Transformation of the sydnone ring into oxadiazolinones. A convenient one-pot synthesis of 3-aryl-5-methyl-1,3,4-oxadiazolin-2-ones from 3- arylsydnones and their antimicrobial activity

Farmaco

Volumn 55, Issue 1, 2000, Pages 65-67

  Mallur, Shanta G ^a   Badami, Bharati V ^a  

^a KARNATAK UNIVERSITY   (India)

Author keywords

Antimicrobial activity; Oxadiazolinones; Sydnone ring

Indexed keywords

ANTIINFECTIVE AGENT; OXADIAZOLE DERIVATIVE; OXADIAZOLIN 2 ONE DERIVATIVE; SYDNONE DERIVATIVE; UNCLASSIFIED DRUG;

ANTIMICROBIAL ACTIVITY; ARTICLE; ASPERGILLUS NIGER; DRUG STRUCTURE; DRUG SYNTHESIS; HYPHOMYCETES; INDIA; NONHUMAN; PSEUDOMONAS AERUGINOSA;

ANTI-INFECTIVE AGENTS; MICROBIAL SENSITIVITY TESTS; OXADIAZOLES; SYDNONES;

EID: 0034112044     PISSN: 0014827X     EISSN: None     Source Type: Journal    
DOI: 10.1016/S0014-827X(99)00103-2     Document Type: Article

References (7)

1. Otha M., Kato H. Snyder J.P. Nonbenzenoid Aromatics. 1969;117-170 Academic Press, New York.
2. Badami B.V., Puranik G.S. Reactions of sydnones. Part I. Indian J. Chem. 12:1974;671-673.
3. Hiremath U.S., Yelamaggad C.V., Badami B.V. 1,3-Dipolar cycloadducts of sydnones. Indian J. Heterocycl. Chem. 5:1995;19-22.
4. Rupe H., Gebhardt H. Ueber unsymmetrische Phenyl-hydrazin Derivate. Berichte. 32:1899;10-17.
5. Kametani T., Sota K., Shio M. Studies on the syntheses of azole derivatives. J. Heterocycl. Chem. 7:1970;821-829.
6. Ugarkar B.G., Badami B.V., Puranik G.S., Bhat K.G.S. Synthesis and central nervous system depression properties of disubstituted sydnones. Arch. Pharm. (Weinheim). 311:1978;109-114.
7. Turnbull K. Bromination of sydnones. J. Heterocycl. Chem. 22:1985;965-968.