Single-cell recombinant pharmacology: Bovine α(1a)-adrenoceptors in rat-1 fibroblasts release intracellular Ca2+, display subtype- characteristic agonism and antagonism, and exhibit an antagonist-reversible inverse concentration-response phase

Journal of Pharmacology and Experimental Therapeutics

Volumn 293, Issue 3, 2000, Pages 887-895

  Pediani, John Daniel ^a,b   Mackenzie, Janet Fraser ^a   Heeley, Robert Paul ^a   Daly, Craig James ^a   McGrath, John Christie ^a  

^a UNIVERSITY OF GLASGOW   (United Kingdom)

^b UNIVERSITY OF GLASGOW   (United Kingdom)

Author keywords

[No Author keywords available]

Indexed keywords

2 [[2 (2,6 DIMETHOXYPHENOXY)ETHYL]AMINOMETHYL] 1,4 BENZODIOXAN; 8 [2 [4 (2 METHOXYPHENYL) 1 PIPERAZINYL]ETHYL] 8 AZASPIRO[4.5]DECANE 7,9 DIONE; ALPHA 1 ADRENERGIC RECEPTOR; CALCIUM; N [5 (4,5 DIHYDRO 1H IMIDAZOL 2 YL) 5,6,7,8 TETRAHYDRO 2 HYDROXY 1 NAPHTHYL]METHANESULFONAMIDE; PRAZOSIN;

ANIMAL CELL; ARTICLE; CALCIUM CELL LEVEL; CALCIUM SIGNALING; CALCIUM TRANSPORT; CATTLE; COMPETITIVE INHIBITION; CONTROLLED STUDY; DRUG POTENCY; DRUG RECEPTOR BINDING; FIBROBLAST; NONHUMAN; PRIORITY JOURNAL; RAT; RECEPTOR AFFINITY;

ANIMALS; CALCIUM SIGNALING; CATTLE; DIOXANES; DOSE-RESPONSE RELATIONSHIP, DRUG; IMIDAZOLES; PHENYLALANINE; PIPERAZINES; PRAZOSIN; RATS; RECEPTORS, ADRENERGIC, ALPHA-1; RECOMBINANT PROTEINS; REVERSE TRANSCRIPTASE POLYMERASE CHAIN REACTION; TETRAHYDRONAPHTHALENES;

EID: 0034089652     PISSN: 00223565     EISSN: None     Source Type: Journal    
DOI: None     Document Type: Article

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