Synthesis, antiplatelet activity and comparative molecular field analysis of substituted 2-amino-4H-pyrido[1,2-a]pyrimidin-4-ones, their congeners and isosteric analogues

Bioorganic and Medicinal Chemistry

Volumn 8, Issue 4, 2000, Pages 751-768

  Roma, Giorgio ^a   Cinone, Nunzia ^b   Di Braccio, Mario ^a   Grossi, Giancarlo ^a   Leoncini, Giuliana ^a   Signorello, Maria Grazia ^a   Carotti, Angelo ^b  

^a UNIVERSITY OF GENOA   (Italy)

^b UNIVERSITY OF BARI   (Italy)

Author keywords

[No Author keywords available]

Indexed keywords

2 (1 PIPERAZINYL) 4H PYRIDO[1,2A]PYRIMIDIN 4 DERIVATIVE; PYRIMIDINE DERIVATIVE; UNCLASSIFIED DRUG;

ARTICLE; DRUG STRUCTURE; ELECTRICITY; MOLECULAR MODEL; QUANTITATIVE STRUCTURE ACTIVITY RELATION; STEREOCHEMISTRY; SYNTHESIS; THROMBOCYTE AGGREGATION; THROMBOCYTE AGGREGATION INHIBITION;

HUMANS; MAGNETIC RESONANCE SPECTROSCOPY; MODELS, MOLECULAR; PLATELET AGGREGATION INHIBITORS; PYRIMIDINONES; STRUCTURE-ACTIVITY RELATIONSHIP;

EID: 0034070030     PISSN: 09680896     EISSN: None     Source Type: Journal    
DOI: 10.1016/S0968-0896(00)00010-9     Document Type: Article

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