메뉴 건너뛰기




Volumn 21, Issue 10, 2000, Pages 376-381

Dynamic mechanisms of non-classical antagonism by competitive AT1 receptor antagonists

Author keywords

[No Author keywords available]

Indexed keywords

ANGIOTENSIN; ANGIOTENSIN 1 RECEPTOR; ANGIOTENSIN 1 RECEPTOR ANTAGONIST; CANDESARTAN; G PROTEIN COUPLED RECEPTOR; LOSARTAN; PARTIAL AGONIST;

EID: 0034306496     PISSN: 01656147     EISSN: None     Source Type: Journal    
DOI: 10.1016/S0165-6147(00)01523-6     Document Type: Review
Times cited : (47)

References (33)
  • 1
    • 0031899432 scopus 로고    scopus 로고
    • The cholecystokinin-B receptor antagonist L-740,093 produces an insurmountable antagonism of CCK-4 stimulated functional response in cells expressing the human CCK-B receptor
    • (1998) Neuropeptides , vol.32 , pp. 157-160
    • Dunlop, J.1
  • 4
    • 0024368819 scopus 로고
    • Unsurmountable antagonism to 5-hydroxytryptamine in rat kidney results from pseudoirreversible inhibition rather than multiple receptors or allosteric receptor modulation
    • (1989) J. Pharmacol. Exp. Ther. , vol.249 , pp. 401-410
    • Bond, R.A.1
  • 5
    • 0033981790 scopus 로고    scopus 로고
    • Pharmacological examination of the neurokinin-1 receptor mediating relaxation of human intralobar pulmonary artery
    • (2000) J. Pharmacol. Exp. Ther. , vol.292 , pp. 319-325
    • Pedersen, K.E.1
  • 7
    • 0024536402 scopus 로고
    • ICI 147,798; a slowly dissociable β adrenoceptor antagonist that causes insurmountable β-1 and surmountable β-2 adrenoceptor antagonism in isolated tissues
    • (1989) J.Pharmacol. Exp. Ther. , vol.248 , pp. 240-248
    • Keith, R.A.1
  • 8
    • 0031037549 scopus 로고    scopus 로고
    • Novel subtype-selective nonpeptide bradykinin receptor antagonists FR167344 and FR173657
    • (1997) Mol. Pharmacol. , vol.51 , pp. 171-176
    • Aramori, I.1
  • 11
    • 0028800752 scopus 로고
    • Elucidation of the insurmountable nature of an angiotensin receptor antagonist, SC-54629
    • (1995) Mol. Pharmacol. , vol.47 , pp. 115-120
    • Olins, G.M.1
  • 13
    • 0027070825 scopus 로고
    • Different types of receptor interaction of peptide and nonpeptide angiotensin II antagonists revealed by receptor binding and functional studies
    • (1992) Mol. Pharmacol. , vol.41 , pp. 1081-1088
    • Wienen, W.1
  • 14
    • 0026510753 scopus 로고
    • Evidence that the apparent complexity of receptor antagonism by angiotensin II analogues is due to a reversible and syntopic action
    • (1992) Br. J. Pharmacol. , vol.106 , pp. 233-241
    • Liu, Y.J.1
  • 15
    • 0018382532 scopus 로고
    • The immediate pressor response to saralasinin man; a test of angiotensin II receptor vacancy
    • (1979) Circ. Res. , vol.44 , pp. 38-44
    • Wallace, J.M.1
  • 16
    • 0019976177 scopus 로고
    • Effect of three angiotensin II antagonists, [Sar1, Thr8]-, [Sar1, Ile8]- and [Sar1, Ala8]angiotensin II on blood pressure and endocrine factors in normal subjects
    • (1982) Eur. J. Clin. Pharmacol. , vol.23 , pp. 7-10
    • Hata, T.1
  • 17
    • 0032230367 scopus 로고    scopus 로고
    • Phosphorylation of the angiotensin II (AT(1A)) receptor carboxyl terminus; a role in receptor endocytosis
    • (1998) Mol. Endocrinol. , vol.12 , pp. 1513-1524
    • Thomas, W.G.1
  • 18
  • 19
    • 0030993594 scopus 로고    scopus 로고
    • Antagonist-stimulated internalization of the G protein-coupled cholecystokinin receptor
    • (1997) Mol. Pharmacol. , vol.51 , pp. 357-362
    • Roettger, B.F.1
  • 21
    • 0032588149 scopus 로고    scopus 로고
    • 1 receptor antagonists on angiotensin II-induced tone in human isolated subcutaneous resistance arteries
    • (1999) Br. J. Pharmacol. , vol.127 , pp. 1876-1882
    • Garcha, R.S.1
  • 23
    • 0027957875 scopus 로고
    • Receptor binding and internalization of a unique biologically active angiotensin II-colloidal gold conjugate; morphological analysis of angiotensin II processing in isolated vascular strips
    • (1994) J. Vasc. Res. , vol.31 , pp. 10-17
    • Anderson, K.M.1    Peach, M.J.2
  • 24
    • 0033622024 scopus 로고    scopus 로고
    • 2+-sensitivity of the contractile apparatus during angiotensin II-induced desensitization in the rabbit femoral artery
    • (2000) Br. J. Pharmacol. , vol.129 , pp. 425-436
    • Ushio-Fukai, M.1
  • 27
    • 0020955681 scopus 로고
    • Desensitization, two-state receptors and pharmacological parameters
    • (1983) J. Theor. Biol. , vol.103 , pp. 137-161
    • Gero, A.1
  • 28
    • 0028237228 scopus 로고
    • Different types of angiotensin II receptor antagonism induced by BIBS 222 in the rat portal vein and rabbit aorta; the influence of receptor reserve
    • (1994) J. Pharmacol. Exp. Ther. , vol.269 , pp. 509-514
    • Zhang, J.S.1
  • 32
    • 0033012299 scopus 로고    scopus 로고
    • Contractile effects by intracellular angiotensin II via receptors with a distinct pharmacological profile in rat aorta
    • (1999) Br.J. Pharmacol. , vol.126 , pp. 1133-1138
    • Brailoiu, E.1
  • 33
    • 0034723193 scopus 로고    scopus 로고
    • Agonist-induced phosphorylation of the angiotensin II (AT(1A)) receptor requires generation of a conformation that is distinct from the inositol phosphate-signaling state
    • (2000) J. Biol. Chem. , vol.275 , pp. 2893-2900
    • Thomas, W.G.1


* 이 정보는 Elsevier사의 SCOPUS DB에서 KISTI가 분석하여 추출한 것입니다.