-
1
-
-
0025609651
-
-
(a) and references cited therein
-
(a) Salvetti, A. Drugs 1990, 40, 800, and references cited therein.
-
(1990)
Drugs
, vol.40
, pp. 800
-
-
Salvetti, A.1
-
3
-
-
0342946937
-
-
(a) Japanese Patent, Jpn Kokai Tokkyo Koho JP 63,63,646, 1988
-
(a) Miyazawa, Y.; Oishi, N.; Maehara, K. Japanese Patent, Jpn Kokai Tokkyo Koho JP 63,63,646, 1988.
-
-
-
Miyazawa, Y.1
Oishi, N.2
Maehara, K.3
-
4
-
-
0343818056
-
-
(b) Japanese Patent, Jpn Kokai Tokkyo Koho JP 63,145,256, 1988
-
(b) Miyazawa, Y.; Oishi, N.; Maehara, K. Japanese Patent, Jpn Kokai Tokkyo Koho JP 63,145,256, 1988.
-
-
-
Miyazawa, Y.1
Oishi, N.2
Maehara, K.3
-
5
-
-
0343382391
-
-
(c) Eur. Pat. Appl. EP 310,012, 1989
-
(c) Keller, R.; Mueller, W. Eur. Pat. Appl. EP 310,012, 1989.
-
-
-
Keller, R.1
Mueller, W.2
-
6
-
-
0342946935
-
-
(d) US Patent 5,552,317, 1996
-
(d) Houng, J.; Hsieh, C. US Patent 5,552,317, 1996.
-
-
-
Houng, J.1
Hsieh, C.2
-
7
-
-
0027999179
-
-
(e)
-
(e) Pugniere, M.; Domergue, N.; Castro, B.; Previero, A. Chirality 1994, 6, 472
-
(1994)
Chirality
, vol.6
, pp. 472
-
-
Pugniere, M.1
Domergue, N.2
Castro, B.3
Previero, A.4
-
8
-
-
0027938138
-
-
(f)
-
(f) Chen, S. T.; Huang, W. H.; Wang, K. T. Chirality 1994, 6, 572.
-
(1994)
Chirality
, vol.6
, pp. 572
-
-
Chen, S.T.1
Huang, W.H.2
Wang, K.T.3
-
9
-
-
0025965448
-
-
(a)
-
(a) Bradshaw, C. W.; Wang, C. H.; Hummel, W.; Kula, M. R. Bioorg. Chem. 1991, 19, 29.
-
(1991)
Bioorg. Chem.
, vol.19
, pp. 29
-
-
Bradshaw, C.W.1
Wang, C.H.2
Hummel, W.3
Kula, M.R.4
-
10
-
-
0025144976
-
-
(b)
-
(b) Asano, Y.; Yamada, A.; Kato, Y.; Yamaguchi, K.; Hibino, Y.; Hirai, K.; Kondo, K. J. Org. Chem. 1990, 55, 5567.
-
(1990)
J. Org. Chem.
, vol.55
, pp. 5567
-
-
Asano, Y.1
Yamada, A.2
Kato, Y.3
Yamaguchi, K.4
Hibino, Y.5
Hirai, K.6
Kondo, K.7
-
11
-
-
0342946929
-
-
(c) Japanese Patent, Jpn Kokai Tokkyo Koho JP 01,47,386, 1989
-
(c) Asano, Y.; Iwasaki, G.; Kondo, S. Japanese Patent, Jpn Kokai Tokkyo Koho JP 01,47,386, 1989.
-
-
-
Asano, Y.1
Iwasaki, G.2
Kondo, S.3
-
12
-
-
0343818053
-
-
(d) Japanese Patent, Jpn Kokai Tokkyo Koho JP 03,112,409, 1991
-
(d) Fujikawa, K.; Sato, H.; Yonehara, T.; Miyata, A. Japanese Patent, Jpn Kokai Tokkyo Koho JP 03,112,409, 1991.
-
-
-
Fujikawa, K.1
Sato, H.2
Yonehara, T.3
Miyata, A.4
-
13
-
-
0037827003
-
-
(e)
-
(e) Senuma, M.; Nakamichi, K.; Nabe, K.; Nishimoto, S.; Tosa, T. Appl. Biochem. Biotechnol. 1989, 22, 141.
-
(1989)
Appl. Biochem. Biotechnol.
, vol.22
, pp. 141
-
-
Senuma, M.1
Nakamichi, K.2
Nabe, K.3
Nishimoto, S.4
Tosa, T.5
-
14
-
-
0343382388
-
-
(f) Japanese Patent, Jpn Kokai Tokkyo Koho JP 03,112,491, 1991
-
(f) Fujikawa, K.; Sato, H.; Yonehara, T.; Miyata, A. Japanese Patent, Jpn Kokai Tokkyo Koho JP 03,112,491, 1991.
-
-
-
Fujikawa, K.1
Sato, H.2
Yonehara, T.3
Miyata, A.4
-
15
-
-
0342512778
-
-
(g) Japanese Patent, Jpn Kokai Tokkyo Koho JP 02,278,585, 1990
-
(g) Nakayama, K.; Ozawa, T. Japanese Patent, Jpn Kokai Tokkyo Koho JP 02,278,585, 1990.
-
-
-
Nakayama, K.1
Ozawa, T.2
-
16
-
-
0342946926
-
-
(h) Japanese Patent, Jpn Kokai Tokkyo Koho JP 02,119,796, 1990
-
(h) Nakayama, K.; Ozawa, T. Japanese Patent, Jpn Kokai Tokkyo Koho JP 02,119,796, 1990.
-
-
-
Nakayama, K.1
Ozawa, T.2
-
17
-
-
0342946925
-
-
(i) Japanese Patent, Jpn Kokai Tokkyo Koho JP 63,273,498, 1988
-
(i) Nabe, K.; Nishida, Y.; Nakamichi, K.; Nishimoto, S. Japanese Patent, Jpn Kokai Tokkyo Koho JP 63,273,498, 1988.
-
-
-
Nabe, K.1
Nishida, Y.2
Nakamichi, K.3
Nishimoto, S.4
-
18
-
-
0342946923
-
-
(j) Japanese Patent, Jpn Kokai Tokkyo Koho JP 06,343,483, 1994
-
(j) Mihara, Y.; Onishi, I. Japanese Patent, Jpn Kokai Tokkyo Koho JP 06,343,483, 1994.
-
-
-
Mihara, Y.1
Onishi, I.2
-
19
-
-
0026548503
-
-
(k)
-
(k) Syldatk, C.; Lehmensiek, V.; Ulrichs, G.; Bilitewski, U.; Krohn, K.; Hoeke, H.; Wagner, F. Biotechnol. Lett. 1992, 14, 99.
-
(1992)
Biotechnol. Lett.
, vol.14
, pp. 99
-
-
Syldatk, C.1
Lehmensiek, V.2
Ulrichs, G.3
Bilitewski, U.4
Krohn, K.5
Hoeke, H.6
Wagner, F.7
-
20
-
-
0026187641
-
-
(l)
-
(l) Fotheringham, I. G.; Kidman, G. E.; McArthur, B. S.; Robinson, L. E.; Scollar, M. P. Biotechnol. Prog. 1991, 7, 380.
-
(1991)
Biotechnol. Prog.
, vol.7
, pp. 380
-
-
Fotheringham, I.G.1
Kidman, G.E.2
McArthur, B.S.3
Robinson, L.E.4
Scollar, M.P.5
-
21
-
-
33845278130
-
-
(a)
-
(a) Williams, R. M.; Sinclair, P. J.; Zhai, D.; Chen, D. J. Am. Chem. Soc. 1988, 110, 1547.
-
(1988)
J. Am. Chem. Soc.
, vol.110
, pp. 1547
-
-
Williams, R.M.1
Sinclair, P.J.2
Zhai, D.3
Chen, D.4
-
22
-
-
0001493681
-
-
(b)
-
(b) Zhai, D.; Zhai, W.; Williams, R. M. J. Am. Chem. Soc. 1988, 110, 2501.
-
(1988)
J. Am. Chem. Soc.
, vol.110
, pp. 2501
-
-
Zhai, D.1
Zhai, W.2
Williams, R.M.3
-
23
-
-
37049068308
-
-
(c)
-
(c) Gasanov, R. G.; II'inskaya, L. V.; Misharin, M. A.; Maleev, V. I.; Raevski, N. I.; Ikonnikov, N. S.; Orlova, S. A.; Kuzmina, N. A.; Belokon, Y. N. J. Chem. Soc., Perkin Trans. 1 1994, 3343.
-
(1994)
J. Chem. Soc., Perkin Trans.
, vol.1
, pp. 3343
-
-
Gasanov, R.G.1
Ii'Inskaya, L.V.2
Misharin, M.A.3
Maleev, V.I.4
Raevski, N.I.5
Ikonnikov, N.S.6
Orlova, S.A.7
Kuzmina, N.A.8
Belokon, Y.N.9
-
24
-
-
0001125476
-
-
(d)
-
(d) Belokon, Y. N.; Sagyan, A. S.; Djamgaryan, S. M.; Bakhmutov, V. I.; Belikov, V. M. Tetrahedron 1988, 44, 5507.
-
(1988)
Tetrahedron
, vol.44
, pp. 5507
-
-
Belokon, Y.N.1
Sagyan, A.S.2
Djamgaryan, S.M.3
Bakhmutov, V.I.4
Belikov, V.M.5
-
25
-
-
0000510339
-
-
(a)
-
(a) Cesarotti, E.; Chiesa, A.; D'Alfonso, G. Tetrahedron Lett. 1982, 23, 2995.
-
(1982)
Tetrahedron Lett.
, vol.23
, pp. 2995
-
-
Cesarotti, E.1
Chiesa, A.2
D'Alfonso, G.3
-
27
-
-
0001838846
-
-
(c)
-
(c) Döbler, C.; Kreuzfeld, H. J.; Pracejus, H. J. Organometal. Chem. 1988, 344, 89.
-
(1988)
J. Organometal. Chem.
, vol.344
, pp. 89
-
-
Döbler, C.1
Kreuzfeld, H.J.2
Pracejus, H.3
-
28
-
-
0000366174
-
-
(d)
-
(d) Krause, H. W.; Foken, H.; Pracejus, H. New J. Chem. 1989, 13, 615.
-
(1989)
New J. Chem.
, vol.13
, pp. 615
-
-
Krause, H.W.1
Foken, H.2
Pracejus, H.3
-
29
-
-
0028897511
-
-
(e)
-
(e) Döbler, C.; Schimidt, U.; Krause, H. W.; Kreuzfeld, H. J.; Michalik, M. Tetrahedron: Asymmetry 1995, 6, 385.
-
(1995)
Tetrahedron: Asymmetry
, vol.6
, pp. 385
-
-
Döbler, C.1
Schimidt, U.2
Krause, H.W.3
Kreuzfeld, H.J.4
Michalik, M.5
-
30
-
-
0029987157
-
-
(f)
-
(f) Kreuzfeld, H. J.; Schimidt, U.; Döbler, C.; Krause, H. W. Tetrahedron: Asymmetry 1996, 7, 1011.
-
(1996)
Tetrahedron: Asymmetry
, vol.7
, pp. 1011
-
-
Kreuzfeld, H.J.1
Schimidt, U.2
Döbler, C.3
Krause, H.W.4
-
32
-
-
0003151014
-
-
(a)
-
(a) Mi, A. Q.; Lou, R. L.; Jiang, Y. Z.; Deng, J. G.; Qin, Y.; Fu, F. M.; Li, Z.; Hu, W. H.; Chan, A. S. C. Synlett 1998, 847.
-
(1998)
Synlett
, pp. 847
-
-
Mi, A.Q.1
Lou, R.L.2
Jiang, Y.Z.3
Deng, J.G.4
Qin, Y.5
Fu, F.M.6
Li, Z.7
Hu, W.H.8
Chan, A.S.C.9
-
33
-
-
0342512771
-
-
(b) Chinese Patent Application No. 97107608.1, July 24, 1997
-
(b) Mi, A. Q.; Lou, R. L.; Qin, Y.; Jiang, Y. Z.; Hu, W. H.; Chan, A. S. C. Chinese Patent Application No. 97107608.1, July 24, 1997.
-
-
-
Mi, A.Q.1
Lou, R.L.2
Qin, Y.3
Jiang, Y.Z.4
Hu, W.H.5
Chan, A.S.C.6
-
34
-
-
0002901254
-
-
(a) Morrison, J. D., Ed.; Academic Press: New York Chapter 3
-
(a) Koenig, K. E. In Asymmetric Synthesis; Morrison, J. D., Ed.; Academic Press: New York, 1985; Vol. 5, Chapter 3.
-
(1985)
In Asymmetric Synthesis
, vol.5
-
-
Koenig, K.E.1
-
38
-
-
0000489118
-
-
2O in the presence of HOAc. See
-
2O in the presence of HOAc. See: Burk, M. J.; Casy, G.; Johnson, N. B. J. Org. Chem. 1998, 63, 6084.
-
(1998)
J. Org. Chem.
, vol.63
, pp. 6084
-
-
Burk, M.J.1
Casy, G.2
Johnson, N.B.3
-
39
-
-
0023205265
-
-
(b) All other (Z)-2-aminocrotonates 3b-g were prepared by condensation of α-keto ester 4a or the corresponding α-keto acid 4b with benzamide or appropriate carbamates, following the procedure outlined by Melillo et al. with a little modification
-
(b) All other (Z)-2-aminocrotonates 3b-g were prepared by condensation of α-keto ester 4a or the corresponding α-keto acid 4b with benzamide or appropriate carbamates, following the procedure outlined by Melillo et al. with a little modification: Melillo, D. G.; Larsen, R. D.; Mathre, D. J.; Shukis, W. F.; Wood, A. W.; Colleluori, J. R. J. Org. Chem. 1987, 52, 5143.
-
(1987)
J. Org. Chem.
, vol.52
, pp. 5143
-
-
Melillo, D.G.1
Larsen, R.D.2
Mathre, D.J.3
Shukis, W.F.4
Wood, A.W.5
Colleluori, J.R.6
-
40
-
-
0026693049
-
-
Kubota, H.; Nunami, K.; Hayashi, K.; Hashimoto, Y.; Ogiku, N.; Matsuoka, Y.; Ishida, R. Chem. Pharm. Bull. Jpn 1992, 40, 1619.
-
(1992)
Chem. Pharm. Bull. Jpn
, vol.40
, pp. 1619
-
-
Kubota, H.1
Nunami, K.2
Hayashi, K.3
Hashimoto, Y.4
Ogiku, N.5
Matsuoka, Y.6
Ishida, R.7
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