Glucuronide and sulfate conjugates of ICI 182,780, a pure anti- estrogenic steroid. Order of addition, catalysis and substitution effects in glucuronidation

Tetrahedron Letters

Volumn 41, Issue 3, 2000, Pages 389-392

  Ferguson, John R ^a   Harding, John R ^b   Lumbard, Keith W ^a   Scheinmann, Feodor ^a   Stachulski, Andrew V ^a  

^a Ultrafine UFC Ltd   (United Kingdom)

^b ASTRAZENECA   (United Kingdom)

Author keywords

[No Author keywords available]

Indexed keywords

FULVESTRANT; GLUCURONIDE; SULFATE;

ARTICLE; BREAST CANCER; CATALYSIS; DRUG ACTIVITY; DRUG GLUCURONIDATION; DRUG STRUCTURE; DRUG SYNTHESIS;

EID: 0034650680     PISSN: 00404039     EISSN: None     Source Type: Journal    
DOI: 10.1016/S0040-4039(99)02067-5     Document Type: Article

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3. Tsuneda, K.; Yamada, J.; Yasuda, K.; Mori, H. Chem. Pharm. Bull. Jpn. 1963, 11, 510.
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12. 1H NMR and high resolution FAB mass spectra were also obtained for 4 and 5.