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Bioorganic and Medicinal Chemistry Letters

Volumn 10, Issue 20, 2000, Pages 2305-2309

Novel, potent and selective chimeric FXa inhibitors featuring hydrophobic P1-ketoamide moieties

(5) Semple, J Edward a Levy, Odile E a Minami, Nathaniel K a Owens, Timothy D a Siev, Daniel V a

a Dendreon (United States)

Author keywords

[No Author keywords available]

Indexed keywords

ANTICOAGULANT PROTEIN; ANTISTASIN; BLOOD CLOTTING FACTOR 10A INHIBITOR; ECOTIN; SERINE PROTEINASE; UNCLASSIFIED DRUG;

ARTICLE; CHEMICAL REACTION; DRUG POTENCY; DRUG SELECTIVITY; DRUG SYNTHESIS; HYDROPHOBICITY; PHARMACOPHORE; REACTION ANALYSIS; STRUCTURE ACTIVITY RELATION;

ANTIFIBRINOLYTIC AGENTS; BACTERIAL PROTEINS; CHIMERIC PROTEINS; DRUG DESIGN; FACTOR XA; HELMINTH PROTEINS; HUMAN; INVERTEBRATE HORMONES; MOLECULAR STRUCTURE; SERINE PROTEINASE INHIBITORS; STRUCTURE-ACTIVITY RELATIONSHIP;

EID: 0034675818 PISSN: 0960894X EISSN: None Source Type: Journal
DOI: 10.1016/S0960-894X(00)00458-3 Document Type: Article

Times cited : (20)

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