A modified Backbone Amide Linker (BAL) solid-phase peptide synthesis strategy accommodating prolyl, N-alkylamino acyl, or histidyl derivatives at the C-terminus

Tetrahedron Letters

Volumn 41, Issue 38, 2000, Pages 7277-7280

  Alsina, Jordi ^a   Yokum, T Scott ^a   Albericio, Fernando ^b   Barany, George ^a  

^a University of Minnesota ^*  (United States)

^b UNIVERSITY OF BARCELONA   (Spain)

Author keywords

Backbone amide linker; C terminal modified peptides; Diketopiperazines; Histidine; Proline; PyBOP; Racemization

Indexed keywords

9 FLUORENYLMETHYL CHLOROFORMATE; ALIPHATIC AMINE; HISTIDINE DERIVATIVE; PIPERAZINEDIONE; PROLINE DERIVATIVE;

ARTICLE; CARBOXY TERMINAL SEQUENCE; CHEMICAL MODIFICATION; CHIRALITY; ESTERIFICATION; MOLECULAR MODEL; PEPTIDE SYNTHESIS;

EID: 0034675389     PISSN: 00404039     EISSN: None     Source Type: Journal    
DOI: 10.1016/S0040-4039(00)01255-7     Document Type: Article

References (21)