Inhibition of bacterial peptide deformylase by biaryl acid analogs

Archives of Biochemistry and Biophysics

Volumn 375, Issue 2, 2000, Pages 355-358

  Green, Barbara Gordon ^a   Toney, Jeffrey H ^a   Kozarich, John W ^a   Grant, Stephan K ^a  

^a MERCK RESEARCH LABORATORIES   (United States)

Author keywords

Biaryl acid analogs; Enzyme inhibitors; Metallo lactamase; Peptide deformylase

Indexed keywords

BACTERIAL ENZYME; BETA LACTAMASE; CARBONATE DEHYDRATASE; CARBOXYLIC ACID DERIVATIVE; ENZYME INHIBITOR; METHIONINE DERIVATIVE; PEPTIDE DEFORMYLASE; SULFONAMIDE; TETRAZOLE DERIVATIVE; UNCLASSIFIED DRUG;

ARTICLE; COMPETITIVE INHIBITION; CONTROLLED STUDY; DRUG ACTIVITY; DRUG STRUCTURE; ENZYME INHIBITION; PHARMACOPHORE; PRIORITY JOURNAL; PROTEIN PROCESSING; STRUCTURE ACTIVITY RELATION;

BACTERIA (MICROORGANISMS); BACTEROIDES FRAGILIS; ESCHERICHIA COLI;

EID: 0034654564     PISSN: 00039861     EISSN: None     Source Type: Journal    
DOI: 10.1006/abbi.1999.1673     Document Type: Article

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