Characterisation of calcitonin gene-related peptide receptors in rat atrium and vas deferens: Evidence for a (Cys(Et)2,7)hCGRP-preferring receptor

European Journal of Pharmacology

Volumn 400, Issue 2-3, 2000, Pages 313-319

  Wu, Dongmei ^a   Eberlein, Wolfgang ^a   Rudolf, Klaus ^a   Engel, Wolfhard ^a   Hallermayer, Gerhard ^a   Doods, Henri ^a  

^a BOEHRINGER INGELHEIM PHARMA GMBH AND CO KG   (Germany)

Author keywords

BIBN4096BS; Calcitonin gene related peptide (CGRP); CGRP (8 38); CGRP receptor subtypes; Left atrium, rat; Vas deferens, rat

Indexed keywords

ADRENOMEDULLIN; CALCITONIN GENE RELATED PEPTIDE; CALCITONIN GENE RELATED PEPTIDE DERIVATIVE; CALCITONIN GENE RELATED PEPTIDE RECEPTOR; N [2 [[5 AMINO 1 [[4 (4 PYRIDYL) 1 PIPERAZINYL]CARBONYL]PENTYL]AMINO] 1 [(3,5 DIBROMO 4 HYDROXYPHENYL)ETHYL] 4 (1,4 DIHYDRO 2 OXO 3(2H) QUINAZOLINYL) 1 PIPERIDINECARBOXAMIDE; OLCEGEPANT; RECEPTOR BLOCKING AGENT; RECEPTOR SUBTYPE; THIORPHAN; UNCLASSIFIED DRUG;

ANIMAL TISSUE; ARTICLE; BINDING AFFINITY; CONTROLLED STUDY; DOSE RESPONSE; DRUG RECEPTOR BINDING; ELECTROSTIMULATION; HEART LEFT ATRIUM; IN VITRO STUDY; MALE; NONHUMAN; PRIORITY JOURNAL; RAT; SMOOTH MUSCLE CONTRACTILITY; VAS DEFERENS;

ANIMALS; CALCITONIN GENE-RELATED PEPTIDE; CARDIOTONIC AGENTS; HEART ATRIA; HUMANS; KINETICS; MALE; MYOCARDIUM; PEPTIDE FRAGMENTS; PIPERAZINES; PROTEASE INHIBITORS; QUINAZOLINES; RATS; RATS, WISTAR; RECEPTORS, CALCITONIN GENE-RELATED PEPTIDE; THIORPHAN; VAS DEFERENS;

EID: 0034698365     PISSN: 00142999     EISSN: None     Source Type: Journal    
DOI: 10.1016/S0014-2999(00)00407-6     Document Type: Article

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