Unique sodium-caged structure of a potent endothelin-1 inhibitor: Crystal structure of BQ123 sodium salt, cyclo(-D-Trp-D-Asp--Pro-D-Val-Leu- )·Na+

Chemical Communications

Volumn , Issue 9, 2000, Pages 743-744

  Doi, Mitsunobu ^a   Ishida, Toshimasa ^a   Katsuya, Yoshio ^b   Mezaki, Yoshihiro ^b   Sasaki, Masahiro ^c   Terashima, Akira ^c   Taniguchi, Taizo ^c   Hasegawa, Hiroshi ^c   Shiono, Masaaki ^d  

^a OSAKA MEDICAL COLLEGE   (Japan)

^b Hyogo Prefectural Institute of Industrial Research Technical Center for Machinery and Metals   (Japan)

^c Hyogo Inst Aging Brain Cogn D   (Japan)

^d KYUSHU UNIVERSITY   (Japan)

Author keywords

[No Author keywords available]

Indexed keywords

CYCLO(DEXTRO TRYPTOPHYL DEXTRO ASPARTYLPROLYL DEXTRO VALYLLEUCYL); ENDOTHELIN 1; ENDOTHELIN RECEPTOR ANTAGONIST; SODIUM;

ARTICLE; CRYSTAL STRUCTURE; NUCLEAR MAGNETIC RESONANCE; X RAY DIFFRACTION;

EID: 0034616505     PISSN: 13597345     EISSN: None     Source Type: Journal    
DOI: 10.1039/a909413j     Document Type: Article

References (15)

1. M. Yanagisawa, H. Kurihara, S. Kimura, Y. Tombe, M. Kobayashi, Y. Mitsui, Y. Yazaki, K. Goto and T. Masaki, Nature (London), 1988, 332, 411.
2. K. Kojiri, M. Ihara, S. Nakajima, K. Kawamura, K. Funaishi, M. Yano and H. Suda, J. Antibiot., 1991, 44, 1342.
3. S. Nakajima, K. Niiyama, M. Ihara, K. Kojiri and H. Suda, J. Antibiot., 1991, 44, 1348.
4. K. Ishikawa, T. Fukami, T. Nagase, K. Fujita, T. Hayama, K. Niiyama, T. Mase, M. Ihara and M. Yano, J. Med. Chem., 1992, 35, 2139.
5. M. Ihara, K. Noguchi, T. Saeki, T. Fukuroda, S. Tsuchida, S. Kimura, T. Fukami, K. Ishikawa, M. Nishikibe and M. Yano, Life Sci., 1992, 50, 247.
6. T. Fukami, T. Nagase, K. Fujita, T. Hayama, K. Niiyama, T. Mase, S. Nakajima, T. Fukuroda, T. Saeki, M. Nishikibe, M. Ihara, M. Yano and K. Ishikawa, J. Med. Chem., 1995, 38, 4309.
7. S. Endo, H. Inooka, Y. Ishibashi, C. Kitada, E. Mizuta and M. Fujino, FEBS Lett., 1989, 257, 149.
8. V. Saudek, J. Hoflack and J. T. Pelton, Int. J. Pept. Protein Res., 1991, 37, 174.
9. M. Coles, V. Sowemimo, D. Scanlon, S. L. Munro and D. J. Craik, J. Med. Chem., 1993, 36, 2658.
10. J. W. Bean, C. E. Peishoff and K. D. Kopple, Int. J. Pept. Protein Res., 1994, 44, 223.
11. C. E. Peishoff, R. W. Janes and B. A. Wallace, FEBS Lett., 1995, 374, 379.
12. M. Wolff, J. Day, A. Greenwood, S. Larson and A. McPherson, Acta Crystallogr. Sect. B, 1992, 48, 239.
13. R. W. Janes, D. H. Peapus and B. A. Wallace, Nat. Struct. Biol., 1997, 1, 311.
14. N. Matsugaki and M. Shiono, LODEM, A Density Modification Program for ab initio Solution of Crystal Structures from X-ray Diffraction Data, Kyushu University, Kyushu, 1998.
15. G. M. Sheldrick, SHELXL-97. Program for the Refinement of Crystal Structures from Diffraction Data. University of Göttingen, Göttingen, 1997.