-
3
-
-
2842532892
-
-
For reviews of tetrazole chemistry see: (a) Moderhack, D. J. Prakt. Chem. 1998, 340, 687-709.
-
(1998)
J. Prakt. Chem.
, vol.340
, pp. 687-709
-
-
Moderhack, D.1
-
4
-
-
84944045553
-
-
Katrinsky, A. R., Rees, C. W., Scriven, E. F. V., Eds.; Pergamon Press: New York
-
(b) Butler, R. N. Comprehensive Heterocyclic Chem. II; Katrinsky, A. R., Rees, C. W., Scriven, E. F. V., Eds.; Pergamon Press: New York, 1996; Vol. 4; pp 621-678.
-
(1996)
Comprehensive Heterocyclic Chem. II
, vol.4
, pp. 621-678
-
-
Butler, R.N.1
-
6
-
-
84943405513
-
-
Potts, K. T., Ed.; Pergamon Press: New York
-
(d) Butler, R. N. Comprehensive Heterocyclic Chemistry; Potts, K. T., Ed.; Pergamon Press: New York, 1984; Vol 5; pp 791-838.
-
(1984)
Comprehensive Heterocyclic Chemistry
, vol.5
, pp. 791-838
-
-
Butler, R.N.1
-
7
-
-
10244252718
-
-
For a few recent examples, see (a) White, A. D.; Creswell, M. W.; Chucholowski, A. W.; Blankley, C. J.; Wilson, M. W.; Bousley, R. F.; Essenburg, A. D.; Hamelehle, K. L.; Krause, B. R.; Stanfield, R. L.; Dominick, M. A.; Neub, M. J. Med. Chem. 1996, 39, 4382-4395.
-
(1996)
J. Med. Chem.
, vol.39
, pp. 4382-4395
-
-
White, A.D.1
Creswell, M.W.2
Chucholowski, A.W.3
Blankley, C.J.4
Wilson, M.W.5
Bousley, R.F.6
Essenburg, A.D.7
Hamelehle, K.L.8
Krause, B.R.9
Stanfield, R.L.10
Dominick, M.A.11
Neub, M.12
-
8
-
-
0028054343
-
-
(b) Larsen, R. D.; King, A. O.; Chen, C. Y.; Corley, E. G.; Foster, B. S.; Roberts, F. E.; Yang, C.; Lieberman, D. R.; Reamer, R. A.; Tschaen, D. M.; Verhoeven, T. R.; Reider, P. J. J. Org. Chem. 1994, 59, 6391-6394.
-
(1994)
J. Org. Chem.
, vol.59
, pp. 6391-6394
-
-
Larsen, R.D.1
King, A.O.2
Chen, C.Y.3
Corley, E.G.4
Foster, B.S.5
Roberts, F.E.6
Yang, C.7
Lieberman, D.R.8
Reamer, R.A.9
Tschaen, D.M.10
Verhoeven, T.R.11
Reider, P.J.12
-
9
-
-
0026514079
-
-
Zabrocki, J.; Dunbar, J. B.; Marshall, K. W.; Toth, M. V.; Marshall, G. R. J. Org. Chem. 1992, 57, 202-209.
-
(1992)
J. Org. Chem.
, vol.57
, pp. 202-209
-
-
Zabrocki, J.1
Dunbar, J.B.2
Marshall, K.W.3
Toth, M.V.4
Marshall, G.R.5
-
10
-
-
0024548868
-
-
Lebl, M.; Slaninova, J.; Johnson, R. L. Int. J. Pept. Protein Res. 1990, 33, 16.
-
(1990)
Int. J. Pept. Protein Res.
, vol.33
, pp. 16
-
-
Lebl, M.1
Slaninova, J.2
Johnson, R.L.3
-
11
-
-
0032554967
-
-
(a) Satoh, Y.; De Lombaert, S.; Marcopulos, N.; Moliterni, J.; Moskal, M.; Tan, J.; Wallace, E. Tetrahedron Lett. 1998, 39, 3367-3370.
-
(1998)
Tetrahedron Lett.
, vol.39
, pp. 3367-3370
-
-
Satoh, Y.1
De Lombaert, S.2
Marcopulos, N.3
Moliterni, J.4
Moskal, M.5
Tan, J.6
Wallace, E.7
-
12
-
-
0029024034
-
-
(b) Beusen, D. D.; Zabrocki, J.; Slomczynska, U.; Head, R. D.; Kao, J. L. F.; Marshall, G. R. Biopolymers 1995, 36, 181-200.
-
(1995)
Biopolymers
, vol.36
, pp. 181-200
-
-
Beusen, D.D.1
Zabrocki, J.2
Slomczynska, U.3
Head, R.D.4
Kao, J.L.F.5
Marshall, G.R.6
-
14
-
-
0001432279
-
-
(d) Zabrocki, J.; Smith, G. D.; Dunbar, J. B.; Iijima, H.; Marshall, G. R. J. Am. Chem. Soc. 1988, 110, 5875-5880.
-
(1988)
J. Am. Chem. Soc.
, vol.110
, pp. 5875-5880
-
-
Zabrocki, J.1
Smith, G.D.2
Dunbar, J.B.3
Iijima, H.4
Marshall, G.R.5
-
16
-
-
0042189223
-
-
For other less general methods utilizing harsh conditions, see (a) Imhof, R.; Ladner, D. W.; Muchowski, J. M. J. Org. Chem. 1977, 42, 3709-3713.
-
(1977)
J. Org. Chem.
, vol.42
, pp. 3709-3713
-
-
Imhof, R.1
Ladner, D.W.2
Muchowski, J.M.3
-
17
-
-
0023128524
-
-
(b) Boyd, G. V.; Cobb, J.; Lindley, P. F.; Mitchell, J. C.; Nicolaou, G. A. J. Chem. Soc., Chem. Commun. 1987, 99-101.
-
(1987)
J. Chem. Soc., Chem. Commun.
, pp. 99-101
-
-
Boyd, G.V.1
Cobb, J.2
Lindley, P.F.3
Mitchell, J.C.4
Nicolaou, G.A.5
-
18
-
-
33845551620
-
-
(c) Gupton, J. T.; Idoux, J. P.; Baker, G.; Colon, C.; Crews, A. D.; Jurss, C. D.; Rampi, R. C. J. Org. Chem. 1983, 48, 2933-2936.
-
(1983)
J. Org. Chem.
, vol.48
, pp. 2933-2936
-
-
Gupton, J.T.1
Idoux, J.P.2
Baker, G.3
Colon, C.4
Crews, A.D.5
Jurss, C.D.6
Rampi, R.C.7
-
20
-
-
0030043963
-
-
(b) Castro, J. L.; Ball, R. G.; Broughton, H. B.; Russell, M. G. N.; Rathbone, D.; Watt, A. P.; Baker, R.; Chapman, K. L.; Fletcher, A. E.; Patel, S.: Smith, A. J.; Marshall, G. R.; Ryecroft, W.; Matassa, V. G. J. Med. Chem. 1996, 39, 842-849.
-
(1996)
J. Med. Chem.
, vol.39
, pp. 842-849
-
-
Castro, J.L.1
Ball, R.G.2
Broughton, H.B.3
Russell, M.G.N.4
Rathbone, D.5
Watt, A.P.6
Baker, R.7
Chapman, K.L.8
Fletcher, A.E.9
Patel, S.10
Smith, A.J.11
Marshall, G.R.12
Ryecroft, W.13
Matassa, V.G.14
-
21
-
-
0012172138
-
-
Kurzer, F.; Godfrey, L. E. A. Angew. Chem., Int. Ed. Engl. 1963, 2, 459-476.
-
(1963)
Angew. Chem., Int. Ed. Engl.
, vol.2
, pp. 459-476
-
-
Kurzer, F.1
Godfrey, L.E.A.2
-
22
-
-
0042690344
-
-
(a) Svetlik, J.; Hrusovsky, I.; Martvon, A. Coll. Czech. Chem. Commun. 1979, 44, 2982-2986.
-
(1979)
Coll. Czech. Chem. Commun.
, vol.44
, pp. 2982-2986
-
-
Svetlik, J.1
Hrusovsky, I.2
Martvon, A.3
-
25
-
-
0027371231
-
-
Kim, K. S.; Qian, L. Tetrahedron Lett. 1993, 34, 7677-7680. The scope of this reaction has been expanded by Levallet, C.; Lerpiniere, J.; Ko, Y. S. Tetrahedron 1997, 53, 5291-5304.
-
(1993)
Tetrahedron Lett.
, vol.34
, pp. 7677-7680
-
-
Kim, K.S.1
Qian, L.2
-
26
-
-
0030936351
-
-
Kim, K. S.; Qian, L. Tetrahedron Lett. 1993, 34, 7677-7680. The scope of this reaction has been expanded by Levallet, C.; Lerpiniere, J.; Ko, Y. S. Tetrahedron 1997, 53, 5291-5304.
-
(1997)
Tetrahedron
, vol.53
, pp. 5291-5304
-
-
Levallet, C.1
Lerpiniere, J.2
Ko, Y.S.3
-
28
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-
0042189220
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note
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4, filtered, and concentrated under reduced pressure. The resulting residue was purified by silica gel chromatography to give tetrazole 1.
-
-
-
-
29
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0042189221
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note
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max = 60.16°, 3122 reflections (unique), R1 = 0.00493, wR2 = 0.1094, GOF = 1.006.
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31
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84987203063
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For the reaction of N-(pyrrolidine-1-carbothioyl)benzamide, we may have obtained a bis-thiomercury(II) complex. See Richter, R.; Seiler, J.; Beyer, L.; Lindqvist, O.; Andersen, L. Z. Anorg. Allg. Chem. 1985, 522, 171-183.
-
(1985)
Z. Anorg. Allg. Chem.
, vol.522
, pp. 171-183
-
-
Richter, R.1
Seiler, J.2
Beyer, L.3
Lindqvist, O.4
Andersen, L.5
-
34
-
-
0026467126
-
-
(a) Poss, M. A.; Iwanowicz, E.; Reid, J. A.; Lin, J.; Gu, Z. Tetrahedron Lett. 1992, 33, 5933-5936.
-
(1992)
Tetrahedron Lett.
, vol.33
, pp. 5933-5936
-
-
Poss, M.A.1
Iwanowicz, E.2
Reid, J.A.3
Lin, J.4
Gu, Z.5
-
35
-
-
0034629104
-
-
(b) Linton, B. R.; Carr, A. J.; Orner, B. P.; Hamilton, A. D. J. Org. Chem. 2000, 65, 1566-1568.
-
(2000)
J. Org. Chem.
, vol.65
, pp. 1566-1568
-
-
Linton, B.R.1
Carr, A.J.2
Orner, B.P.3
Hamilton, A.D.4
-
36
-
-
0000911184
-
-
Yong, Y. F.; Kowalski, J. A.; Lipton, M. A. J. Org. Chem. 1997, 62, 1540-1542.
-
(1997)
J. Org. Chem.
, vol.62
, pp. 1540-1542
-
-
Yong, Y.F.1
Kowalski, J.A.2
Lipton, M.A.3
-
37
-
-
84981948207
-
-
(a) Scheffold, R.; Saladin, E. Angew. Chem., Int. Ed. Engl. 1972, 11, 229-231.
-
(1972)
Angew. Chem., Int. Ed. Engl.
, vol.11
, pp. 229-231
-
-
Scheffold, R.1
Saladin, E.2
-
38
-
-
84981425825
-
-
(b) Hartke, K.; Rossbach, F.; Radau, M. Justus Liebigs Ann. Chem. 1972, 762, 167-177.
-
(1972)
Justus Liebigs Ann. Chem.
, vol.762
, pp. 167-177
-
-
Hartke, K.1
Rossbach, F.2
Radau, M.3
-
39
-
-
85087999654
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-
note
-
2, which did not give any guanidine product, even after heating to 60°C for 24 h.
-
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40
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0030865140
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-
Avalos, M.; Babiano, R.; Cintas, P.; Duran, C. J.; Higes, F. J.; Jimenez, J. L.; Lopez, I.; Palacios, J. C. Tetrahedron 1997, 53, 14463-14480.
-
(1997)
Tetrahedron
, vol.53
, pp. 14463-14480
-
-
Avalos, M.1
Babiano, R.2
Cintas, P.3
Duran, C.J.4
Higes, F.J.5
Jimenez, J.L.6
Lopez, I.7
Palacios, J.C.8
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