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Bioorganic and Medicinal Chemistry Letters

Volumn 10, Issue 17, 2000, Pages 2041-2044

Phenyloxazoles and phenylthiazoles as benzamide bioisosteres: Synthesis and dopamine receptor binding profiles

(4) Einsiedel, Jürgen a Thomas, Christoph a Hübner, Harald a Gmeiner, Peter a

a UNIVERSITY OF ERLANGEN NUREMBERG (Germany)

Author keywords

[No Author keywords available]

Indexed keywords

BENZAMIDE DERIVATIVE; CLOZAPINE; DOPAMINE RECEPTOR; OXAZOLE DERIVATIVE; THIAZOLE DERIVATIVE;

ALKYLATION; ARTICLE; BINDING AFFINITY; CHIRALITY; CONFORMATIONAL TRANSITION; DERIVATIZATION; DRUG SYNTHESIS; LIGAND BINDING; RECEPTOR BINDING; RECEPTOR BLOCKING;

ANTIPSYCHOTIC AGENTS; BENZAMIDES; HUMANS; OXAZOLES; RECEPTORS, DOPAMINE; STRUCTURE-ACTIVITY RELATIONSHIP; THIAZOLES;

EID: 0034605131 PISSN: 0960894X EISSN: None Source Type: Journal
DOI: 10.1016/S0960-894X(00)00405-4 Document Type: Article

Times cited : (38)

References (33)

1
- 0030768589
- For review: and references cited therein
- (1997) Curr. Pharm. Design , vol.3 , pp. 391
- Wustrow, D.J.¹ Wise, L.D.²

2
- 0030755226
- For review: and references cited therein
- (1997) Curr. Pharm. Design , vol.3 , pp. 355
- Kulagowski, J.J.¹ Patel, S.²

3
- 0025179967
- (1990) Nature , vol.347 , pp. 146
- Sokoloff, P.¹ Giros, P.² Martres, M.-P.³ Bouthenet, M.-L.⁴ Schwartz, J.-C.⁵

4
- 0020030994
- (1982) Gen. Pharmacol. , vol.13 , pp. 185
- O'Connor, S.E.¹ Brown, R.A.²

5
- 8244235137
- (1997) J. Pharmacol. Exp. Ther. , vol.280 , pp. 83
- Schoemaker, H.¹ Claustre, Y.² Fage, D.³ Rouquier, L.⁴ Chergui, K.⁵ Curet, O.⁶ Oblin, A.⁷ Gonon, F.⁸ Carter, C.⁹ Benavides, J.¹⁰ Scatton, B.¹¹

6
- 0029891127
- (1996) Bioorg. Med. Chem. Lett. , vol.6 , pp. 1361
- Glase, S.A.¹ Akunne, H.C.² Heffner, T.G.³ Johnson, S.J.⁴ Kesten, S.R.⁵ Mackenzie, R.G.⁶ Manley, P.J.⁷ Pugsley, T.A.⁸ Wright, J.L.⁹ Wise, L.D.¹⁰

7
- 0031552093
- (1997) Bioorg. Med. Chem. Lett. , vol.7 , pp. 327
- Boyfield, I.¹ Coldwell, M.C.² Hadley, M.S.³ Healy, M.A.M.⁴ Johnson, C.N.⁵ Nash, D.J.⁶ Riley, G.J.⁷ Scott, E.E.⁸ Smith, S.A.⁹ Stemp, G.¹⁰

8
- 0031576837
- (1997) Bioorg. Med. Chem. Lett. , vol.7 , pp. 485
- Bolton, D.¹ Boyfield, I.² Coldwell, M.C.³ Hadley, M.S.⁴ Johns, A.⁵ Johnson, C.N.⁶ Markwell, R.E.⁷ Nash, D.J.⁸ Riley, G.J.⁹ Scott, E.E.¹⁰ Smith, S.A.¹¹ Stemp, G.¹² Wadsworth, H.J.¹³ Watts, E.A.¹⁴

9
- 17344375725
- (1997) J. Med. Chem. , vol.40 , pp. 1
- Thurkauf, A.¹ Yuan, J.² Chen, X.³ He, S.H.⁴ Wasley, J.W.F.⁵ Hutchison, A.⁶ Woodruff, K.H.⁷ Meade, R.⁸ Hoffman, D.C.⁹ Donovan, H.¹⁰ Jones-Hertzog, D.K.¹¹

10
- 0008207132
- (1999) Bioorg. Med. Chem. Lett. , vol.9 , pp. 41
- Thomas, C.¹ Hubner, H.² Gmeiner, P.³

11
- 0025283137
- (1990) J. Med. Chem. , vol.33 , pp. 2305
- Hogberg, T.¹ De Paulis, T.² Johansson, L.³ Kumar, Y.⁴ Hall, H.⁵ Ogren, S.O.⁶

12
- 0030948120
- (1997) J. Med. Chem. , vol.40 , pp. 833
- Nilsson, J.¹ Wikstrom, H.² Smilde, A.³ Glase, S.⁴ Pugsley, T.⁵ Cruciani, G.⁶ Pastor, M.⁷ Clementi, S.⁸

13
- 0015073128
- 1,3-Dichloroacetone (2 eq) was added in 2 portions
- (1971) Arch. Pharm. (Weinheim Ger.) , vol.304 , pp. 425
- Simiti, I.¹ Chindris, E.²

14
- 0028999904
- (1995) J. Med. Chem. , vol.38 , pp. 2251
- Thurkauf, A.¹ Hutchison, A.² Peterson, J.³ Cornfield, L.⁴ Meade, R.⁵ Huston, K.⁶ Harris, K.⁷ Ross, P.C.⁸ Gerber, K.⁹ Ramabhadran, T.V.¹⁰

15
- 84984191293
- (1980) Synthesis , pp. 243
- Cacchi, S.¹ Misiti, D.²

16
- 0008166785
- Eur. Patent 539, 281 A1, 1992
- (1993) Chem. Abstr. , vol.119 , pp. 139085
- Rognan, D.¹ Mann, A.² Wermuth, C.-G.³ Martres, M.-P.⁴ Giros, B.⁵ Sokoloff, P.⁶ Schwartz, J.-C.⁷ Lecomte, J.-M.⁸ Garrido, F.⁹

17
- 0029878138
- (1996) Arch. Pharm.- Pharm. Med. Chem. , vol.329 , pp. 73
- Von der Saal, W.¹ Engh, R.A.² Eichinger, A.³ Gabriel, B.⁴ Kucznierz, R.⁵ Sauer, J.⁶

18
- 84980144059
- (1961) Chem. Ber. , vol.94 , pp. 2887
- Silberg, A.¹ Simiti, I.² Mantsch, H.³

19
- 33947460144
- (1959) J. Am. Chem. Soc. , vol.81 , pp. 4113
- Kornblum, N.¹ Powers, J.W.² Anderson, G.J.³

20
- 0031757775
- (1998) Synthesis , pp. 1491
- Thomas, C.¹ Orecher, F.² Gmeiner, P.³

21
- 0028104847
- (1994) J. Org. Chem. , vol.59 , pp. 6766
- Gmeiner, P.¹ Junge, D.² Kartner, A.³

22
- 0023688489
- (1988) J. Med. Chem. , vol.31 , pp. 1586
- Rosen, T.¹ Chu, D.T.W.² Lico, I.M.³ Fernandes, P.B.⁴ Shen, L.⁵ Borodkin, S.⁶ Pernet, A.G.⁷

23
- 0025854273
- (1991) Tetrahedron , vol.47 , pp. 5161
- Roussi, G.¹ Zhang, J.²

24
- 0003137407
- (1964) Croat. Chem. Acta , vol.36 , pp. 27
- Fles, D.¹ Ghyczy, T.²

25
- 0017408543
- (1977) Chem. Pharm. Bull. , vol.25 , pp. 1911
- Nagai, Y.¹ Uno, H.² Susumu, U.³

26
- 0008248131
- JP 2,169,569, 1990
- (1991) Chem. Abstr. , vol.114 , pp. 6302
- Sugimoto, H.¹ Tsuchiya, Y.² Higure, K.³ Karibe, N.⁴ Iimura, Y.⁵ Sasaki, A.⁶ Yamanishi, Y.⁷ Ogura, H.⁸ Araki, S.⁹

27
- 0000844109
- (1996) J. Org. Chem. , vol.61 , pp. 3849
- Abdel-Magid, A.F.¹ Carson, K.G.² Harris, B.D.³ Maryanoff, C.A.⁴ Shah, R.D.⁵

28
- 0008204805
- Note

29
- 0026695537
- (1992) Mol. Endocrinol. , vol.6 , pp. 920
- Hayes, G.¹ Biden, T.J.² Selbie, L.A.³ Shine, J.⁴

30
- 0026604248
- (1992) Eur. J. Pharmacol. , vol.225 , pp. 331
- Sokoloff, P.¹ Andrieux, M.² Besancon, R.³ Pilon, C.⁴ Martres, M.-P.⁵ Giros, B.⁶ Schwartz, J.-C.⁷

31
- 0029120447
- (1995) J. Neurochem. , vol.65 , pp. 1157
- Agashari, V.¹ Sanyal, S.² Buchwaldt, S.³ Paterson, A.⁴ Jovanovic, V.⁵ Van Tol, H.H.M.⁶

32
- 0038248584
- (2000) J. Med. Chem. , vol.43 , pp. 756
- Hubner, H.¹ Haubmann, C.² Utz, W.³ Gmeiner, P.⁴

33
- 0008169142
- Note

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