Synthesis, modelling, and μ-opioid receptor affinity of N-3(9)-arylpropenyl-N-9(3)-propionyl-3,9-diazabicyclo[3.3.1]nonanes

Farmaco

Volumn 55, Issue 8, 2000, Pages 553-562

  Pinna, G A ^a   Murineddu, G ^a   Curzu, M M ^a   Villa, S ^b   Vianello, P ^b   Borea, P A ^c   Gessi, S ^c   Toma, L ^d   Colombo, D ^b   Cignarella, G ^b  

^a UNIVERSITY OF SASSARI   (Italy)

^b UNIVERSITY OF MILAN   (Italy)

^c Dipartimento di Medicina Clinica e Sperimentale   (Italy)

^d UNIVERSITY OF PAVIA   (Italy)

Author keywords

Affinity; Diazabicyclononanes; Modelling

Indexed keywords

ANALGESIC AGENT; KAPPA OPIATE RECEPTOR; MU OPIATE RECEPTOR; N 3 PROPIONYL N 9 PROPENYL DERIVATIVE; N 3(9H) PROPENYL N 9(3H) PROPIONYL 3,9 DIAZABICYCLO[3.3.1]NONANE DERIVATIVE; PROPIONIC ACID DERIVATIVE; SIGMA OPIATE RECEPTOR; UNCLASSIFIED DRUG;

ANIMAL TISSUE; ARTICLE; BINDING AFFINITY; CONFORMATION; CONTROLLED STUDY; ISOMER; MALE; MOLECULAR MODEL; NONHUMAN; RAT; RECEPTOR AFFINITY; RECEPTOR BINDING; SYNTHESIS;

ANALGESICS; ANIMALS; BICYCLO COMPOUNDS; BRAIN; GUINEA PIGS; MAGNETIC RESONANCE SPECTROSCOPY; MALE; MODELS, MOLECULAR; RATS; RATS, WISTAR; RECEPTORS, OPIOID, MU;

EID: 0034530169     PISSN: 0014827X     EISSN: None     Source Type: Journal    
DOI: 10.1016/S0014-827X(00)00036-7     Document Type: Article

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