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Tetrahedron Letters

Volumn 41, Issue 41, 2000, Pages 7837-7841

Design and synthesis of histone deacetylase inhibitors: The development of apicidin transition state analogs

(7) Colletti, Steven L a Myers, Robert W a Darkin Rattray, Sandra J a Schmatz, Dennis M a Fisher, Michael H a Wyvratt, Matthew J a Meinke, Peter T a

a MERCK RESEARCH LABORATORIES (United States)

Author keywords

Apicidin; Histone deacetylase; Side chain; Transition state inhibitors

Indexed keywords

APICIDIN; APICIDIN DERIVATIVE; ENZYME INHIBITOR; HISTONE DEACETYLASE; UNCLASSIFIED DRUG;

ARTICLE; CHEMICAL ANALYSIS; CHEMICAL REACTION; CHEMICAL STRUCTURE; DRUG DESIGN; DRUG SYNTHESIS;

EID: 0034619133 PISSN: 00404039 EISSN: None Source Type: Journal
DOI: 10.1016/S0040-4039(00)01366-6 Document Type: Article

Times cited : (19)

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