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Volumn 129, Issue 4, 2000, Pages 820-821

Agonist binding to G-protein coupled receptors

Author keywords

Agonist binding; G protein coupled receptors; Receptor activation; Receptor theory

Indexed keywords

BETA 2 ADRENERGIC RECEPTOR; G PROTEIN COUPLED RECEPTOR; MUTANT PROTEIN; SODIUM ION;

EID: 0034116151     PISSN: 00071188     EISSN: None     Source Type: Journal    
DOI: 10.1038/sj.bjp.0702991     Document Type: Letter
Times cited : (5)

References (16)
  • 2
    • 0023893314 scopus 로고
    • Site directed mutagenesis and continuous expression of the human β-adrenergic receptor
    • Chung, F., Wang, C., Potter, P.C., Venter, J.C. & Fraser, C.M. (1988). Site directed mutagenesis and continuous expression of the human β-adrenergic receptor. J. Biol. Chem., 263, 4052-4055.
    • (1988) J. Biol. Chem. , vol.263 , pp. 4052-4055
    • Chung, F.1    Wang, C.2    Potter, P.C.3    Venter, J.C.4    Fraser, C.M.5
  • 3
    • 0032199006 scopus 로고    scopus 로고
    • Binding, gating and efficacy: The interpretation of structure-activity relationships for agonists and of the effects of mutating receptors
    • Colquhoun, D. (1998). Binding, gating and efficacy: the interpretation of structure-activity relationships for agonists and of the effects of mutating receptors. Br. J. Pharmacol., 125, 924-947.
    • (1998) Br. J. Pharmacol. , vol.125 , pp. 924-947
    • Colquhoun, D.1
  • 4
    • 0024847889 scopus 로고
    • Site directed mutagenesis of m1 muscarinic acetylcholine receptors: Conserved aspartic acids play important roles in receptor function
    • Fraser, C.M., Wang, C., Robinson, D.A., Gocayne, J.D. & Venter, J.C. (1990). Site directed mutagenesis of m1 muscarinic acetylcholine receptors: conserved aspartic acids play important roles in receptor function. Mol. Pharmacol., 36, 840-847.
    • (1990) Mol. Pharmacol. , vol.36 , pp. 840-847
    • Fraser, C.M.1    Wang, C.2    Robinson, D.A.3    Gocayne, J.D.4    Venter, J.C.5
  • 5
    • 0025642404 scopus 로고
    • An aspartate conserved among G-protein coupled receptors confers allosteric regulation of α2 adrenergic receptors by sodium ions
    • Horstman, D.A., Brandon, S., Wilson, A.L., Guyer, C.A., Crago, E.J. & Limbird, L.E. (1990). An aspartate conserved among G-protein coupled receptors confers allosteric regulation of α2 adrenergic receptors by sodium ions. J. Biol. Chem., 265, 21590-21595.
    • (1990) J. Biol. Chem. , vol.265 , pp. 21590-21595
    • Horstman, D.A.1    Brandon, S.2    Wilson, A.L.3    Guyer, C.A.4    Crago, E.J.5    Limbird, L.E.6
  • 6
    • 0027297275 scopus 로고
    • Constitutive activity of receptors coupled to guanine nucleotide regulatory proteins
    • Lefkowitz, R.J., Cotecchia, S., Samama, P. & Costa, T. (1993). Constitutive activity of receptors coupled to guanine nucleotide regulatory proteins. Trends Pharmacol. Sci., 14, 303-307.
    • (1993) Trends Pharmacol. Sci. , vol.14 , pp. 303-307
    • Lefkowitz, R.J.1    Cotecchia, S.2    Samama, P.3    Costa, T.4
  • 7
    • 0025863465 scopus 로고
    • Pivotal role for aspartate 80 in the regulation of dopamine D2 receptor affinity for drugs and inhibition of adenylyl cyclase
    • Neve, K.A., Cox, B.A., Henningsen, R.A., Spanoyannis, A. & Neve, R.L. (1991). Pivotal role for aspartate 80 in the regulation of dopamine D2 receptor affinity for drugs and inhibition of adenylyl cyclase. Mol. Pharmacol., 39, 733-739.
    • (1991) Mol. Pharmacol. , vol.39 , pp. 733-739
    • Neve, K.A.1    Cox, B.A.2    Henningsen, R.A.3    Spanoyannis, A.4    Neve, R.L.5
  • 9
    • 0023740863 scopus 로고
    • Conserved aspartic acid residues 79 and 113 of the β-adrenergic receptor have different roles in receptor function
    • Strader, C.D., Sigal, I.S., Candelore, M.R., Rands, E., Hill, W.S. & Dixon, R.A.F. (1988). Conserved aspartic acid residues 79 and 113 of the β-adrenergic receptor have different roles in receptor function. J. Biol. Chem., 263, 10267-10271.
    • (1988) J. Biol. Chem. , vol.263 , pp. 10267-10271
    • Strader, C.D.1    Sigal, I.S.2    Candelore, M.R.3    Rands, E.4    Hill, W.S.5    Dixon, R.A.F.6
  • 11
    • 0030176923 scopus 로고    scopus 로고
    • The energetics of ligand binding at catecholamine receptors
    • Strange, P.G. (1996). The energetics of ligand binding at catecholamine receptors. Trends. Pharmacol. Sci., 17, 238-244.
    • (1996) Trends. Pharmacol. Sci. , vol.17 , pp. 238-244
    • Strange, P.G.1
  • 12
    • 0032033681 scopus 로고    scopus 로고
    • Three state and two state models
    • Strange P.G. (1998) Three state and two state models. Trends. Pharmacol. Sci., 19, 85-86.
    • (1998) Trends. Pharmacol. Sci. , vol.19 , pp. 85-86
    • Strange, P.G.1
  • 13
    • 0032804984 scopus 로고    scopus 로고
    • G-protein coupled receptors: Conformations and states
    • Strange, P.G. (1999). G-protein coupled receptors: conformations and states. Biochem. Pharmacol., 58, 1081-1088.
    • (1999) Biochem. Pharmacol. , vol.58 , pp. 1081-1088
    • Strange, P.G.1
  • 14
    • 0029919840 scopus 로고    scopus 로고
    • Molecular architecture of G-protein coupled receptors
    • Van Rhee, A.M. & Jacobsen, K.A. (1996). Molecular architecture of G-protein coupled receptors. Drug Dev. Res., 37, 1-38.
    • (1996) Drug Dev. Res. , vol.37 , pp. 1-38
    • Van Rhee, A.M.1    Jacobsen, K.A.2
  • 15
    • 0026006986 scopus 로고
    • 2A adrenergic receptors: Identification of amino acids involved in ligand binding and receptor activation by agonist
    • 2A adrenergic receptors: identification of amino acids involved in ligand binding and receptor activation by agonist. Mol. Pharmacol., 40, 168-179.
    • (1991) Mol. Pharmacol. , vol.40 , pp. 168-179
    • Wang, C.1    Buck, M.A.2    Fraser, C.M.3
  • 16
    • 0027175853 scopus 로고
    • Site directed mutagenesis of the serotonin 5HT2 receptor: Identification of amino acids necessary for ligand binding and receptor activation
    • Wang, C., Gallagher, T.K. & Shih, J.C. (1993). Site directed mutagenesis of the serotonin 5HT2 receptor: identification of amino acids necessary for ligand binding and receptor activation. Mol. Pharmacol., 43, 931-940.
    • (1993) Mol. Pharmacol. , vol.43 , pp. 931-940
    • Wang, C.1    Gallagher, T.K.2    Shih, J.C.3


* 이 정보는 Elsevier사의 SCOPUS DB에서 KISTI가 분석하여 추출한 것입니다.