Synthesis and in vivo evaluation of [11C]ICI 118551 as a putative subtype selective β2-adrenergic radioligand

International Journal of Pharmaceutics

Volumn 204, Issue 1-2, 2000, Pages 101-109

  Moresco, R M ^a   Matarrese, M ^a   Soloviev, D ^a   Simonelli, P ^a   Rigamonti, M ^a   Gobbo, C ^a   Todde, S ^a   Carpinelli, A ^a   Galli Kienle, M ^a,b   Fazio, F ^a  

^a UNIVERSITY OF MILANO BICOCCA   (Italy)

^b SAN RAFFAELE HOSPITAL   (Italy)

Author keywords

2 Adrenergic receptors; ( ) 11C ICI 118551; Emission tomography; Monkeys; Rats

Indexed keywords

3 ISOPROPYLAMINO 1 (7 METHYL 4 INDANYLOXY) 2 BUTANOL; BETA ADRENERGIC RECEPTOR; BETA ADRENERGIC RECEPTOR BLOCKING AGENT; CARBON 11; FORMOTEROL; PROPRANOLOL; TRACER;

ANIMAL CELL; ANIMAL MODEL; ANIMAL TISSUE; ARTICLE; BETA ADRENERGIC RECEPTOR BLOCKING; CONTROLLED STUDY; DRUG RECEPTOR BINDING; DRUG SYNTHESIS; IMAGE ANALYSIS; ISOTOPE LABELING; MACACA; MALE; NONHUMAN; POSITRON EMISSION TOMOGRAPHY; PRIORITY JOURNAL; RADIOCHEMISTRY; RADIODIAGNOSIS; RAT;

ADRENERGIC BETA-ANTAGONISTS; ANIMAL; CARBON RADIOISOTOPES; FEMALE; LUNG; MACACA NEMESTRINA; MALE; PROPANOLAMINES; RATS; RECEPTORS, ADRENERGIC, BETA-2; TISSUE DISTRIBUTION; TOMOGRAPHY, EMISSION-COMPUTED;

EID: 0034690946     PISSN: 03785173     EISSN: None     Source Type: Journal    
DOI: 10.1016/S0378-5173(00)00480-4     Document Type: Article

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