An alternate preparation of thioester resin linkers for solid-phase synthesis of peptide C-terminal thioacids

Tetrahedron Letters

Volumn 41, Issue 16, 2000, Pages 2797-2800

  Goldstein, Alex S ^a   Gelb, Michael H ^a  

^a UNIVERSITY OF WASHINGTON   (United States)

Author keywords

Peptide analogues mimetics; Supported reagents reactions; Thioacids; Thioesters; Thiopeptides

Indexed keywords

RESIN; THIOACID; THIOESTER;

ARTICLE; CARBOXY TERMINAL SEQUENCE; CHEMICAL REACTION; REACTION ANALYSIS; SYNTHESIS;

EID: 0034655782     PISSN: 00404039     EISSN: None     Source Type: Journal    
DOI: 10.1016/S0040-4039(00)00266-5     Document Type: Article

References (7)

1. Blake, J.; Li, C. H. Proc. Natl. Acad. Sci. USA 1981, 78, 4055-4058.
2. Schnolzer, M.; Kent, S. B. H. Science 1992, 256, 221-225.
3. Canne, L. E.; Walker, S. M.; Kent, S. B. H. Tetrahedron Lett. 1995, 38, 1217-1220.
4. Yamashiro, D.; Li, C. H. Int. J. Peptide Protein Res. 1988, 31, 322-334.
5. Gauthier, J. Y.; Bourdon, F.; Young, R. N. Tetrahedron Lett. 1986, 27, 15-18.
6. 1H NMR to their oxyacid analogues.
7. 1H NMR are identical to the superimposition of the N-BOC-aminothioacid with 4-benzoylphenoxyacetic acid (3).