vi). J. Chem. Soc., Dalton Trans. 1984, 2395-2400.
    • (1984) J. Chem. Soc., Dalton Trans. , pp. 2395-2400
    • Baldas, J.1    Boas, J.F.2    Bonnyman, J.3    Williams, G.A.4
  • 39
    • 0028062169 scopus 로고
    • Technetium-99m N,N′-bis-(2-mercapto-2-methylpropyl)-2-aminobenzylamine: Technetium-99m complexes of a novel bis(aminoethanethiol) ligand
    • Francesconi, L. C.; Yang, Y. Y.; Kung, M.-P.; Zhang, X. X.; Billings, J.; Guo, Y. Z.; Kung, H. F. Technetium-99m N,N′-bis-(2-mercapto-2-methylpropyl)-2-aminobenzylamine: technetium-99m complexes of a novel bis(aminoethanethiol) ligand. J. Med. Chem. 1994, 37, 3282-3288.
    • (1994) J. Med. Chem. , vol.37 , pp. 3282-3288
    • Francesconi, L.C.1    Yang, Y.Y.2    Kung, M.-P.3    Zhang, X.X.4    Billings, J.5    Guo, Y.Z.6    Kung, H.F.7
  • 40
    • 0003879532 scopus 로고
    • Structural aspects of technetium nitrido complexes
    • Nicolini, M., Bandoli, G., Mazzi, U., Eds.; Cortinal International-Verona Raven Press: New York
    • Colmanet, S. F.; Williams, G. A. Structural aspects of technetium nitrido complexes. In Technetium and Rhenium in Chemistry and Nuclear Medicine; Nicolini, M., Bandoli, G., Mazzi, U., Eds.; Cortinal International-Verona Raven Press: New York, 1990; Vol. 3, pp 55-62.
    • (1990) Technetium and Rhenium in Chemistry and Nuclear Medicine , vol.3 , pp. 55-62
    • Colmanet, S.F.1    Williams, G.A.2
  • 41
    • 37049067740 scopus 로고
    • Formation of the Tc=N multiple bond from the reaction of ammonium pertechnetate with S-methyl dithiocarbazate and its application to the preparation of technetium-99m radiopharmaceuticals
    • Duatti, A.; Marchi, A.; Pasqualini, R. Formation of the Tc=N multiple bond from the reaction of ammonium pertechnetate with S-methyl dithiocarbazate and its application to the preparation of technetium-99m radiopharmaceuticals. J. Chem. Soc., Dalton Trans. 1990, 3729-3733.
    • (1990) J. Chem. Soc., Dalton Trans. , pp. 3729-3733
    • Duatti, A.1    Marchi, A.2    Pasqualini, R.3


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