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Ojima, I.1
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(a) Reviews: Iseki, K. Tetrahedron 1998, 54, 13887.
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Tetrahedron
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Iseki, K.; Oishi, S.; Sasai, H.; Shibasaki, M. Tetrahedron Lett. 1996,37,9081.
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Mikami, K.; Yajima, T.; Takasaki, T.; Matsukawa, S.; Terada, M.; Uchimaru, T.; Manila, M. Tetrahedron 1996, 52, 85.
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(1996)
Tetrahedron
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Mikami, K.1
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Terada, M.5
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Manila, M.7
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7591.
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(e) Mikami, K.; Yajima, T.; Terada, M.; Uchimaru, T. Tetrahedron Lett. 1993,34,7591.
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(1993)
Tetrahedron Lett.
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Mikami, K.1
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(b) Heaney, H. In Comprehensive Organic Synthesis; Trost, B. M., Fleming, I., Eds.; Pergamon Press: Oxford, 1991; Vol. 2, p 733.
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(1991)
Comprehensive Organic Synthesis; Trost, B. M., Fleming, I., Eds.; Pergamon Press: Oxford
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Heaney, H.1
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16
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0030817245
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Diastereoselective F-C type reaction: (a) Costa, P. R. R.; Cabrai, L. M.; Alencar, K. G.; Schmidt, L. L.; Vasconcellos, M. L. A. A. Tetrahedron Lett. 1997,38, 7021.
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(1997)
Tetrahedron Lett.
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Costa, P.R.R.1
Cabrai, L.M.2
Alencar, K.G.3
Schmidt, L.L.4
Vasconcellos, M.L.A.A.5
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(b) El Kaim, L.; Guyoton, S.; Meyer, C. Tetrahedron Lett. 1996,37, 375.
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(1996)
Tetrahedron Lett.
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El Kaim, L.1
Guyoton, S.2
Meyer, C.3
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18
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0027135611
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and references therein. Double asymmetric synthesis: (d) Terada, M.; Sayo, N.; Mikami, K. Synlett 1995, 411.
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Bigi, F.; Sartori, G.; Maggi, R.; Cantarelli, E.; Galavema, G. Tetrahedron: Asymmetry 1993,4, 2411, and references therein. Double asymmetric synthesis: (d) Terada, M.; Sayo, N.; Mikami, K. Synlett 1995, 411.
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(1993)
Tetrahedron: Asymmetry
, vol.4
, pp. 2411
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Bigi, F.1
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Cantarelli, E.4
Galavema, G.5
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19
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0000582255
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Pictet-Spengler reaction: 0 Cox, E. D.; Hameker, L. K.; Li, J.; Yu, P.; Czerwinski, K. M.; Deng, L.; Bennett. D. W.; Cook, J. M. J. Org. Chem. 1997, 62, 44.
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(e) Casiraghi, G.; Bigi, F.; Casnati, G.; Sartori, G.; Soncini, P.; Gasparri Fava, G.; Ferrari Belicchi, M. 'J. Org. Chem. 1988, 53, 1779. Pictet-Spengler reaction: (0 Cox, E. D.; Hameker, L. K.; Li, J.; Yu, P.; Czerwinski, K. M.; Deng, L.; Bennett. D. W.; Cook, J. M. J. Org. Chem. 1997, 62, 44.
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Ferrari Belicchi, M.7
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(g) Dai, W.M.; Zhu, H. J.; Hao, X.-J. Tetrahedron Lett. 1996, 37, 5971.
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Dai, W.M.1
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(h) Soe, T.; Kawate, T.; Fukui, N.; Hino, T.; Nakagawa, M. Heterocycles 1996, 42, 347.
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Soe, T.1
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Nakagawa, M.5
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22
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33748216328
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Enantioselective F-C type reaction: (a) Erker, G.; van der Zeijden, A. A. H. Angeiv. Chem., Int. Ed. Engl. 1990,29, 512.
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(1990)
Angeiv. Chem., Int. Ed. Engl.
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Erker, G.1
Van Der Zeijden, A.A.H.2
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33845378131
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Pictet-Spengler reaction: (c) Kawate, T.; Yamada, H.; Soe, T.; Nakagawa, M. Tetrahedron: Asymmetry 1996, 7, 1249.
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(b) Bigi, F.; Casiraghi, G.; Casnati, G.; Sartori, G.; Gasparri Fava, G.; Ferrari Belicchi, M. J. Org. Chem. 1985, 50, 5018. Pictet-Spengler reaction: (c) Kawate, T.; Yamada, H.; Soe, T.; Nakagawa, M. Tetrahedron: Asymmetry 1996, 7, 1249.
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J. Org. Chem.
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Bigi, F.1
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Sartori, G.4
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Ferrari Belicchi, M.6
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(b) Muehldorf, A. V.; Guzman-Perez, A.; Kluge, A. F. Tetrahedron Lett. 1994, 35, 8755.
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Muehldorf, A.V.1
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27
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33751499929
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and references therein, (c) Corey, E. J.; Cheng, X.-M.; Cimprich, K A.; Sarshar, S. Tetrahedron Lett. 1991,32,6835.
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(b) Chong, J. M.; Mar, E. K. J. Org. Chem. 1991,56,893, and references therein, (c) Corey, E. J.; Cheng, X.-M.; Cimprich, K A.; Sarshar, S. Tetrahedron Lett. 1991,32,6835.
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Mar, E.K.2
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Ramachandran, P. V.; Teodorovic, A. V.; Gong, B.; Brown, H. C. Tetrahedron: Asymmetry 1994,5, 1075.
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Tetrahedron: Asymmetry
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Brown, H.C.4
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(e) Fujisawa, T.; Sugimoto, T.; Shimizu, M. Tetrahedron: Asymmetry 1994, 5, 1095.
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(1994)
Tetrahedron: Asymmetry
, vol.5
, pp. 1095
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84989546359
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(b) Mikami, K; Terada, M.; Narisawa, S.; Nakai, T. Synlett 1992, 255.
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Synlett
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Mikami, K.1
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1989, 111, 1940; Mikami, K.; Terada, M.; Narisawa, S.; Nakai, T. Org. Synth. 1993, 71, 14.
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Mikami, K.; Terada, M.; Nakai, T. J. Am. Chem. Soc. 1990,112, 3949; 1989, 111, 1940; Mikami, K.; Terada, M.; Narisawa, S.; Nakai, T. Org. Synth. 1993, 71, 14.
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Mikami, K.1
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37
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0042732610
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[a]20D -35.9' (c 1.35, EtOH) for 80.2% ee of R isomer.
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Ohno, A.; Nakai, J.; Nakamura, K.; Goto, T.; Oka, S. Bull. Chem. Soc. Jpn., 1981,54,3486 [a]20D -35.9' (c 1.35, EtOH) for 80.2% ee of R isomer.
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(1981)
Bull. Chem. Soc. Jpn.
, vol.54
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Ohno, A.1
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Corey, E. J.; Barnes-Seeman, D.; Lee, T. W.; Goodman, S. N. Tetrahedron Lett. 1997, 37, 6513.
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Corey, E.J.1
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39
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0031575791
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(a) Mikami, K.; Matsukawa, S.; Sawa, E.; Harada, A.; Koga, N. Tetrahedron Lett. 1997, 38, 1951.
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(1997)
Tetrahedron Lett.
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40
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0031031933
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and references therein.
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(b) Mikami, K.; Matsukawa, S.; Nagashima, M.; Funabashi, H.; Morishima, H. Tetrahedron Lett. 1997, 38, 579, and references therein.
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(1997)
Tetrahedron Lett.
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Mikami, K.1
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Funabashi, H.4
Morishima, H.5
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41
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33847569967
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note
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The same reaction in the presence of YhCOTffo (10 mol %) gave the F-C products in 78% yield (para/ortho = 7). The addition of (R)6,6'-Br2-BINOL (1 or 2 equiv) decreased the chemical yields (42% (para/ ortho = 13) or 45% (paralortho = 16), respectively).
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